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Found 69 with Last Name = 'johansen' and Initial = 'nl'
TargetNeurotensin receptor type 1(Rattus norvegicus)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50369070(CHEMBL1793839)
Affinity DataIC50:  5nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033671((S)-2-{(R)-2-[2-({1-[2-(2-Amino-5-guanidino-pentan...)
Affinity DataIC50:  8nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50240845((S)-2-{(2S,3R)-2-[(S)-2-({(S)-1-[(S)-2-((S)-2-Amin...)
Affinity DataIC50:  10nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033670((S)-2-[(R)-5-({1-[2-(2-Amino-5-guanidino-pentanoyl...)
Affinity DataIC50:  15nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033677((S,R)5-[1-{1-[2-[1-amino-4-amino(imino)methylamino...)
Affinity DataIC50:  120nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033667((S,S)2-{1-[2-{1-[2-[1-amino-4-amino(imino)methylam...)
Affinity DataIC50:  180nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT (neurotensin) as tracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033668((R,S)5-[1-{1-[2-[1-amino-4-amino(imino)methylamino...)
Affinity DataIC50:  900nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033678((S,S)5-[1-{1-[2-[1-amino-4-amino(imino)methylamino...)
Affinity DataIC50:  1.20E+3nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033675((S)-2-[(S)-5-({1-[2-(2-Amino-5-guanidino-pentanoyl...)
Affinity DataIC50:  1.20E+3nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033679((R,R)5-[1-{1-[2-[1-amino-4-amino(imino)methylamino...)
Affinity DataIC50:  1.50E+3nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50369071(CHEMBL1793838)
Affinity DataIC50:  6.31E+3nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50369072(CHEMBL1793837)
Affinity DataIC50:  8.00E+3nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033674((S,S)2-{1-[2-{1-[2-[1-amino-4-amino(imino)methylam...)
Affinity DataIC50:  1.00E+4nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT (neurotensin) as tracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066812((E)-5-Amino-5-methyl-hex-2-enoic acid ((R)-1-{[(R)...)
Affinity DataEC50:  8.90nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066809((E)-5-Amino-5-methyl-hex-2-enoic acid {(R)-2-benzo...)
Affinity DataEC50:  35nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066810((E)-5-Amino-5-methyl-hex-2-enoic acid {(R)-1-[((R)...)
Affinity DataEC50:  13nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066811((E)-5-Amino-5-methyl-hex-2-enoic acid {(R)-2-benzy...)
Affinity DataEC50:  5nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066812((E)-5-Amino-5-methyl-hex-2-enoic acid ((R)-1-{[(R)...)
Affinity DataEC50:  8.90nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066814((E)-5-Amino-5-methyl-hex-2-enoic acid [(R)-1-{[(R)...)
Affinity DataEC50:  6nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066813((E)-5-Amino-5-methyl-hex-2-enoic acid ((R)-1-{[(R)...)
Affinity DataEC50:  45nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066819((E)-5-Amino-5-methyl-hex-2-enoic acid {(R)-2-biphe...)
Affinity DataEC50:  3nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066816((E)-2-methyl-6-(methyl((R)-1-(methyl((R)-1-(methyl...)
Affinity DataEC50:  18nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066817((E)-5-Amino-5-methyl-hex-2-enoic acid ((R)-1-{[(R)...)
Affinity DataEC50:  5nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066818((E)-5-Amino-5-methyl-hex-2-enoic acid methyl-[(R)-...)
Affinity DataEC50:  21nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066820((E)-5-Amino-5-methyl-hex-2-enoic acid ((R)-1-{[(R)...)
Affinity DataEC50:  20nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066823((E)-5-Amino-5-methyl-hex-2-enoic acid ((R)-1-{[(R)...)
Affinity DataEC50:  17nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066822((E)-5-Amino-5-methyl-hex-2-enoic acid methyl-[(R)-...)
Affinity DataEC50:  16nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066821((E)-5-Amino-5-methyl-hex-2-enoic acid ((R)-1-{[(R)...)
Affinity DataEC50:  8nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066824((E)-5-Amino-5-methyl-hex-2-enoic acid methyl-{(R)-...)
Affinity DataEC50:  24nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066825((E)-5-Amino-5-methyl-hex-2-enoic acid [(R)-1-{[(R)...)
Affinity DataEC50:  1.5nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066826((E)-5-Amino-5-methyl-hex-2-enoic acid ((R)-1-{[(R)...)
Affinity DataEC50:  1.80nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50066827((E)-5-Amino-5-methyl-hex-2-enoic acid methyl-{(R)-...)
Affinity DataEC50:  2nMAssay Description:Tested for GH-releasing property using classical rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087749(CHEMBL261911 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  0.0360nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087726(CHEMBL409983 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  0.0540nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087758(CHEMBL409270 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  0.0270nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087738(CHEMBL412541 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  0.0360nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087728(CHEMBL412234 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  0.135nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087740(CHEMBL437467 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  0.328nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087732(CHEMBL424733 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  0.687nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087735(CHEMBL428152 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  0.00800nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087747(CHEMBL439305 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  61nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087730(CHEMBL427768 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  0.177nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087736(CHEMBL412948 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  0.0270nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087752(CHEMBL429398 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  0.0300nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087751(CHEMBL269543 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  0.0530nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087759(CHEMBL414971 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  0.0350nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087733(CHEMBL440075 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  7nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087741(CHEMBL266046 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  1.26nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087760(CHEMBL439091 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  0.210nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50087748(CHEMBL269494 | Glucagon like peptide-1(GLP-1)analo...)
Affinity DataEC50:  0.0840nMAssay Description:Potency measured using recombinant human GLP-1 receptor expressed in Baby Hamster Kidney (BHK)cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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