Affinity DataKi: 0.0200nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 0.630nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.790nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 103nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 109nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 121nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 137nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 143nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 152nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 238nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 288nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 379nMAssay Description:Inhibition of FAAH activity in Wistar rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 398nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 690nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Rattus norvegicus)
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 710nMAssay Description:Inhibition of GluT1-mediated [14C]D-glucose uptake in Wistar rat brain by perfusion techniqueMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio
Curated by ChEMBL
University Of Kuopio
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair