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Found 185 with Last Name = 'jadav' and Initial = 'ss'
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493741(CHEMBL2437020)
Affinity DataKi:  4nMAssay Description:Competitive inhibition of human recombinant MAO-A expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate by Lineweaver-Burk...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM15613(4-chloro-N-(2-morpholin-4-ylethyl)benzamide | 4-ch...)
Affinity DataKi:  5nMAssay Description:Competitive reversible inhibition of human recombinant MAO-A expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493741(CHEMBL2437020)
Affinity DataKi:  5nMAssay Description:Competitive reversible inhibition of human recombinant MAO-A expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50537558(Narlaprevir | SCH 900518 | SCH-900518)
Affinity DataKi:  6nMAssay Description:Inhibition of Epidermal growth factor receptor autophosphorylation in A431 human epidermoid carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))TBA
LigandPNGBDBM50407493(CHEMBL5288446)
Affinity DataKi:  15nMAssay Description:Relative potency against Histamine H1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50537563(CHEMBL4634405)
Affinity DataKi:  20nMAssay Description:Inhibition of Epidermal growth factor receptor from human A431 cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50103860(2-{[2-(5-Carbamoyl-1H-benzoimidazol-2-ylmethyl)-3-...)
Affinity DataKi:  27nMAssay Description:Inhibitory activity against HIV-1 wild-type reverse transcriptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493747(CHEMBL2437021)
Affinity DataKi:  30nMAssay Description:Competitive reversible inhibition of human recombinant MAO-A expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50537564(CHEMBL4644516)
Affinity DataKi:  40nMAssay Description:Inhibition of Epidermal growth factor receptor autophosphorylation in A431 human epidermoid carcinoma cellsMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM15579(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Affinity DataKi:  90nMAssay Description:Competitive reversible inhibition of human recombinant MAO-B expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))TBA
LigandPNGBDBM50407492(CHEMBL5280732)
Affinity DataKi:  120nMAssay Description:Apparent pA2 value of compound at 50 nM concentration of mepyramine in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493742(CHEMBL2437022)
Affinity DataKi:  250nMAssay Description:Competitive reversible inhibition of human recombinant MAO-A expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493744(CHEMBL2437019)
Affinity DataKi:  310nMAssay Description:Competitive reversible inhibition of human recombinant MAO-A expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50537569(CHEMBL4646328)
Affinity DataKi:  600nMAssay Description:Inhibitory activity against HIV-1 Mutant Reverse transcriptase K103NMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493748(CHEMBL2437015)
Affinity DataKi:  610nMAssay Description:Competitive reversible inhibition of human recombinant MAO-A expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493745(CHEMBL2437017)
Affinity DataKi:  760nMAssay Description:Competitive reversible inhibition of human recombinant MAO-A expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493743(CHEMBL2437018)
Affinity DataKi:  810nMAssay Description:Competitive reversible inhibition of human recombinant MAO-A expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493746(CHEMBL2437016)
Affinity DataKi:  880nMAssay Description:Competitive reversible inhibition of human recombinant MAO-A expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50103860(2-{[2-(5-Carbamoyl-1H-benzoimidazol-2-ylmethyl)-3-...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibitory activity against HIV-1 Mutant Reverse transcriptase G190AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM15613(4-chloro-N-(2-morpholin-4-ylethyl)benzamide | 4-ch...)
Affinity DataKi:  1.08E+3nMAssay Description:Competitive reversible inhibition of human recombinant MAO-B expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))TBA
LigandPNGBDBM50407464(CHEMBL5289275)
Affinity DataKi:  2.41E+3nMAssay Description:Apparent pA2 value of compound at 10 nM concentration of mepyramine in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))TBA
LigandPNGBDBM50407467(CHEMBL5289169)
Affinity DataKi:  3.12E+3nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))TBA
LigandPNGBDBM50407491(CHEMBL5282293)
Affinity DataKi:  3.80E+3nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493748(CHEMBL2437015)
Affinity DataKi:  5.00E+3nMAssay Description:Competitive reversible inhibition of human recombinant MAO-B expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493746(CHEMBL2437016)
Affinity DataKi:  6.00E+3nMAssay Description:Competitive reversible inhibition of human recombinant MAO-B expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM15579(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Affinity DataKi:  9.06E+3nMAssay Description:Competitive reversible inhibition of human recombinant MAO-A expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493743(CHEMBL2437018)
Affinity DataKi:  1.10E+4nMAssay Description:Competitive reversible inhibition of human recombinant MAO-B expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493745(CHEMBL2437017)
Affinity DataKi:  1.56E+4nMAssay Description:Competitive reversible inhibition of human recombinant MAO-B expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))TBA
LigandPNGBDBM50407461(CHEMBL5274458)
Affinity DataKi:  4.46E+4nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493747(CHEMBL2437021)
Affinity DataKi:  4.50E+4nMAssay Description:Competitive reversible inhibition of human recombinant MAO-B expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493741(CHEMBL2437020)
Affinity DataKi:  5.60E+4nMAssay Description:Competitive reversible inhibition of human recombinant MAO-B expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493744(CHEMBL2437019)
Affinity DataKi:  3.05E+5nMAssay Description:Competitive reversible inhibition of human recombinant MAO-B expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50493742(CHEMBL2437022)
Affinity DataKi:  5.30E+5nMAssay Description:Competitive reversible inhibition of human recombinant MAO-B expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target7-dehydrocholesterol reductase(Homo sapiens (Human))TBA
LigandPNGBDBM50407454(CHEMBL5281526)
Affinity DataIC50:  0.100nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50495950(Danoprevir | R-05190591 | R05190591 | RO-5190591 |...)
Affinity DataIC50:  0.200nMAssay Description:Inhibitory activity against HIV-1 Mutant Reverse transcriptase K103NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50485492(Grazoprevir | Grazoprevir monohydrate | MK-5172 | ...)
Affinity DataIC50:  2nMAssay Description:Inhibition of Epidermal growth factor receptor autophosphorylation in A431 human epidermoid carcinoma cellsMore data for this Ligand-Target Pair
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50537589(CHEMBL4287268)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against HIV-1 Y188L reverse transcriptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50407449(CHEMBL5285995)
Affinity DataIC50:  3nMAssay Description:Antagonistic affinity tested against isolated Rat Thoracic Aorta Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))TBA
LigandPNGBDBM50407495(CHEMBL5286471)
Affinity DataIC50:  4nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50537581(CHEMBL4638107)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against HIV-1 Mutant Reverse transcriptase G190AMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50537583(CHEMBL4638630)
Affinity DataIC50:  4.30nMAssay Description:Inhibitory activity against HIV-1 wild-type reverse transcriptase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50537585(CHEMBL4646449)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against HIV-1 Y181C reverse transcriptase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Homo sapiens (Human))TBA
LigandPNGBDBM50407496(CHEMBL5284382)
Affinity DataIC50:  5nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50537587(CHEMBL4633142)
Affinity DataIC50:  6nMAssay Description:Inhibitory activity against HIV-1 Y181C reverse transcriptase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50537579(CHEMBL4635161)
Affinity DataIC50:  6nMAssay Description:Inhibitory activity against HIV-1 wild-type reverse transcriptase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50537578(CHEMBL245328)
Affinity DataIC50:  7.20nMAssay Description:Inhibitory activity against HIV-1 wild-type reverse transcriptase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50379197(CHEMBL2011266)
Affinity DataIC50:  8nMAssay Description:Inhibitory activity against HIV-1 Y188L reverse transcriptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50407448(CHEMBL4454956)
Affinity DataIC50:  9.40nMAssay Description:Antagonistic affinity tested against isolated Rat Thoracic Aorta Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50537575(CHEMBL4638877)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against HIV-1 Y181C reverse transcriptase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM50537574(CHEMBL4643906)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against HIV-1 wild-type reverse transcriptase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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