Affinity DataKi: 0.300nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 138nMAssay Description:Inhibition of human LCK using peptide poly[Glu:Tyr] (4:1) substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
University Of South Florida
Curated by ChEMBL
University Of South Florida
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of human TYK2 using KKSRGDYMTMQIG peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human LCK using peptide poly[Glu:Tyr] (4:1) substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
University Of South Florida
Curated by ChEMBL
University Of South Florida
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of human JAK2 using poly[Glu:Tyr] (4:1) peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of ACK1 kinase (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 85nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 95nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 99nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 106nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 122nMAssay Description:Inhibition of human LCK using peptide poly[Glu:Tyr] (4:1) substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
University Of South Florida
Curated by ChEMBL
University Of South Florida
Curated by ChEMBL
Affinity DataIC50: 124nMAssay Description:Inhibition of human ROS/ROS1 using KKKSPGEYVNIEFG peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 136nMAssay Description:Inhibition of human LCK using peptide poly[Glu:Tyr] (4:1) substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
University Of South Florida
Curated by ChEMBL
University Of South Florida
Curated by ChEMBL
Affinity DataIC50: 143nMAssay Description:Inhibition of human ALK using poly[Glu:Tyr] (4:1) peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
University Of South Florida
Curated by ChEMBL
University Of South Florida
Curated by ChEMBL
Affinity DataIC50: 154nMAssay Description:Inhibition of human CHK1 using KKKVSRSGLYRSPSMPENLNRPR peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
University Of South Florida
Curated by ChEMBL
University Of South Florida
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of human FGFR1 using KKKSPGEYVNIEFG peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 164nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 169nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University Of South Florida
Curated by ChEMBL
University Of South Florida
Curated by ChEMBL
Affinity DataIC50: 206nMAssay Description:Inhibition of human ABL1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 231nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 299nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of South Florida
Curated by ChEMBL
University Of South Florida
Curated by ChEMBL
Affinity DataIC50: 438nMAssay Description:Inhibition of human c-Src using poly[Glu:Tyr] (4:1) peptide substrate by 33P Hotspot assayMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 6nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair