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Found 158 with Last Name = 'kashimoto' and Initial = 's'
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM465744(2-{3-[2-amino-6-(pyridin-4-yl)-7H- pyrrolo[2,3-d]p...)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of human BTK-A using phosphorylated substrate in presence of ATP by microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)
Affinity DataIC50:  0.210nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468314(2-{3-[2-amino-6- (1,1-dioxido-3,6- dihydro-2H- thi...)
Affinity DataIC50:  0.25nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM465733(2-[3-(2-amino-6-{4-[(4-methylpiperazin- 1-yl)methy...)
Affinity DataIC50:  0.330nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468318(2-(3-{2-amino-6-[1- (methylsulfonyl)- 1,2,3,6- tet...)
Affinity DataIC50:  0.340nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468311(2-{3-[2-amino-6-(4- {[4-(2-hydroxy- ethyl)piperazi...)
Affinity DataIC50:  0.360nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468313(2-(3-{2-amino-6- [1-(4-methylpiperazine-1- carbony...)
Affinity DataIC50:  0.390nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468315(2-{3-[2-amino-6- (1-propionyl-1,2,3,6- tetrahydrop...)
Affinity DataIC50:  0.410nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468320(2-{3-[2-amino-6-(1,2,3,6- tetrahydropyridin-4-yl)-...)
Affinity DataIC50:  0.410nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM465733(2-[3-(2-amino-6-{4-[(4-methylpiperazin- 1-yl)methy...)
Affinity DataIC50:  0.430nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468308(2-[3-(2-amino-6-{4- [(diethyl- amino)methyl]phenyl...)
Affinity DataIC50:  0.430nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468307(2-[3-(2-amino-6-{4- [(dimethyl- amino)methyl]pheny...)
Affinity DataIC50:  0.430nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM465748(2-(3-{2-amino-6-[1-(oxetan-3-yl)-1,2,3,6-tetrahydr...)
Affinity DataIC50:  0.460nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468312(2-[3-(2-amino-6-{4- [(3-oxopiperazin-1- yl)methyl]...)
Affinity DataIC50:  0.470nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468319(2-{3-[2-amino-6-(1- ethyl-1,2,3,6- tetrahydropyrid...)
Affinity DataIC50:  0.470nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM465738(2-{3-[2-amino-6-(1-methyl-1H-pyrazol- 4-yl)-7H-pyr...)
Affinity DataIC50:  0.490nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468309(2-(3-{2-amino-6-[4- (pyrrolidin-1- ylmethyl)phenyl...)
Affinity DataIC50:  0.510nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468316(4-{2-amino-4-[3- (6-cyclopropyl-8- fluoro-1-oxoiso...)
Affinity DataIC50:  0.520nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468316(4-{2-amino-4-[3- (6-cyclopropyl-8- fluoro-1-oxoiso...)
Affinity DataIC50:  0.540nMAssay Description:Inhibition of human BTK-A using phosphorylated substrate in presence of ATP by microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM468311(2-{3-[2-amino-6-(4- {[4-(2-hydroxy- ethyl)piperazi...)
Affinity DataIC50:  0.570nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM468313(2-(3-{2-amino-6- [1-(4-methylpiperazine-1- carbony...)
Affinity DataIC50:  0.580nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468310(2-(3-{2-amino-6-[4- (piperidin-1- ylmethyl)phenyl]...)
Affinity DataIC50:  0.580nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468313(2-(3-{2-amino-6- [1-(4-methylpiperazine-1- carbony...)
Affinity DataIC50:  0.580nMAssay Description:Inhibition of human BTK C481S mutant using phosphorylated substrate in presence of ATP by microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM468314(2-{3-[2-amino-6- (1,1-dioxido-3,6- dihydro-2H- thi...)
Affinity DataIC50:  0.580nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM465738(2-{3-[2-amino-6-(1-methyl-1H-pyrazol- 4-yl)-7H-pyr...)
Affinity DataIC50:  0.600nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468320(2-{3-[2-amino-6-(1,2,3,6- tetrahydropyridin-4-yl)-...)
Affinity DataIC50:  0.650nMAssay Description:Inhibition of human BTK-A using phosphorylated substrate in presence of ATP by microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468313(2-(3-{2-amino-6- [1-(4-methylpiperazine-1- carbony...)
Affinity DataIC50:  0.650nMAssay Description:Inhibition of human BTK-A using phosphorylated substrate in presence of ATP by microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50586595(CHEMBL5083974)
Affinity DataIC50:  0.690nMAssay Description:Inhibition of human BTK-A using phosphorylated substrate in presence of ATP by microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM468318(2-(3-{2-amino-6-[1- (methylsulfonyl)- 1,2,3,6- tet...)
Affinity DataIC50:  0.700nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50586593(CHEMBL5076374)
Affinity DataIC50:  0.710nMAssay Description:Inhibition of human BTK-A using phosphorylated substrate in presence of ATP by microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM465766(2-(3-{2-amino-6-[4- (methylsulfonyl)phenyl]- 7H-py...)
Affinity DataIC50:  0.730nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM468308(2-[3-(2-amino-6-{4- [(diethyl- amino)methyl]phenyl...)
Affinity DataIC50:  0.760nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468306(2-(3-{2-amino-6-[2- (methylamino)pyridin- 4-yl]-7H...)
Affinity DataIC50:  0.770nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM468307(2-[3-(2-amino-6-{4- [(dimethyl- amino)methyl]pheny...)
Affinity DataIC50:  0.780nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM468315(2-{3-[2-amino-6- (1-propionyl-1,2,3,6- tetrahydrop...)
Affinity DataIC50:  0.820nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM465748(2-(3-{2-amino-6-[1-(oxetan-3-yl)-1,2,3,6-tetrahydr...)
Affinity DataIC50:  0.850nMAssay Description:Inhibition of human BTK-A using phosphorylated substrate in presence of ATP by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM468310(2-(3-{2-amino-6-[4- (piperidin-1- ylmethyl)phenyl]...)
Affinity DataIC50:  0.860nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM465767(2-{3-[2-amino-6-(6- fluoropyridin-2-yl)-7H- pyrrol...)
Affinity DataIC50:  0.870nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM468309(2-(3-{2-amino-6-[4- (pyrrolidin-1- ylmethyl)phenyl...)
Affinity DataIC50:  0.900nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM468312(2-[3-(2-amino-6-{4- [(3-oxopiperazin-1- yl)methyl]...)
Affinity DataIC50:  0.930nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468317(2-(3-{2-amino-6-[1- (pyrrolidine-1-carbonyl)- 1,2,...)
Affinity DataIC50:  0.940nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM468316(4-{2-amino-4-[3- (6-cyclopropyl-8- fluoro-1-oxoiso...)
Affinity DataIC50:  0.950nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468316(4-{2-amino-4-[3- (6-cyclopropyl-8- fluoro-1-oxoiso...)
Affinity DataIC50:  0.950nMAssay Description:Inhibition of human BTK C481S mutant using phosphorylated substrate in presence of ATP by microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM465727(2-[3-(2-amino-8-phenyl-9H-purin-6-yl)-2-(hydroxyme...)
Affinity DataIC50:  0.970nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trade mark) MSA (commercially available kit manufactured by Carna Biosciences, In...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM465727(2-[3-(2-amino-8-phenyl-9H-purin-6-yl)-2-(hydroxyme...)
Affinity DataIC50:  0.990nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)
Affinity DataIC50:  0.990nMAssay Description:Inhibition of BTK in human Ramos cells assessed as reduction of IgM stimulated PLCgamma2 (Y1217) phosphorylation after 24 hrs by western blot assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM465748(2-(3-{2-amino-6-[1-(oxetan-3-yl)-1,2,3,6-tetrahydr...)
Affinity DataIC50:  0.990nMAssay Description:Inhibition of human BTK C481S mutant using phosphorylated substrate in presence of ATP by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM468320(2-{3-[2-amino-6-(1,2,3,6- tetrahydropyridin-4-yl)-...)
Affinity DataIC50:  0.990nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM468320(2-{3-[2-amino-6-(1,2,3,6- tetrahydropyridin-4-yl)-...)
Affinity DataIC50:  0.990nMAssay Description:Inhibition of human BTK C481S mutant using phosphorylated substrate in presence of ATP by microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Carna Biosciences

US Patent
LigandPNGBDBM465748(2-(3-{2-amino-6-[1-(oxetan-3-yl)-1,2,3,6-tetrahydr...)
Affinity DataIC50:  0.990nMAssay Description:The kinase activity was measured using QuickScout Screening Assist (trademark) MSA (commercially available kit manufactured by Carna Biosciences, Inc...More data for this Ligand-Target Pair
In DepthDetails US Patent
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