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Found 143 with Last Name = 'inoue' and Initial = 'r'
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50088512(CHEBI:59609 | CHEMBL3527338)
Affinity DataKi:  4.32E+3nMAssay Description:Reversible inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50088513(CHEMBL3526940)
Affinity DataKi:  2.48E+4nMAssay Description:Reversible inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50088514(CHEBI:88735 | CHEMBL3526740)
Affinity DataKi:  3.55E+5nMAssay Description:Reversible inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50003616(2-n-propyl-n-valeric acid | CHEMBL109 | DPA | Di-n...)
Affinity DataKi:  3.63E+5nMAssay Description:Inhibition of human CES1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50088516(CHEMBL3526990)
Affinity DataKi:  4.68E+5nMAssay Description:Reversible inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50088515(CHEMBL3526991)
Affinity DataKi:  7.07E+5nMAssay Description:Reversible inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50003616(2-n-propyl-n-valeric acid | CHEMBL109 | DPA | Di-n...)
Affinity DataKi:  7.90E+6nMAssay Description:Inhibition of human CES2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50088512(CHEBI:59609 | CHEMBL3527338)
Affinity DataIC50:  1.96E+3nMAssay Description:Time-dependent inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NP preincubated for 30 mins followed by 4NPA additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50088512(CHEBI:59609 | CHEMBL3527338)
Affinity DataIC50:  2.27E+3nMAssay Description:Time-dependent inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NP preincubated for 60 mins followed by 4NPA additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50088512(CHEBI:59609 | CHEMBL3527338)
Affinity DataIC50:  2.51E+3nMAssay Description:Time-dependent inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NP preincubated for 10 mins followed by 4NPA additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364594(CHEMBL1951148)
Affinity DataEC50:  850nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364595(CHEMBL1951149)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364596(CHEMBL1951150)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364597(CHEMBL1951151)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364598(CHEMBL1951152)
Affinity DataEC50:  8.5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364599(CHEMBL1951153)
Affinity DataEC50:  34nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364600(CHEMBL1951154)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364601(CHEMBL1951155)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364602(CHEMBL1951156)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364603(CHEMBL1951157)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364604(CHEMBL1951158)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364605(CHEMBL1951159)
Affinity DataEC50:  600nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364606(CHEMBL1951303)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364607(CHEMBL1951304)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364608(CHEMBL1951305)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364609(CHEMBL1951306)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364610(CHEMBL1951307)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364611(CHEMBL1951308)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364612(CHEMBL1951309)
Affinity DataEC50:  8.5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364613(CHEMBL1951310)
Affinity DataEC50:  6.5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364614(CHEMBL1951311)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364615(CHEMBL1951312)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364616(CHEMBL1951313)
Affinity DataEC50:  6.5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364617(CHEMBL1951314)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364618(CHEMBL1949690)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364619(CHEMBL1951315)
Affinity DataEC50:  4.5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364620(CHEMBL1951316)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364621(CHEMBL1951317)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364622(CHEMBL1951318)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364623(CHEMBL1951319)
Affinity DataEC50:  7.5nMAssay Description:Agonist activity at human S1P1 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50158349(1-(4-(5-(4-phenyl-5-(trifluoromethyl)thiophen-2-yl...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364624(CHEMBL1951147)
Affinity DataEC50:  800nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364594(CHEMBL1951148)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364595(CHEMBL1951149)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364596(CHEMBL1951150)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364597(CHEMBL1951151)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364598(CHEMBL1951152)
Affinity DataEC50:  4.60E+3nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364599(CHEMBL1951153)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364600(CHEMBL1951154)
Affinity DataEC50:  900nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364601(CHEMBL1951155)
Affinity DataEC50:  1.20E+4nMAssay Description:Agonist activity at human S1P3 receptor assessed as stimulation of [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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