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Found 44 with Last Name = 'kaiser' and Initial = 'sm'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50366574(CHEMBL609646)
Affinity DataKi:  610nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain using [3H]R-PIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50366575(CHEMBL609645)
Affinity DataKi:  1.02E+3nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain using [3H]R-PIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50366573(CHEMBL607912)
Affinity DataKi:  3.82E+3nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain using [3H]R-PIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50366572(CHEMBL607911)
Affinity DataKi:  4.54E+3nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain using [3H]R-PIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59162(8047577)
Affinity DataIC50:  2.10E+3nMpH: 7.9Assay Description:Inhibition of factor X activation assay. A commercially available chromogenic assay that measures the rate of factor X activation to measure inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59159(6190013)
Affinity DataIC50:  2.11E+3nMpH: 8.0Assay Description:Inhibition of factor VIII ELISA. The interaction between factor VIII and PS was measured by using an enzyme-linked immunoadsorbent assay (ELISA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59162(8047577)
Affinity DataIC50:  2.44E+3nMT: 2°CAssay Description:Inhibition of factor VIII C2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59162(8047577)
Affinity DataIC50:  2.56E+3nMpH: 8.0Assay Description:Inhibition of factor VIII ELISA. The interaction between factor VIII and PS was measured by using an enzyme-linked immunoadsorbent assay (ELISA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59164(8048422)
Affinity DataIC50:  3.89E+3nMpH: 8.0Assay Description:Inhibition of factor VIII ELISA. The interaction between factor VIII and PS was measured by using an enzyme-linked immunoadsorbent assay (ELISA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59164(8048422)
Affinity DataIC50:  4.17E+3nMT: 2°CAssay Description:Inhibition of factor VIII C2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59154(5739991)
Affinity DataIC50:  4.63E+3nMT: 2°CAssay Description:Inhibition of factor VIII C2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59163(6789536)
Affinity DataIC50:  4.81E+3nMpH: 8.0Assay Description:Inhibition of factor VIII ELISA. The interaction between factor VIII and PS was measured by using an enzyme-linked immunoadsorbent assay (ELISA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59161(5738875)
Affinity DataIC50:  5.00E+3nMpH: 7.9Assay Description:Inhibition of factor X activation assay. A commercially available chromogenic assay that measures the rate of factor X activation to measure inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59163(6789536)
Affinity DataIC50:  5.60E+3nMpH: 7.9Assay Description:Inhibition of factor X activation assay. A commercially available chromogenic assay that measures the rate of factor X activation to measure inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59161(5738875)
Affinity DataIC50:  5.65E+3nMT: 2°CAssay Description:Inhibition of factor VIII C2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59163(6789536)
Affinity DataIC50:  5.85E+3nMT: 2°CAssay Description:Inhibition of factor VIII C2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59165(8056354)
Affinity DataIC50:  6.29E+3nMT: 2°CAssay Description:Inhibition of factor VIII C2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59165(8056354)
Affinity DataIC50:  6.51E+3nMpH: 8.0Assay Description:Inhibition of factor VIII ELISA. The interaction between factor VIII and PS was measured by using an enzyme-linked immunoadsorbent assay (ELISA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59153(5737176)
Affinity DataIC50:  6.66E+3nMT: 2°CAssay Description:Inhibition of factor VIII C2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59164(8048422)
Affinity DataIC50:  6.70E+3nMpH: 7.9Assay Description:Inhibition of factor X activation assay. A commercially available chromogenic assay that measures the rate of factor X activation to measure inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59165(8056354)
Affinity DataIC50:  6.80E+3nMpH: 7.9Assay Description:Inhibition of factor X activation assay. A commercially available chromogenic assay that measures the rate of factor X activation to measure inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59161(5738875)
Affinity DataIC50:  6.83E+3nMpH: 8.0Assay Description:Inhibition of factor VIII ELISA. The interaction between factor VIII and PS was measured by using an enzyme-linked immunoadsorbent assay (ELISA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59159(6190013)
Affinity DataIC50:  7.50E+3nMpH: 7.9Assay Description:Inhibition of factor X activation assay. A commercially available chromogenic assay that measures the rate of factor X activation to measure inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59159(6190013)
Affinity DataIC50:  8.48E+3nMT: 2°CAssay Description:Inhibition of factor VIII C2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59153(5737176)
Affinity DataIC50:  8.50E+3nMpH: 7.9Assay Description:Inhibition of factor X activation assay. A commercially available chromogenic assay that measures the rate of factor X activation to measure inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59153(5737176)
Affinity DataIC50:  9.25E+3nMpH: 8.0Assay Description:Inhibition of factor VIII ELISA. The interaction between factor VIII and PS was measured by using an enzyme-linked immunoadsorbent assay (ELISA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59154(5739991)
Affinity DataIC50:  1.04E+4nMpH: 8.0Assay Description:Inhibition of factor VIII ELISA. The interaction between factor VIII and PS was measured by using an enzyme-linked immunoadsorbent assay (ELISA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59154(5739991)
Affinity DataIC50:  1.17E+4nMpH: 7.9Assay Description:Inhibition of factor X activation assay. A commercially available chromogenic assay that measures the rate of factor X activation to measure inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59157(6126765)
Affinity DataIC50:  1.19E+4nMT: 2°CAssay Description:Inhibition of factor VIII C2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59160(6209549)
Affinity DataIC50:  1.24E+4nMT: 2°CAssay Description:Inhibition of factor VIII C2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59155(5924029)
Affinity DataIC50:  2.45E+4nMT: 2°CAssay Description:Inhibition of factor VIII C2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59156(6072484 | cid_726942)
Affinity DataIC50:  2.68E+4nMT: 2°CAssay Description:Inhibition of factor VIII C2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59152(5523453)
Affinity DataIC50:  2.77E+4nMT: 2°CAssay Description:Inhibition of factor VIII C2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59158(6168356)
Affinity DataIC50:  4.96E+4nMT: 2°CAssay Description:Inhibition of factor VIII C2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VIII(Homo sapiens (Human))
University of Washington

LigandPNGBDBM59151(5247489)
Affinity DataIC50:  5.61E+4nMT: 2°CAssay Description:Inhibition of factor VIII C2 domain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50069320((2S,3S,4S,5S)-2-(6-Amino-purin-9-yl)-5-(1-methyl-1...)
Affinity DataEC50:  1.23E+3nMAssay Description:[S]GTP gamma-S binding against adenosine A1 receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50069319((2R,3R,4S,5R)-2-(6-Amino-purin-9-yl)-5-(1-methyl-1...)
Affinity DataEC50:  28nMAssay Description:Binding against human adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataEC50:  59nMAssay Description:Binding against human adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Griffith University

Curated by ChEMBL
LigandPNGBDBM35804((CGS21680) 3-(4-{2-[6-Amino-9-(5-ethylcarbamoylmet...)
Affinity DataEC50: >100nMAssay Description:[S]GTP gamma-S binding against adenosine A1 receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Griffith University

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataEC50:  87nMAssay Description:[S]GTP gamma-S binding against adenosine A1 receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50366575(CHEMBL609645)
Affinity DataEC50:  1.00E+5nMAssay Description:Binding against Human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50069320((2S,3S,4S,5S)-2-(6-Amino-purin-9-yl)-5-(1-methyl-1...)
Affinity DataEC50:  869nMAssay Description:Binding against human adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50069319((2R,3R,4S,5R)-2-(6-Amino-purin-9-yl)-5-(1-methyl-1...)
Affinity DataEC50:  17nMAssay Description:[S]GTP gamma-S binding against adenosine A1 receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM35804((CGS21680) 3-(4-{2-[6-Amino-9-(5-ethylcarbamoylmet...)
Affinity DataEC50:  6.44E+3nMAssay Description:Binding against human adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed