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Found 150 with Last Name = 'juliano' and Initial = 'l'
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50505323(CHEMBL4556848)
Affinity DataKi:  2nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50505321(CHEMBL2402091)
Affinity DataKi:  8nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50396164(CHEMBL2171751)
Affinity DataKi:  8nMAssay Description:Inhibition of human KLK1 using Pro-Phe-Arg-MCA as substrate for 2 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50505321(CHEMBL2402091)
Affinity DataKi:  33nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112584(2-(2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylami...)
Affinity DataKi:  50nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50396166(CHEMBL2171749)
Affinity DataKi:  50nMAssay Description:Inhibition of human KLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50298759((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi:  65nMAssay Description:Inhibition of human KLK3 using Mu-SRKSQQY-AMC as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50229129(4-Methyl-piperazine-1-carboxylic acid [(S)-1-((E)-...)
Affinity DataKi:  80nMAssay Description:Irreversible inhibition of human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50370072(CHEMBL1790422)
Affinity DataKi:  100nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50396165(CHEMBL2171750)
Affinity DataKi:  110nMAssay Description:Inhibition of human KLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112580(CHEMBL268148 | PWGF(CH2NH)WWFW)
Affinity DataKi:  200nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50229129(4-Methyl-piperazine-1-carboxylic acid [(S)-1-((E)-...)
Affinity DataKi:  220nMAssay Description:Irreversible inhibition of Trypanosoma cruzi cruzipainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50229129(4-Methyl-piperazine-1-carboxylic acid [(S)-1-((E)-...)
Affinity DataKi:  270nMAssay Description:Irreversible inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446220(CHEMBL3109164)
Affinity DataKi:  300nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50396162(CHEMBL2171878)
Affinity DataKi:  300nMAssay Description:Inhibition of KLK3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50229129(4-Methyl-piperazine-1-carboxylic acid [(S)-1-((E)-...)
Affinity DataKi:  390nMAssay Description:Irreversible inhibition of human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446221(CHEMBL3109163)
Affinity DataKi:  400nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112597(2-{2-[2-(2-{2-[2-[2-(2-Amino-3-carboxy-propionylam...)
Affinity DataKi:  500nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50396161(CHEMBL2171879)
Affinity DataKi:  500nMAssay Description:Inhibition of KLK3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112581(6-Amino-2-(2-{2-[2-(6-amino-2-{2-[6-amino-2-(2-ami...)
Affinity DataKi:  600nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446218(CHEMBL3109166)
Affinity DataKi:  600nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50505323(CHEMBL4556848)
Affinity DataKi:  690nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446219(CHEMBL3109165)
Affinity DataKi:  700nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112596(6-Amino-2-{2-[2-(2-{2-[2-[6-amino-2-(2-amino-3-car...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112594(CHEMBL266692 | ChaALF(CH2NH)YMYY)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446218(CHEMBL3109166)
Affinity DataKi:  1.30E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446219(CHEMBL3109165)
Affinity DataKi:  1.40E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50396163(CHEMBL2171880)
Affinity DataKi:  1.41E+3nMAssay Description:Inhibition of human KLK2 after 1 hr by phage-display based Immunofluorometric AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50292533(CHEMBL446790 | Fukugetin)
Affinity DataKi:  1.60E+3nMAssay Description:Mixed-type inhibition of human tissue kallikrein-2 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446228(CHEMBL3109061)
Affinity DataKi:  1.70E+3nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446227(CHEMBL3109056)
Affinity DataKi:  1.80E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50391075(CHEMBL2087343)
Affinity DataKi:  1.80E+3nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446220(CHEMBL3109164)
Affinity DataKi:  1.90E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446224(CHEMBL3109160)
Affinity DataKi:  2.30E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446211(CHEMBL3109058)
Affinity DataKi:  2.40E+3nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446228(CHEMBL3109061)
Affinity DataKi:  2.40E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446224(CHEMBL3109160)
Affinity DataKi:  2.40E+3nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446221(CHEMBL3109163)
Affinity DataKi:  2.80E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446211(CHEMBL3109058)
Affinity DataKi:  2.90E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50391078(CHEMBL2087346)
Affinity DataKi:  3.00E+3nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446229(CHEMBL3109060)
Affinity DataKi:  3.40E+3nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50292533(CHEMBL446790 | Fukugetin)
Affinity DataKi:  3.60E+3nMAssay Description:Mixed-type inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446229(CHEMBL3109060)
Affinity DataKi:  3.80E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50446230(CHEMBL3109059)
Affinity DataKi:  4.40E+3nMAssay Description:Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112583(1-{2-[2-[2-(6-Amino-2-{2-[2-(2-amino-3-methyl-pent...)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112579(6-Amino-2-(2-{2-[2-(6-amino-2-{2-[2-(2-amino-3-cyc...)
Affinity DataKi:  6.30E+3nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112591(2-(2-{2-[2-(2-{2-[2-(2-Amino-4-methylsulfanyl-buty...)
Affinity DataKi:  6.50E+3nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112585(2-[3-Cyclohexyl-2-(2-{2-[2-(3-(3H-imidazol-4-yl)-2...)
Affinity DataKi:  6.60E+3nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50112582(6-Amino-2-[2-(2-{2-[2-(2-{6-amino-2-[(pyrrolidine-...)
Affinity DataKi:  8.80E+3nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Carlsberg Laboratory

Curated by ChEMBL
LigandPNGBDBM50370073(CHEMBL1790421)
Affinity DataKi:  1.01E+4nMAssay Description:Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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