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Found 45 with Last Name = 'jubault' and Initial = 'p'
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313785((2S,4S,5R,6R)-5-acetamido-2-((2S,3R,4S,5S,6R)-2-((...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313791(3-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-3,4,5-trihydro...)
Affinity DataIC50:  2.50E+6nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313791(3-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-3,4,5-trihydro...)
Affinity DataIC50:  2.50E+6nMAssay Description:Inhibition of human recombinant P-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313788((S)-2-(2,2-difluoro-2-((2S,3S,4S,5S,6R)-3,4,5-trih...)
Affinity DataIC50:  3.00E+6nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313788((S)-2-(2,2-difluoro-2-((2S,3S,4S,5S,6R)-3,4,5-trih...)
Affinity DataIC50:  3.00E+6nMAssay Description:Inhibition of human recombinant P-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313787(3-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-2,3,4,5-tetrah...)
Affinity DataIC50:  5.00E+6nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313789(3-(2,2-difluoro-2-((2S,3S,4S,5S,6R)-3,4,5-trihydro...)
Affinity DataIC50:  5.00E+6nMAssay Description:Inhibition of human recombinant P-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313785((2S,4S,5R,6R)-5-acetamido-2-((2S,3R,4S,5S,6R)-2-((...)
Affinity DataIC50: >5.00E+6nMAssay Description:Inhibition of human recombinant P-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313789(3-(2,2-difluoro-2-((2S,3S,4S,5S,6R)-3,4,5-trihydro...)
Affinity DataIC50:  5.00E+6nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313792(CHEMBL1088214 | beta-mannosylglutamate)
Affinity DataIC50:  6.00E+6nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313787(3-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-2,3,4,5-tetrah...)
Affinity DataIC50:  6.50E+6nMAssay Description:Inhibition of human recombinant P-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313790((S)-2-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-3,4,5-trih...)
Affinity DataIC50:  1.10E+7nMAssay Description:Inhibition of human recombinant P-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313786((S)-2-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-2,3,4,5-te...)
Affinity DataIC50:  1.10E+7nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313786((S)-2-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-2,3,4,5-te...)
Affinity DataIC50:  1.10E+7nMAssay Description:Inhibition of human recombinant P-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313790((S)-2-(2,2-difluoro-2-((2R,3S,4S,5S,6R)-3,4,5-trih...)
Affinity DataIC50:  1.50E+7nMAssay Description:Inhibition of human recombinant E-Selectin assessed as inhibition of binding of HL-60 cells expressing tetrasaccharide sialyl Lewis x to selectin coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataEC50:  1.83E+4nMAssay Description:Agonist activity at rat mGluR2 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataEC50:  1.26E+4nMAssay Description:Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataEC50:  8.22E+4nMAssay Description:Agonist activity at rat mGluR6 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at rat mGluR7 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataEC50:  2.15E+4nMAssay Description:Agonist activity at rat mGluR8 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataEC50:  2.32E+4nMAssay Description:Agonist activity at rat mGluR1 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataEC50:  1.37E+4nMAssay Description:Agonist activity at rat mGluR5 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataEC50:  2.88E+3nMAssay Description:Agonist activity at rat mGlu4 receptor expressed in HEK293 cells coexpressing Gq/Gi and EAAC1 assessed as intracellular calcium production measured e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at rat mGlu4 receptor expressed in HEK293 cells coexpressing Gq/Gi and EAAC1 assessed as intracellular calcium production measured e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50387817(CHEMBL2058378)
Affinity DataEC50:  340nMAssay Description:Agonist activity at rat mGlu4 receptor expressed in HEK293 cells coexpressing Gq/Gi and EAAC1 assessed as intracellular calcium production measured e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50387818(CHEMBL2058379)
Affinity DataEC50:  6.09E+5nMAssay Description:Agonist activity at rat mGlu4 receptor expressed in HEK293 cells coexpressing Gq/Gi and EAAC1 assessed as intracellular calcium production measured e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50387819(CHEMBL2058380)
Affinity DataEC50:  4.65E+5nMAssay Description:Agonist activity at rat mGlu4 receptor expressed in HEK293 cells coexpressing Gq/Gi and EAAC1 assessed as intracellular calcium production measured e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50387820(CHEMBL2058381)
Affinity DataEC50:  8.56E+4nMAssay Description:Agonist activity at rat mGlu4 receptor expressed in HEK293 cells coexpressing Gq/Gi and EAAC1 assessed as intracellular calcium production measured e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50387821(CHEMBL2058382)
Affinity DataEC50:  2.74E+4nMAssay Description:Agonist activity at rat mGlu4 receptor expressed in HEK293 cells coexpressing Gq/Gi and EAAC1 assessed as intracellular calcium production measured e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)
Affinity DataEC50:  120nMAssay Description:Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)
Affinity DataEC50:  100nMAssay Description:Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)
Affinity DataEC50:  120nMAssay Description:Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)
Affinity DataEC50:  1.13E+4nMAssay Description:Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)
Affinity DataEC50:  300nMAssay Description:Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)
Affinity DataEC50:  1.25E+3nMAssay Description:Agonist activity at rat mGluR8 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at rat mGluR7 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)
Affinity DataEC50:  6.01E+3nMAssay Description:Agonist activity at rat mGluR6 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)
Affinity DataEC50:  300nMAssay Description:Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at rat mGluR2 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50217031((1S,2R)-1-amino-2-phosphonomethylcyclopropane-carb...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Affinity DataEC50:  110nMAssay Description:Agonist activity at rat mGluR8 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Affinity DataEC50:  4.26E+5nMAssay Description:Agonist activity at rat mGluR7 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50387822(CHEMBL2058383)
Affinity DataEC50:  1.40E+6nMAssay Description:Agonist activity at rat mGlu4 receptor expressed in HEK293 cells coexpressing Gq/Gi and EAAC1 assessed as intracellular calcium production measured e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Affinity DataEC50:  3.45E+3nMAssay Description:Agonist activity at rat mGluR6 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed