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Found 59 with Last Name = 'junager' and Initial = 'f'
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118351((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  3nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118349((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  120nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118348((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  180nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118360(CHEMBL336586 | tert-Butyl-(2-chloro-7,7-dioxo-4,7-...)
Affinity DataIC50:  230nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118359((2-Chloro-7,7-dioxo-4,7-dihydro-1,7-dithia-4,6-dia...)
Affinity DataIC50:  320nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118343((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  340nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50023475(CHEMBL2111887)
Affinity DataIC50:  640nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118355((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  2.27E+3nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at high...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118351((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at low ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107950((RS)-2-amino-3-(1-hydroxy-1,2,3-triazol-5-yl)propi...)
Affinity DataIC50:  1.00E+5nMAssay Description:Binding affinity for Excitatory amino acid transporter 1 (EAAT-1) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118349((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  1.46E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at low ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118359((2-Chloro-7,7-dioxo-4,7-dihydro-1,7-dithia-4,6-dia...)
Affinity DataIC50:  1.65E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at low ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118343((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  1.87E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at low ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM86248(CAS_364-98-7 | NSC_3019 | diazoxide)
Affinity DataIC50:  1.98E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at low ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50023475(CHEMBL2111887)
Affinity DataIC50:  2.24E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at low ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107954(2-Amino-3-(3-hydroxy-isoxazol-4-yl)-propionic acid...)
Affinity DataIC50:  2.40E+5nMAssay Description:Binding affinity for Excitatory amino acid transporter 2 (EAAT-2) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107954(2-Amino-3-(3-hydroxy-isoxazol-4-yl)-propionic acid...)
Affinity DataIC50:  2.70E+5nMAssay Description:Binding affinity for Excitatory amino acid transporter 1 (EAAT-1) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107950((RS)-2-amino-3-(1-hydroxy-1,2,3-triazol-5-yl)propi...)
Affinity DataIC50:  3.00E+5nMAssay Description:Binding affinity for Excitatory amino acid transporter 2 (EAAT-2) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118348((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  3.75E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at low ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118360(CHEMBL336586 | tert-Butyl-(2-chloro-7,7-dioxo-4,7-...)
Affinity DataIC50:  3.93E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at low ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107948(2-Amino-3-(2-hydroxy-2H-pyrazol-3-yl)-propionic ac...)
Affinity DataIC50:  4.30E+5nMAssay Description:Binding affinity for Excitatory amino acid transporter 2 (EAAT-2) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50023475(CHEMBL2111887)
Affinity DataIC50:  4.87E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 without...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107949(2-Amino-3-(3-hydroxy-5-methyl-3H-[1,2,3]triazol-4-...)
Affinity DataIC50:  4.90E+5nMAssay Description:Binding affinity for Excitatory amino acid transporter 2 (EAAT-2) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118343((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  5.54E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 without...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118355((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  5.84E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 at low ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118359((2-Chloro-7,7-dioxo-4,7-dihydro-1,7-dithia-4,6-dia...)
Affinity DataIC50:  6.85E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 without...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM86248(CAS_364-98-7 | NSC_3019 | diazoxide)
Affinity DataIC50:  7.50E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 without...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118351((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  8.59E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 without...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118348((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  8.99E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 without...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118355((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  9.24E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 without...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11(Homo sapiens (Human))
Novo Nordisk Research And Development

Curated by ChEMBL
LigandPNGBDBM50118349((2-Chloro-7,7-dioxo-4,7-dihydro-1,7lambda*6*-dithi...)
Affinity DataIC50:  9.43E+5nMAssay Description:Inhibition of [3H]glibenclamide binding to HEK293 cells co-expressing human Sulfonylurea receptor SUR1 and Inward rectifier K+ channel Kir6.2 without...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107950((RS)-2-amino-3-(1-hydroxy-1,2,3-triazol-5-yl)propi...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 3 (EAAT-3) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107952(2-Amino-3-(3-hydroxy-2-methyl-3H-imidazol-4-yl)-pr...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 1 (EAAT-1) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107953(2-Amino-3-(3-hydroxy-5-methyl-3H-imidazol-4-yl)-pr...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 2 (EAAT-2) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107946(2-Amino-3-(3-hydroxy-3H-imidazol-4-yl)-propionic a...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 3 (EAAT-3) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107949(2-Amino-3-(3-hydroxy-5-methyl-3H-[1,2,3]triazol-4-...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 3 (EAAT-3) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107947(2-Amino-3-(1-hydroxy-5-methyl-1H-imidazol-2-yl)-pr...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 1 (EAAT-1) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107955(2-Amino-3-(1-hydroxy-1H-imidazol-2-yl)-propionic a...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 1 (EAAT-1) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50002370((R,S)-alpha-amino-3-hydroxy-5-methyl-4-isooxazole-...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 1 (EAAT-1) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107948(2-Amino-3-(2-hydroxy-2H-pyrazol-3-yl)-propionic ac...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 1 (EAAT-1) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107952(2-Amino-3-(3-hydroxy-2-methyl-3H-imidazol-4-yl)-pr...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 3 (EAAT-3) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107947(2-Amino-3-(1-hydroxy-5-methyl-1H-imidazol-2-yl)-pr...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 3 (EAAT-3) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107953(2-Amino-3-(3-hydroxy-5-methyl-3H-imidazol-4-yl)-pr...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 3 (EAAT-3) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107946(2-Amino-3-(3-hydroxy-3H-imidazol-4-yl)-propionic a...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 2 (EAAT-2) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107946(2-Amino-3-(3-hydroxy-3H-imidazol-4-yl)-propionic a...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 1 (EAAT-1) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107951(2-Amino-3-(2-hydroxy-4-methyl-2H-pyrazol-3-yl)-pro...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 2 (EAAT-2) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50002370((R,S)-alpha-amino-3-hydroxy-5-methyl-4-isooxazole-...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 2 (EAAT-2) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107948(2-Amino-3-(2-hydroxy-2H-pyrazol-3-yl)-propionic ac...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 3 (EAAT-3) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107953(2-Amino-3-(3-hydroxy-5-methyl-3H-imidazol-4-yl)-pr...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 1 (EAAT-1) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50107955(2-Amino-3-(1-hydroxy-1H-imidazol-2-yl)-propionic a...)
Affinity DataIC50: >1.00E+6nMAssay Description:Binding affinity for Excitatory amino acid transporter 3 (EAAT-3) in Glu uptake systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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