TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 0.121nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 0.394nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 4.30nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 78nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 131nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 131nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 630nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 857nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 1.01E+3nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 1.36E+3nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: 1.77E+3nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]paroxetine binding to serotonin transport sites in rat frontal cortex membranes.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataIC50: 0.0430nMAssay Description:Inhibition of [125I]RTI-55 binding to dopamine transport sites in rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Very late antigen 4/vascular cell adhesion molecule 1 interaction in ELISAMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataIC50: 0.115nMAssay Description:Inhibition of [125I]RTI-55 binding to dopamine transport sites in rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Inhibition of Very late antigen 4/vascular cell adhesion molecule 1 interaction in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Inhibition of Very late antigen 4/vascular cell adhesion molecule 1 interaction in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.260nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataIC50: 0.280nMAssay Description:Inhibition of [125I]RTI-55 binding to dopamine transport sites in rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 0.290nMAssay Description:Inhibition of Very late antigen 4/vascular cell adhesion molecule 1 interaction in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in RamosMore data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.370nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.370nMAssay Description:Antagonistic activity against VLA-4 (derived from ramos cells) binding to recombinant human VCAM by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.420nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.460nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.470nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in RamosMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.520nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.530nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.550nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.610nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in RamosMore data for this Ligand-Target Pair
Affinity DataIC50: 0.640nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.740nMAssay Description:Antagonistic activity against VLA-4 (derived from ramos cells) binding to recombinant human VCAM by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.75nMAssay Description:Antagonistic activity against VLA-4 (derived from ramos cells) binding to recombinant human VCAM by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in RamosMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibitory binding concentration determined against VCAM/VLA-4 in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.820nMAssay Description:Inhibition of human VCAM and Ramos cell VLA-4 interactionMore data for this Ligand-Target Pair