Compile Data Set for Download or QSAR
maximum 50k data
Found 391 with Last Name = 'igawa' and Initial = 'h'
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50332808((8R,9S,10S,13S,14S)-10-(hydroxymethyl)-13-methyl-2...)
Affinity DataKi:  13nMAssay Description:Inhibition of 1 uM [1-beta-3H]-androstenedione binding to human placental microsome Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50332807((8R,9S,10R,13S,14S)-10,13-dimethyl-2,3,7,8,9,10,11...)
Affinity DataKi:  37nMAssay Description:Binding affinity for human placental microsome cytochrome P450 19A1 with 1 uM [1-beta-3H]-androstenedioneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50009437(10-Hydroxymethyl-13-methyl-2,3,6,7,8,9,10,11,12,13...)
Affinity DataKi:  170nMAssay Description:Inhibition of 1 uM [1-beta-3H]-androstenedione binding to human placental microsome Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50009430(16-Bromo-10,13-dimethyl-1,2,3,6,7,8,9,10,11,12,13,...)
Affinity DataKi:  228nMAssay Description:Binding affinity for human placental microsome cytochrome P450 19A1 with 1 uM [1-beta-3H]-androstenedioneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50009436(Acetic acid 13-methyl-17-oxo-1,2,3,6,7,8,9,11,12,1...)
Affinity DataKi:  289nMAssay Description:Binding affinity for human placental microsome cytochrome P450 19A1 with 1 uM [1-beta-3H]-androstenedioneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50009435(10-Difluoromethyl-13-methyl-1,2,3,6,7,8,9,10,11,12...)
Affinity DataKi:  443nMAssay Description:Binding affinity for human placental microsome cytochrome P450 19A1 with 1 uM [1-beta-3H]-androstenedioneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50009431(16-Bromo-10,13-dimethyl-1,2,3,6,7,8,9,10,11,12,13,...)
Affinity DataKi:  455nMAssay Description:Binding affinity for human placental microsome cytochrome P450 19A1 with 1 uM [1-beta-3H]-androstenedioneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50009434(10,13-Dimethyl-2,3,6,7,8,9,10,11,12,13,14,15,16,17...)
Affinity DataKi:  830nMAssay Description:Binding affinity for human placental microsome cytochrome P450 19A1 with 1 uM [1-beta-3H]-androstenedioneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50009433(10-(1-Hydroxy-prop-2-ynyl)-13-methyl-1,2,3,6,7,8,9...)
Affinity DataKi:  7.75E+3nMAssay Description:Binding affinity for human placental microsome cytochrome P450 19A1 with 1 uM [1-beta-3H]-androstenedioneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99943(US8501750, 56)
Affinity DataIC50:  0.340nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99950(US8501750, 83)
Affinity DataIC50:  0.770nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107366(US8592431, 167)
Affinity DataIC50:  0.800nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107347(US8592431, 135)
Affinity DataIC50:  0.900nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99949(US8501750, 76)
Affinity DataIC50:  1nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107364(US8592431, 264)
Affinity DataIC50:  1nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107354(US8592431, 147)
Affinity DataIC50:  1nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99952(US8501750, 105)
Affinity DataIC50:  1nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99946(US8501750, 60)
Affinity DataIC50:  1nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99947(US8501750, 63)
Affinity DataIC50:  1.10nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99953(US8501750, 107)
Affinity DataIC50:  1.10nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99961(US8501750, 131)
Affinity DataIC50:  1.20nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107445(US8592431, 376)
Affinity DataIC50:  1.20nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107435(US8592431, 354)
Affinity DataIC50:  1.20nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99980(US8501750, 181)
Affinity DataIC50:  1.20nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99981(US8501750, 186)
Affinity DataIC50:  1.20nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99951(US8501750, 99)
Affinity DataIC50:  1.20nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107361(US8592431, 241 | US8592431, 242)
Affinity DataIC50:  1.20nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99945(US8501750, 59)
Affinity DataIC50:  1.20nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107365(US8592431, 166)
Affinity DataIC50:  1.30nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107361(US8592431, 241 | US8592431, 242)
Affinity DataIC50:  1.30nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107350(US8592431, 138)
Affinity DataIC50:  1.30nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107348(US8592431, 136)
Affinity DataIC50:  1.30nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107346(US8592431, 134)
Affinity DataIC50:  1.30nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107340(US8592431, 117)
Affinity DataIC50:  1.30nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107318(US8592431, 2)
Affinity DataIC50:  1.30nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99992(US8501750, 215)
Affinity DataIC50:  1.30nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99974(US8501750, 153)
Affinity DataIC50:  1.30nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107368(US8592431, 169)
Affinity DataIC50:  1.40nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99958(US8501750, 127)
Affinity DataIC50:  1.40nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107330(US8592431, 69)
Affinity DataIC50:  1.40nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99988(US8501750, 209)
Affinity DataIC50:  1.40nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99954(US8501750, 109)
Affinity DataIC50:  1.40nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107349(US8592431, 137)
Affinity DataIC50:  1.40nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99984(US8501750, 197)
Affinity DataIC50:  1.40nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107431(US8592431, 339)
Affinity DataIC50:  1.40nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107434(US8592431, 352)
Affinity DataIC50:  1.40nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99977(US8501750, 157)
Affinity DataIC50:  1.40nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99993(US8501750, 221)
Affinity DataIC50:  1.40nMAssay Description:Binding assay using human AT1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107353(US8592431, 144)
Affinity DataIC50:  1.40nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-coenzyme A transporter 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM107356(US8592431, 150)
Affinity DataIC50:  1.40nMpH: 7.4Assay Description:The binding assay was performed using 22.5 pM [125I]-angiotensin II [manufactured by PerkinElmer, USA] (9 μg) in the presence of AT1 membrane an...More data for this Ligand-Target Pair
In DepthDetails US Patent
Displayed 1 to 50 (of 391 total ) | Next | Last >>
Jump to: