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Found 8 with Last Name = 'hradilek' and Initial = 'm'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM520(1,3-thiazol-5-ylmethyl N-[(2S,3S,5S)-3-hydroxy-5-[...)
Affinity DataKi:  0.0150nMAssay Description:Tested for inhibitor binding of wild-type HIV PRMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50581791(CHEMBL5073221)
Affinity DataKi:  0.0320nMAssay Description:Inhibition of wild type HIV-1 protease assessed as initial inhibition constant by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50143837((S)-4-[(S)-2-((2R,3S)-3-Benzyloxycarbonylamino-2-h...)
Affinity DataKi:  0.110nMAssay Description:Tested for inhibitor binding of Val82Ala mutant of HIV PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM520(1,3-thiazol-5-ylmethyl N-[(2S,3S,5S)-3-hydroxy-5-[...)
Affinity DataKi:  0.120nMAssay Description:Tested for inhibitor binding of D25N/V82A mutant of HIV PRMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50143837((S)-4-[(S)-2-((2R,3S)-3-Benzyloxycarbonylamino-2-h...)
Affinity DataKi:  0.180nMAssay Description:Tested for inhibitor binding of wild-type HIV PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetCathepsin E(Homo sapiens (Human))
Institute Of Organic Chemistry And Biochemistry Of The Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50581791(CHEMBL5073221)
Affinity DataKi:  440nMAssay Description:Inhibition of human cathepsin E assessed as inhibition constant using ACC-GKPILFFRILK-(DNP)-(dR)-NH2 as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Institute Of Organic Chemistry And Biochemistry Of The Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50581791(CHEMBL5073221)
Affinity DataKi:  620nMAssay Description:Inhibition of human cathepsin D assessed as inhibition constant using ACC-GKPILFFRILK-(DNP)-(dR)-NH2 as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Institute Of Organic Chemistry And Biochemistry Of The Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50581791(CHEMBL5073221)
Affinity DataKi:  1.90E+4nMAssay Description:Inhibition of human renin assessed as inhibition constant using H-R-E(EDANS)-1HPFHLVIHT-K(DABCYL)-R-OH as susbtrate by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed