BindingDB PrimarySearch_ki

Found 1516 with Last Name = 'jha' and Initial = 't'

72 kDa type IV collagenase(Homo sapiens (Human))TBA

PNG

BDBM50082556((S)-2,2-Dimethyl-4-[4-(pyridin-4-yloxy)-benzenesul...)

Ki: 0.0500nMAssay Description:Inhibition of human MMP-2 assessed as inhibition constant using MCA-Pro-Leu-Gly-Leu-DPA-Ala-Arg-NH2 substrate by fluorimetric analysisMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Aromatase(Homo sapiens (Human))TBA

PNG

BDBM50240798((8R,9S,10R,13S,14S)-4-Hydroxy-10,13-dimethyl-1,6,7...)

Ki: 0.160nMAssay Description:Binding affinity to aromatase (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

ChEBI
CHEMBL PC cid PC sid Patents Similars

Neutrophil collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)

Ki: 0.180nMAssay Description:Inhibition of MMP-8 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Macrophage metalloelastase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50592891(CHEMBL5191016)

Ki: 0.190nMAssay Description:Inhibition of human MMP-12 expressed in Escherichia coli BL21(DE3) using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 30 mins fo...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Matrix metalloproteinase-9(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)

Ki: 0.200nMAssay Description:Inhibition of MMP-9 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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72 kDa type IV collagenase(Homo sapiens (Human))TBA

PNG

BDBM11870(4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxy ...)

Ki: 0.220nMAssay Description:Inhibition of MMP-2 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid Patents Similars

Matrix metalloproteinase-9(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50082556((S)-2,2-Dimethyl-4-[4-(pyridin-4-yloxy)-benzenesul...)

Ki: 0.260nMAssay Description:Inhibition of human MMP-9 assessed as inhibition constant using MCA-Pro-Leu-Gly-Leu-DPA-Ala-Arg-NH2 substrate by fluorimetric analysisMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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72 kDa type IV collagenase(Homo sapiens (Human))TBA

PNG

BDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)

Ki: 0.390nMAssay Description:Inhibition of MMP-2 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Interstitial collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)

Ki: 0.400nMAssay Description:Inhibition of MMP-1 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Collagenase 3(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM11870(4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxy ...)

Ki: 0.520nMAssay Description:Inhibition of MMP-13 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid Patents Similars

Matrix metalloproteinase-9(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)

Ki: 0.570nMAssay Description:Inhibition of MMP-9 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Matrix metalloproteinase-9(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM11870(4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxy ...)

Ki: 0.580nMAssay Description:Inhibition of MMP-9 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid Patents Similars

Aminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50457465(CHEMBL4204736)

Ki: 0.600nMAssay Description:Inhibition of APN in porcine kidney using Ala-p-NA as substrateMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Aromatase(Homo sapiens (Human))TBA

PNG

BDBM50398447(Aromasin | EXEMESTANE)

Ki: 0.950nMAssay Description:Binding affinity to aromatase (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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PDB

3D Structure (crystal)

Protease(Human immunodeficiency virus 1 (HIV-1))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50482863(CHEMBL1255913)

Ki: 0.979nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair

PDB
UniProtKB/TrEMBL
B.MOAD GoogleScholar

Details Article PubMed

Protease(Human immunodeficiency virus 1 (HIV-1))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50482863(CHEMBL1255913)

Ki: 0.980nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair

PDB
UniProtKB/TrEMBL
B.MOAD GoogleScholar

Details Article PubMed

Aminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50457475(CHEMBL4216408)

Ki: 1.5nMAssay Description:Inhibition of APN in porcine kidney using Ala-p-NA as substrateMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Neutrophil collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM13126((2R)-2-[benzyl(4-methoxybenzene)sulfonamido]-N-hyd...)

Ki: 1.90nMAssay Description:Inhibition of MMP-8 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Protease(Human immunodeficiency virus 1 (HIV-1))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50482855(CHEMBL1255911)

Ki: 2.10nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair

PDB
UniProtKB/TrEMBL
B.MOAD GoogleScholar

Details Article PubMed

Protease(Human immunodeficiency virus 1 (HIV-1))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50482855(CHEMBL1255911)

Ki: 2.10nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair

PDB
UniProtKB/TrEMBL
B.MOAD GoogleScholar

Details Article PubMed

Protease(Human immunodeficiency virus 1 (HIV-1))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50482870(CHEMBL1255912)

Ki: 2.60nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair

PDB
UniProtKB/TrEMBL
B.MOAD GoogleScholar

Details Article PubMed

Protease(Human immunodeficiency virus 1 (HIV-1))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50482870(CHEMBL1255912)

Ki: 2.60nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair

PDB
UniProtKB/TrEMBL
B.MOAD GoogleScholar

Details Article PubMed

Collagenase 3(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50592900(CHEMBL5175770)

Ki: 3nMAssay Description:Inhibition of MMP-13 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Interstitial collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50592900(CHEMBL5175770)

Ki: 3nMAssay Description:Inhibition of MMP-1 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Interstitial collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50592900(CHEMBL5175770)

Ki: 3nMAssay Description:Inhibition of human recombinant MMP-1 assessed as inhibition constantMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Matrix metalloproteinase-9(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50592895(CHEMBL5187653)

Ki: 3nMAssay Description:Inhibition of MMP-9 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Neutrophil collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50592895(CHEMBL5187653)

Ki: 3nMAssay Description:Inhibition of MMP-8 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Collagenase 3(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM13126((2R)-2-[benzyl(4-methoxybenzene)sulfonamido]-N-hyd...)

Ki: 3.40nMAssay Description:Inhibition of MMP-13 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Protease(Human immunodeficiency virus 1 (HIV-1))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50482856(CHEMBL1255914)

Ki: 3.5nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair

PDB
UniProtKB/TrEMBL
B.MOAD GoogleScholar

Details Article PubMed

Protease(Human immunodeficiency virus 1 (HIV-1))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50482856(CHEMBL1255914)

Ki: 3.5nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair

PDB
UniProtKB/TrEMBL
B.MOAD GoogleScholar

Details Article PubMed

72 kDa type IV collagenase(Homo sapiens (Human))TBA

PNG

BDBM11548(CHEMBL100570 | N-hydroxy-2-[(4-methoxy-1,1-bipheny...)

Ki: 3.80nMAssay Description:Inhibition of MMP-2 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Neutrophil collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50592900(CHEMBL5175770)

Ki: 4nMAssay Description:Inhibition of MMP-8 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Neutrophil collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50077789((2S,3R,6S)-4-Oxo-3-(3-phenyl-propyl)-1-oxa-5,10-di...)

Ki: 4nMAssay Description:Inhibition of MMP-8 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

72 kDa type IV collagenase(Homo sapiens (Human))TBA

PNG

BDBM50592895(CHEMBL5187653)

Ki: 4nMAssay Description:Inhibition of MMP-2 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Neutrophil collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50592900(CHEMBL5175770)

Ki: 4.40nMAssay Description:Inhibition of MMP-8 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Macrophage metalloelastase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50433864(CHEMBL2380403)

Ki: 4.80nMAssay Description:Inhibition of MMP12 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Macrophage metalloelastase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50592895(CHEMBL5187653)

Ki: 5nMAssay Description:Inhibition of MMP-12 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Histone deacetylase 3(Homo sapiens (Human))TBA

PNG

BDBM207629(US9265734, R01 | US9796664, Compound R01)

Ki: 5nMAssay Description:Binding affinity to human recombinant HDAC3 assessed as inhibition constantMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Matrix metalloproteinase-14(Homo sapiens (Human))TBA

PNG

BDBM50433864(CHEMBL2380403)

Ki: 5nMAssay Description:Inhibition of MMP14 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Matrix metalloproteinase-9(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50335495(4-(4-(thiiran-2-ylmethylsulfonyl)phenoxy)phenyl me...)

Ki: 5nMAssay Description:Competitive inhibition of human MMP-9 assessed as inhibition constantMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

72 kDa type IV collagenase(Homo sapiens (Human))TBA

PNG

BDBM50388914(CHEMBL2063274 | US10357546, p-OH SB-3CT)

Ki: 6nMAssay Description:Competitive inhibition of human MMP-2 assessed as inhibition constantMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Protease(Human immunodeficiency virus 1 (HIV-1))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50482862(CHEMBL1255922)

Ki: 7nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair

PDB
UniProtKB/TrEMBL
B.MOAD GoogleScholar

Details Article PubMed

Collagenase 3(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50592895(CHEMBL5187653)

Ki: 7nMAssay Description:Inhibition of MMP-13 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Protease(Human immunodeficiency virus 1 (HIV-1))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50482862(CHEMBL1255922)

Ki: 7nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair

PDB
UniProtKB/TrEMBL
B.MOAD GoogleScholar

Details Article PubMed

Matrix metalloproteinase-9(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM13126((2R)-2-[benzyl(4-methoxybenzene)sulfonamido]-N-hyd...)

Ki: 8nMAssay Description:Inhibition of MMP-9 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Matrix metalloproteinase-9(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM13126((2R)-2-[benzyl(4-methoxybenzene)sulfonamido]-N-hyd...)

Ki: 8nMAssay Description:Inhibition of recombinant human MMP-9 assessed as inhibition constantMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Aminopeptidase N(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50457479(CHEMBL1159812)

Ki: 8nMAssay Description:Inhibition of APN in human placenta using AlabetaNA as substrateMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Interstitial collagenase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50592895(CHEMBL5187653)

Ki: 8nMAssay Description:Inhibition of MMP-1 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Protease(Human immunodeficiency virus 1 (HIV-1))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50482857(CHEMBL1255915)

Ki: 8.10nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair

PDB
UniProtKB/TrEMBL
B.MOAD GoogleScholar

Details Article PubMed

Protease(Human immunodeficiency virus 1 (HIV-1))
Jadavpur University

Curated by ChEMBL

PNG

BDBM50482857(CHEMBL1255915)

Ki: 8.10nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair

PDB
UniProtKB/TrEMBL
B.MOAD GoogleScholar

Details Article PubMed

Displayed 1 to 50 (of 1516 total ) | Next | Last >>

Filter my 1516 hits

Targets 44▿
- 72 kDa type IV collagenase 309
- Matrix metalloproteinase-9 154
- Interstitial collagenase 89
- Histone deacetylase 3 86
- Replicase polyprotein 1ab 82
- Histone deacetylase 1 75
- Histone deacetylase 2 68
- Stromelysin-1 58
- Neutrophil collagenase 55
- Matrix metalloproteinase-14 53
- Kynurenine 3-monooxygenase 51
- Aminopeptidase N 47
- Histone deacetylase 8 45
- Collagenase 3 45
- Macrophage metalloelastase 42
- Matrilysin 39
- Protease 32
- Adenosine kinase 32
- Histone deacetylase 6 29
- Histone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2) 25
- Vascular endothelial growth factor receptor 2 15
- Epidermal growth factor receptor 13
- Polyamine deacetylase HDAC10 8
- Broad substrate specificity ATP-binding cassette transporter ABCG2 8
- Stromelysin-2 8
- Disintegrin and metalloproteinase domain-containing protein 17 7
- Platelet-derived growth factor receptor alpha/beta 5
- Glutamyl aminopeptidase 5
- Nuclear receptor corepressor 1 5
- Histone deacetylase 4 4
- Cytosol aminopeptidase 4
- Histone deacetylase 5 3
- Aromatase 2
- Proto-oncogene tyrosine-protein kinase Src 2
- Cytosol aminopeptidase [33-68,L62W] 2
- Cytosol aminopeptidase [435-519] 1
- Leukotriene A-4 hydrolase 1
- Histone deacetylase 1
- Aminopeptidase B 1
- M1 family aminopeptidase 1
- Matrix metalloproteinase-16 1
- Matrix metalloproteinase-15 1
- Matrix metalloproteinase-26 1
- Histone deacetylase 7 1
- ...
Publications 14▿
- J Med Chem 65: 10709-10754 (2022) 314
- Bioorg Med Chem 24: 4291-4309 (2016) 241
- Bioorg Med Chem 29: (2021) 70
- Eur J Med Chem 166: 369-380 (2019) 69
- J Med Chem 61: 6468-6490 (2018) 63
- Bioorg Med Chem Lett 26: 5712-5718 (2016) 51
- Eur J Med Chem 141: 37-50 (2017) 48
- Bioorg Med Chem Lett 20: 6082-7 (2010) 32
- Bioorg Med Chem Lett 12: 899-902 (2002) 32
- Eur J Med Chem 238: (2022) 31
- Eur J Med Chem 157: 1127-1142 (2018) 30
- Bioorg Med Chem 53: (2022) 30
- Eur J Med Chem 164: 214-240 (2019) 22
- Eur J Med Chem 241: (2022) 8
Institutions 4▿
- Jadavpur University 921
- Dr. Hari Singh Gour University 51
- Dr. Harisingh Gour University 38
- Birla Institute Of Technology And Science-Pilani Hyderabad Campus 31
Affinity: 0.010 to 5.0E+5 nM▿
- Ki 238
- IC50 1277
- Kd 1
- Affinity ≤ nM
Xtal structures: 18
Docked structures: 5
Catalog Cmpds: 95