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Found 168 with Last Name = 'ishii' and Initial = 's'
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118202(6-(4-azido-2,3,5,6-tetrafluorobenzyloxy)-8-(tert-b...)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123637(6-benzyloxy-8-(tert-butyl)-9-flouro-12,17-dihydrox...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123639(8-(tert-butyl)-9-chloro-6,12,17-trihydroxy-16-meth...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123644(6-benzyloxy-8-(tert-butyl)-12,17-dihydroxy-16-meth...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118204(6-(4-benzoylphenylcarbonyloxy)-8-(tert-butyl)-12,1...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118194(8-(tert-butyl)-12,17-dihydroxy-16-methyl-6-[4-(3-t...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118201(6-(4-benzoylbenzyloxy)-8-(tert-butyl)-12,17-dihydr...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118203(8-(tert-butyl)-9,12,17-trihydroxy-16-methyl-6-[4-(...)
Affinity DataKi:  470nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123638(9-azido-8-(tert-butyl)-6,12,17-trihydroxy-16-methy...)
Affinity DataKi:  550nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118195(3'-(tert-butyl)-4,9',14'-trihydroxy-2-methoxy-10'-...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118196(6-(4-benzoylbenzyloxy)-8-(tert-butyl)-9,12,17-trih...)
Affinity DataKi:  580nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123643(6-benzyloxy-8-(tert-butyl)-9,12,17-trihydroxy-16-m...)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123633(8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-9-meth...)
Affinity DataKi:  610nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118200(6-(4-azido-2,3,5,6-tetrafluorobenzyloxy)-8-(tert-b...)
Affinity DataKi:  790nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50251276(BN 52021 | CHEMBL514432 | GINKOLIDE B | Gingkolide...)
Affinity DataKi:  880nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123642(8-(tert-butyl)-9-flouro-6,12,17-trihydroxy-16-meth...)
Affinity DataKi:  990nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118205(3'-(tert-butyl)-4,9'-dihydroxy-2-methoxy-10'-methy...)
Affinity DataKi:  1.46E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123631(8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-9-ethy...)
Affinity DataKi:  1.62E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123632(6-benzyloxy-8-(tert-butyl)-9,12,17-trihydroxy-16-m...)
Affinity DataKi:  1.67E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123645(CHEMBL348623 | benzyl (6R,9R,12R,16S,17R)-8-tert-b...)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123635(8-(tert-butyl)-6,9,12,17-tetrahydroxy-16-methyl-(6...)
Affinity DataKi:  4.26E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123636(8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-5,15,1...)
Affinity DataKi:  7.84E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123640(8-(tert-butyl)-6,12,17-trihydroxy-16-methyl-9-amin...)
Affinity DataKi:  8.64E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118193(3'-(tert-butyl)-4,4',9'-trihydroxy-2-methoxy-10'-m...)
Affinity DataKi:  9.90E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50123641(8-(tert-butyl)-6,9,12,17-tetrahydroxy-16-methyl-(6...)
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118197(3'-(tert-butyl)-4,4',9',14'-tetrahydroxy-2-methoxy...)
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118199(9-tert-Butyl-8,9-dihydroxy-dihydro-furo[2,3-b]furo...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Mus musculus)
Columbia University

Curated by ChEMBL
LigandPNGBDBM50118198(3'-(tert-butyl)-4,4',14'-trihydroxy-2-methoxy-10'-...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391561(CHEMBL2147704)
Affinity DataIC50:  0.180nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391559(CHEMBL2147703)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391561(CHEMBL2147704)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50166315(6-((3S,5S)-5-((S)-2-cyanopyrrolidine-1-carbonyl)py...)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391559(CHEMBL2147703)
Affinity DataIC50:  0.260nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391565(CHEMBL2147777)
Affinity DataIC50:  0.290nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391570(CHEMBL2147712)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391567(CHEMBL2147709)
Affinity DataIC50:  0.310nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391567(CHEMBL2147709)
Affinity DataIC50:  0.320nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388112(CHEMBL2058971)
Affinity DataIC50:  0.370nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391565(CHEMBL2147777)
Affinity DataIC50:  0.370nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391570(CHEMBL2147712)
Affinity DataIC50:  0.490nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391571(CHEMBL2147713)
Affinity DataIC50:  0.530nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391576(CHEMBL2147773)
Affinity DataIC50:  0.620nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391568(CHEMBL2147771)
Affinity DataIC50:  0.630nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391564(CHEMBL2147707)
Affinity DataIC50:  0.690nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391568(CHEMBL2147771)
Affinity DataIC50:  0.720nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391576(CHEMBL2147773)
Affinity DataIC50:  0.770nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391571(CHEMBL2147713)
Affinity DataIC50:  0.850nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391564(CHEMBL2147707)
Affinity DataIC50:  0.940nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388117(CHEMBL2058969)
Affinity DataIC50:  0.950nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388117(CHEMBL2058969)
Affinity DataIC50:  1nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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