TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Inhibition of PI3Kalpha by HTRF assay in presence of ATPMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 8.30nMAssay Description:Inhibition of PI3Kdelta by HTRF assay in presence of ATPMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of PI3Kbeta by HTRF assay in presence of ATPMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of PI3Kgamma by HTRF assay in presence of ATPMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 96nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of PI3Kalpha by HTRF assay in presence of ATPMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of PI3Kbeta by HTRF assay in presence of ATPMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:The assays of DNA-PK were performed by Reaction Biology Corporation, One Great Valley Parkway, Suite 2 Malvern, PA 19355 USA. All Compounds were diss...More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of DNA-PK using EPPLSQEAFADLWKK as substrate after 5 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of DNA-PK using EPPLSQEAFADLWKK as substrate after 5 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of DNA-PK using EPPLSQEAFADLWKK as substrate after 5 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of DNA-PK using EPPLSQEAFADLWKK as substrate after 5 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Inhibition of PI3Kbeta by HTRF assay in presence of ATPMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 620nMAssay Description:Inhibition of DNA-PK using EPPLSQEAFADLWKK as substrate after 5 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 717nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of PI3Kgamma by HTRF assay in presence of ATPMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 760nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 930nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 950nMAssay Description:Inhibition of PI3Kdelta by HTRF assay in presence of ATPMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of DNA-PK using EPPLSQEAFADLWKK as substrate after 5 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of DNA-PK using EPPLSQEAFADLWKK as substrate after 5 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of PI3Kgamma by HTRF assay in presence of ATPMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of DNA-PK using EPPLSQEAFADLWKK as substrate after 5 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of DNA-PK using EPPLSQEAFADLWKK as substrate after 5 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 2.02E+3nMAssay Description:Inhibition of PI3Kdelta by HTRF assay in presence of ATPMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 2.34E+3nMAssay Description:Inhibition of PI3Kbeta by HTRF assay in presence of ATPMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 2.43E+3nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of DNA-PK using EPPLSQEAFADLWKK as substrate after 5 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:The assays of DNA-PK were performed by Reaction Biology Corporation, One Great Valley Parkway, Suite 2 Malvern, PA 19355 USA. All Compounds were diss...More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of DNA-PK using EPPLSQEAFADLWKK as substrate after 5 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of DNA-PK using EPPLSQEAFADLWKK as substrate after 5 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 3.09E+3nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 3.36E+3nMAssay Description:Inhibition of PI3Kbeta by HTRF assay in presence of ATPMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 3.41E+3nMAssay Description:Inhibition of PI3Kalpha by HTRF assay in presence of ATPMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:The assays of DNA-PK were performed by Reaction Biology Corporation, One Great Valley Parkway, Suite 2 Malvern, PA 19355 USA. All Compounds were diss...More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of DNA-PKMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:The assays of DNA-PK were performed by Reaction Biology Corporation, One Great Valley Parkway, Suite 2 Malvern, PA 19355 USA. All Compounds were diss...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 4.07E+3nMAssay Description:Inhibition of PI3Kalpha by HTRF assay in presence of ATPMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of DNA-PK using EPPLSQEAFADLWKK as substrate after 5 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:The assays of DNA-PK were performed by Reaction Biology Corporation, One Great Valley Parkway, Suite 2 Malvern, PA 19355 USA. All Compounds were diss...More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of DNA-PK using EPPLSQEAFADLWKK as substrate after 5 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair