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Found 108 with Last Name = 'hupe' and Initial = 'l'
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043804(5-(2-Amino-3-phenyl-propionylamino)-3-isobutyl-7-m...)
Affinity DataKi:  13nMAssay Description:Inhibition of recombinant full length stromelysin (FLS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043804(5-(2-Amino-3-phenyl-propionylamino)-3-isobutyl-7-m...)
Affinity DataKi:  15nMAssay Description:Inhibition of recombinant stromelysin catalytic domain (SCD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043807((S)-2-Benzyloxycarbonylamino-3-(1H-indol-3-yl)-pro...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of recombinant stromelysin catalytic domain (SCD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043807((S)-2-Benzyloxycarbonylamino-3-(1H-indol-3-yl)-pro...)
Affinity DataKi:  6.30E+3nMAssay Description:Inhibition of recombinant full length stromelysin (FLS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043801((S)-2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-p...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of recombinant stromelysin catalytic domain (SCD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043805((S)-2-Benzyloxycarbonylamino-3-(1H-indol-3-yl)-pro...)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of recombinant stromelysin catalytic domain (SCD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043803((S)-2-Benzyloxycarbonylamino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of recombinant full length stromelysin (FLS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043803((S)-2-Benzyloxycarbonylamino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of recombinant stromelysin catalytic domain (SCD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043813((S)-2-tert-Butoxycarbonylamino-3-(1-formyl-1H-indo...)
Affinity DataKi:  2.80E+4nMAssay Description:Inhibition of recombinant stromelysin catalytic domain (SCD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043796((S)-2-Benzyloxycarbonylamino-3-phenyl-propionic ac...)
Affinity DataKi:  3.30E+4nMAssay Description:Inhibition of recombinant stromelysin catalytic domain (SCD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043806((S)-2-tert-Butoxycarbonylamino-3-[1-(2,4,6-trimeth...)
Affinity DataKi:  5.20E+4nMAssay Description:Inhibition of recombinant stromelysin catalytic domain (SCD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043809((R)-2-Benzyloxycarbonylamino-3-(1H-indol-3-yl)-pro...)
Affinity DataKi:  7.10E+4nMAssay Description:Inhibition of recombinant stromelysin catalytic domain (SCD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043796((S)-2-Benzyloxycarbonylamino-3-phenyl-propionic ac...)
Affinity DataKi:  8.30E+4nMAssay Description:Inhibition of recombinant full length stromelysin (FLS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043812((S)-2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-p...)
Affinity DataKi:  8.40E+4nMAssay Description:Inhibition of recombinant stromelysin catalytic domain (SCD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043800((S)-2-((E)-3-Furan-2-yl-acryloylamino)-3-(1H-indol...)
Affinity DataKi:  1.20E+5nMAssay Description:Inhibition of recombinant stromelysin catalytic domain (SCD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043809((R)-2-Benzyloxycarbonylamino-3-(1H-indol-3-yl)-pro...)
Affinity DataKi:  2.41E+5nMAssay Description:Inhibition of recombinant full length stromelysin (FLS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043797((R)-2-Benzyloxycarbonylamino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  3.56E+5nMAssay Description:Inhibition of recombinant stromelysin catalytic domain (SCD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043797((R)-2-Benzyloxycarbonylamino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  3.77E+5nMAssay Description:Inhibition of recombinant full length stromelysin (FLS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043804(5-(2-Amino-3-phenyl-propionylamino)-3-isobutyl-7-m...)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant full length stromelysin (FLS).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043804(5-(2-Amino-3-phenyl-propionylamino)-3-isobutyl-7-m...)
Affinity DataIC50:  18nMAssay Description:In vitro inhibition of recombinant stromelysin catalytic domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109692(3,4,5-Trihydroxy-benzoic acid 2-(3,4-dihydroxy-phe...)
Affinity DataIC50:  600nMAssay Description:Tested for its ability to inhibit HIV-1 reverse transcriptase strand transfer using A17 double mutant HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin gallate | (-)-Epigallocatechi...)
Affinity DataIC50:  730nMAssay Description:Inhibition of polymerization in wild type HIV-1 RT with poly rC/dG12-18 template primer and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50153015((-)-Epicatechin-3-gallate | (-)-epicatechin 3-O-ga...)
Affinity DataIC50:  760nMAssay Description:Inhibition of polymerization in wild type HIV-1 RT with poly rC/dG12-18 template primer and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109689(3,4,5-Trihydroxy-benzoic acid 5,7-dimethoxy-chroma...)
Affinity DataIC50:  900nMAssay Description:Tested for its ability to inhibit HIV-1 reverse transcriptase polymerization using A17 double mutant HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50105589(2,3,4-Trihydroxy-benzoic acid 5,7-dihydroxy-chroma...)
Affinity DataIC50:  2.36E+3nMAssay Description:Inhibitory concentration against polymerization in A17 double mutant HIV-1 RT using a template primer of poly rC/dG12-18 and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109688(3,4,5-Trihydroxy-benzoic acid 5,7-dihydroxy-chroma...)
Affinity DataIC50:  2.40E+3nMAssay Description:Tested for its ability to inhibit HIV-1 reverse transcriptase polymerization using A17 double mutant HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043807((S)-2-Benzyloxycarbonylamino-3-(1H-indol-3-yl)-pro...)
Affinity DataIC50:  2.50E+3nMAssay Description:In vitro inhibition of recombinant stromelysin catalytic domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109694(3,4,5-Trihydroxy-benzoic acid chroman-3-yl ester |...)
Affinity DataIC50:  2.60E+3nMAssay Description:Tested for its ability to inhibit HIV-1 reverse transcriptase strand transfer using A17 double mutant HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109688(3,4,5-Trihydroxy-benzoic acid 5,7-dihydroxy-chroma...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptase polymerization using wild type HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50105589(2,3,4-Trihydroxy-benzoic acid 5,7-dihydroxy-chroma...)
Affinity DataIC50:  3.83E+3nMAssay Description:Inhibition of polymerization in wild type HIV-1 RT with poly rC/dG12-18 template primer and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109690(3,4,5-Trihydroxy-benzoic acid 2-(4-hydroxy-phenyl)...)
Affinity DataIC50:  4.50E+3nMAssay Description:Tested for its ability to inhibit HIV-1 reverse transcriptase strand transfer using wild type HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109688(3,4,5-Trihydroxy-benzoic acid 5,7-dihydroxy-chroma...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptase polymerization using wild type HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109694(3,4,5-Trihydroxy-benzoic acid chroman-3-yl ester |...)
Affinity DataIC50:  6.10E+3nMAssay Description:Tested for its ability to inhibit HIV-1 reverse transcriptase strand transfer using wild type HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109688(3,4,5-Trihydroxy-benzoic acid 5,7-dihydroxy-chroma...)
Affinity DataIC50:  6.20E+3nMAssay Description:Tested for its ability to inhibit HIV-1 reverse transcriptase polymerization using A17 double mutant HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109692(3,4,5-Trihydroxy-benzoic acid 2-(3,4-dihydroxy-phe...)
Affinity DataIC50:  6.30E+3nMAssay Description:Tested for its ability to inhibit HIV-1 reverse transcriptase polymerization using A17 double mutant HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50105592(2,3,4-Trihydroxy-benzoic acid 2-(6,7-dihydroxy-chr...)
Affinity DataIC50:  6.33E+3nMAssay Description:Inhibitory concentration against polymerization in A17 double mutant HIV-1 RT using a template primer of poly rC/dG12-18 and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109689(3,4,5-Trihydroxy-benzoic acid 5,7-dimethoxy-chroma...)
Affinity DataIC50:  6.90E+3nMAssay Description:Tested for its ability to inhibit HIV-1 reverse transcriptase strand transfer using wild type HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109695(3,4,5-Trihydroxy-benzoic acid phenethyl ester | CH...)
Affinity DataIC50:  6.90E+3nMAssay Description:Tested for its ability to inhibit HIV-1 reverse transcriptase polymerization using A17 double mutant HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043807((S)-2-Benzyloxycarbonylamino-3-(1H-indol-3-yl)-pro...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of recombinant full length stromelysin (FLS).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109696(3,4,5-Trihydroxy-benzoic acid 7-hydroxy-chroman-3-...)
Affinity DataIC50:  7.60E+3nMAssay Description:Tested for its ability to inhibit HIV-1 reverse transcriptase polymerization using A17 double mutant HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109690(3,4,5-Trihydroxy-benzoic acid 2-(4-hydroxy-phenyl)...)
Affinity DataIC50:  7.90E+3nMAssay Description:Tested for its ability to inhibit HIV-1 reverse transcriptase strand transfer using A17 double mutant HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109697(3,4,5-Trihydroxy-benzoic acid 5-hydroxy-chroman-3-...)
Affinity DataIC50:  8.70E+3nMAssay Description:Tested for its ability to inhibit HIV-1 reverse transcriptase strand transfer using wild type HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043801((S)-2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-p...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of recombinant stromelysin catalytic domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109692(3,4,5-Trihydroxy-benzoic acid 2-(3,4-dihydroxy-phe...)
Affinity DataIC50:  1.05E+4nMAssay Description:Tested for its ability to inhibit HIV-1 reverse transcriptase strand transfer using wild type HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109692(3,4,5-Trihydroxy-benzoic acid 2-(3,4-dihydroxy-phe...)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase polymerization using wild type HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50105592(2,3,4-Trihydroxy-benzoic acid 2-(6,7-dihydroxy-chr...)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of polymerization in wild type HIV-1 RT with poly rC/dG12-18 template primer and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043805((S)-2-Benzyloxycarbonylamino-3-(1H-indol-3-yl)-pro...)
Affinity DataIC50:  1.30E+4nMAssay Description:In vitro inhibition of recombinant stromelysin catalytic domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043803((S)-2-Benzyloxycarbonylamino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of recombinant full length stromelysin (FLS).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043803((S)-2-Benzyloxycarbonylamino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50:  2.40E+4nMAssay Description:In vitro inhibition of recombinant stromelysin catalytic domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50109696(3,4,5-Trihydroxy-benzoic acid 7-hydroxy-chroman-3-...)
Affinity DataIC50:  3.08E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase polymerization using wild type HIV-1-RT enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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