Affinity DataKi: 0.0390nMAssay Description:Compound was evaluated for its binding affinity by displacing [3H]U-69593 to human cloned Kappa opioid receptor transfected into CHO cells using [35S...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 0.0610nMAssay Description:Compound was evaluated for its binding affinity to CHO cells expressing cloned human Opioid receptor kappa 1 by displacing [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Binding affinity against 5-hydroxytryptamine 4 receptor in guinea pig striatum using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:In vitro ability to displace [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Compound was evaluated for its binding affinity by displacing [3H]U-69593 to human cloned Kappa opioid receptor transfected into CHO cells using [35S...More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Compound was evaluated for its binding affinity by displacing [3H]U-69593 to human cloned Kappa opioid receptor transfected into CHO cells using [35S...More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]U-69593 from human recombinant Opioid receptor kappa 1 on CHO cell membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Compound was evaluated for its binding affinity to CHO cells expressing cloned human Opioid receptor kappa 1 by displacing [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]DAMGO from human recombinant Opioid receptor mu 1 on CHO cell membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]C1-DPDPE from human recombinant Opioid receptor delta 1 on CHO cell membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Ability to displace [3H]U-69593 from human recombinant Opioid receptor kappa 1 in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:In vitro ability to displace [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:In vitro ability to displace [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Ability to displace [3H]U-69593 from human recombinant Opioid receptor kappa 1 in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:In vitro ability to displace [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Ability to displace [3H]U-69593 from human recombinant Opioid receptor kappa 1 in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Ability to displace [3H]U-69593 from human recombinant Opioid receptor kappa 1 in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]U-69593 from human recombinant Opioid receptor kappa 1 on CHO cell membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Ability to displace [3H]U-69593 from human recombinant Opioid receptor kappa 1 in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Compound was evaluated for its binding affinity to CHO cells expressing cloned human Opioid receptor kappa 1 by displacing [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 0.316nMAssay Description:In vitro by displacement of [3H]LY-278584 from 5-hydroxytryptamine 3 receptor on rat entorhinal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.316nMAssay Description:In vitro by displacement of [3H]LY-278584 from 5-hydroxytryptamine 3 receptor on rat entorhinal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.316nMAssay Description:In vitro by displacement of [3H]LY-278584 from 5-hydroxytryptamine 3 receptor on rat entorhinal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:In vitro ability to displace [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
Affinity DataKi: 0.398nMAssay Description:In vitro by displacement of [3H]LY-278584 from 5-hydroxytryptamine 3 receptor on rat entorhinal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Hartely guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Hartely guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]U-69593 from human recombinant Opioid receptor kappa 1 on CHO cell membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]DAMGO from human recombinant Opioid receptor mu 1 on CHO cell membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibitory concentration against 5-hydroxytryptamine 3 receptor in rat enthorinal cortex using [3H]-LY 278584 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]U69,593 from kappa opioid receptor in Hartely guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.620nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 3 receptor was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 0.630nMAssay Description:In vitro ability to displace [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor sites of rat brain cortex.More data for this Ligand-Target Pair
Affinity DataKi: 0.631nMAssay Description:Binding affinity was evaluated in vitro by displacement of [3H]ketanserin from 5-hydroxytryptamine 2A receptor on rat cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.631nMAssay Description:In vitro by displacement of [3H]LY-278584 from 5-hydroxytryptamine 3 receptor on rat entorhinal cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.631nMAssay Description:In vitro by displacement of [3H]raclopride from Dopamine receptor D2 on rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.680nMAssay Description:Ability to displace [3H]U-69593 from human recombinant Opioid receptor kappa 1 in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity to the serotonin transporter (SERT) measured by displacement of [3H]paroxetine in male wistar ratsMore data for this Ligand-Target Pair