Affinity DataKi: 120nM ΔG°: -39.1kJ/molepH: 7.2 T: 2°CAssay Description:Hydrolysis of substrate p-nitrophenyl phosphate was monitored on a 96-well microplate reader. Concentrations of PTP1B inhibitors that resulted in 50%...More data for this Ligand-Target Pair
Affinity DataKi: 250nM ΔG°: -37.3kJ/molepH: 7.2 T: 2°CAssay Description:Hydrolysis of substrate p-nitrophenyl phosphate was monitored on a 96-well microplate reader. Concentrations of PTP1B inhibitors that resulted in 50%...More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nM ΔG°: -33.5kJ/molepH: 7.2 T: 2°CAssay Description:Hydrolysis of substrate p-nitrophenyl phosphate was monitored on a 96-well microplate reader. Concentrations of PTP1B inhibitors that resulted in 50%...More data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nM ΔG°: -31.4kJ/molepH: 7.2 T: 2°CAssay Description:Hydrolysis of substrate p-nitrophenyl phosphate was monitored on a 96-well microplate reader. Concentrations of PTP1B inhibitors that resulted in 50%...More data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nM ΔG°: -30.9kJ/molepH: 7.2 T: 2°CAssay Description:Hydrolysis of substrate p-nitrophenyl phosphate was monitored on a 96-well microplate reader. Concentrations of PTP1B inhibitors that resulted in 50%...More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nM ΔG°: -30.0kJ/molepH: 7.2 T: 2°CAssay Description:Hydrolysis of substrate p-nitrophenyl phosphate was monitored on a 96-well microplate reader. Concentrations of PTP1B inhibitors that resulted in 50%...More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+4nM ΔG°: -27.8kJ/molepH: 7.2 T: 2°CAssay Description:Hydrolysis of substrate p-nitrophenyl phosphate was monitored on a 96-well microplate reader. Concentrations of PTP1B inhibitors that resulted in 50%...More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+4nM ΔG°: -25.6kJ/molepH: 7.2 T: 2°CAssay Description:Hydrolysis of substrate p-nitrophenyl phosphate was monitored on a 96-well microplate reader. Concentrations of PTP1B inhibitors that resulted in 50%...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nM ΔG°: >-22.6kJ/molepH: 7.2 T: 2°CAssay Description:Hydrolysis of substrate p-nitrophenyl phosphate was monitored on a 96-well microplate reader. Concentrations of PTP1B inhibitors that resulted in 50%...More data for this Ligand-Target Pair
Affinity DataIC50: 850nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: >7.50E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: >7.50E+4nMAssay Description:In vitro inhibitory activity against ADP-induced human platelet aggregationMore data for this Ligand-Target Pair