Affinity DataKi: 4.32E+3nMAssay Description:Reversible inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NPMore data for this Ligand-Target Pair
Affinity DataKi: 2.48E+4nMAssay Description:Reversible inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NPMore data for this Ligand-Target Pair
Affinity DataKi: 3.55E+5nMAssay Description:Reversible inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NPMore data for this Ligand-Target Pair
Affinity DataKi: 3.63E+5nMAssay Description:Inhibition of human CES1More data for this Ligand-Target Pair
Affinity DataKi: 4.68E+5nMAssay Description:Reversible inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NPMore data for this Ligand-Target Pair
Affinity DataKi: 7.07E+5nMAssay Description:Reversible inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NPMore data for this Ligand-Target Pair
Affinity DataKi: 7.90E+6nMAssay Description:Inhibition of human CES2More data for this Ligand-Target Pair
Affinity DataIC50: 1.96E+3nMAssay Description:Time-dependent inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NP preincubated for 30 mins followed by 4NPA additionMore data for this Ligand-Target Pair
Affinity DataIC50: 2.27E+3nMAssay Description:Time-dependent inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NP preincubated for 60 mins followed by 4NPA additionMore data for this Ligand-Target Pair
Affinity DataIC50: 2.51E+3nMAssay Description:Time-dependent inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NP preincubated for 10 mins followed by 4NPA additionMore data for this Ligand-Target Pair
Affinity DataEC50: 850nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 8.5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 34nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 21nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 600nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 75nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 8.5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 6.5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 6.5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 9nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 4.5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 7.5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+3nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 800nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 4.60E+3nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 900nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+4nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair