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Found 117 with Last Name = 'kim' and Initial = 'yj'
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379308(CHEMBL2011816)
Affinity DataKi:  4.40nMAssay Description:Displacement of [125I]Ghrelin from human GHSR1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast cell carboxypeptidase A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281176((S)-2-Mercaptomethyl-3-phenyl-propionic acid | 2-T...)
Affinity DataKi:  7.80nMAssay Description:Compound was tested for inhibitory activity against carboxypeptidase AMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50085045(5-((4-((6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-...)
Affinity DataKi:  400nMAssay Description:Binding affinity to human recombinant PPARgamma by Cheng-Prusoff equation based competitive binding TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM24566(2-({4-chloro-6-[(2,3-dimethylphenyl)amino]pyrimidi...)
Affinity DataKi:  4.50E+3nMAssay Description:Binding affinity to human recombinant PPARalpha by Cheng-Prusoff equation based competitive binding TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50548252(CHEMBL4765137)
Affinity DataKi:  6.70E+3nMAssay Description:Binding affinity to human recombinant PPARgamma by Cheng-Prusoff equation based competitive binding TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50548251(CHEMBL4797877)
Affinity DataKi:  7.00E+3nMAssay Description:Binding affinity to human recombinant PPARgamma by Cheng-Prusoff equation based competitive binding TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50548252(CHEMBL4765137)
Affinity DataKi:  8.00E+3nMAssay Description:Binding affinity to human recombinant PPARalpha by Cheng-Prusoff equation based competitive binding TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50548251(CHEMBL4797877)
Affinity DataKi:  9.50E+3nMAssay Description:Binding affinity to human recombinant PPARalpha by Cheng-Prusoff equation based competitive binding TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379328(CHEMBL2011825)
Affinity DataIC50:  0.200nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379309(CHEMBL2011826)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379312(CHEMBL2011892)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379320(CHEMBL2011834)
Affinity DataIC50:  2.5nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379322(CHEMBL2011832)
Affinity DataIC50:  2.5nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379310(CHEMBL2011894)
Affinity DataIC50:  3nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379334(CHEMBL2011819)
Affinity DataIC50:  3nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379319(CHEMBL2011835)
Affinity DataIC50:  4.10nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379314(CHEMBL2011890)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Chung-Ang University

Curated by ChEMBL
LigandPNGBDBM50121975((6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2...)
Affinity DataIC50: <6nMAssay Description:Inhibition of CYP2D6 in human liver microsomeMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379308(CHEMBL2011816)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at mouse GHSR1 receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379311(CHEMBL2011893)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379335(CHEMBL2011818)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379323(CHEMBL2011831)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50153547(3-(2,6-Dichloro-phenyl)-5-[2-(2-oxo-piperidin-1-yl...)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as blockade of intracellular Ca2+ mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379308(CHEMBL2011816)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379336(CHEMBL2011817)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379326(CHEMBL2011828)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 142(Mus musculus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50395775(CHEMBL2164857)
Affinity DataIC50:  15nMAssay Description:Partial agonist activity at mouse GPR142 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50158327((+/-)isobutyl 2-((4-(diethylamino)phenyl)carbamoyl...)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as blockade of intracellular Ca2+ mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379321(CHEMBL2011833)
Affinity DataIC50:  16.5nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379313(CHEMBL2011891)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379331(CHEMBL2011822)
Affinity DataIC50:  26nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379332(CHEMBL2011821)
Affinity DataIC50:  28nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379317(CHEMBL2011887)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Chung-Ang University

Curated by ChEMBL
LigandPNGBDBM31768(CHEMBL295698 | Ketoconazole | Nizoral | Panfungol)
Affinity DataIC50: <62nMAssay Description:Inhibition of CYP3A4 in human liver microsomeMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50435297(CHEMBL2393244)
Affinity DataIC50:  63nMAssay Description:Displacement of [3H]-methylspiperone from dopamine D2L receptor (unknown origin) after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379329(CHEMBL2011824)
Affinity DataIC50:  79nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50435300(CHEMBL2393245)
Affinity DataIC50:  86nMAssay Description:Displacement of [3H]-methylspiperone from dopamine D2L receptor (unknown origin) after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379330(CHEMBL2011823)
Affinity DataIC50:  143nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50435299(CHEMBL2393243)
Affinity DataIC50:  147nMAssay Description:Displacement of [3H]-methylspiperone from dopamine D2L receptor (unknown origin) after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50435298(CHEMBL2393246)
Affinity DataIC50:  163nMAssay Description:Displacement of [3H]-methylspiperone from dopamine D2L receptor (unknown origin) after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379333(CHEMBL2011820)
Affinity DataIC50:  171nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Chung-Ang University

Curated by ChEMBL
LigandPNGBDBM50090677(4-Amino-N-(2-phenyl-2H-pyrazol-3-yl)-benzenesulfon...)
Affinity DataIC50:  180nMAssay Description:Inhibition of CYP2C9 in human liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379325(CHEMBL2011829)
Affinity DataIC50:  196nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Chung-Ang University

Curated by ChEMBL
LigandPNGBDBM50100556(CHEMBL3321845)
Affinity DataIC50:  250nMAssay Description:Inhibition of CYP3A4 in human liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Chung-Ang University

Curated by ChEMBL
LigandPNGBDBM50100557(CHEMBL3321846)
Affinity DataIC50:  260nMAssay Description:Inhibition of CYP3A4 in human liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Chung-Ang University

Curated by ChEMBL
LigandPNGBDBM50100558(CHEMBL3321850)
Affinity DataIC50:  270nMAssay Description:Inhibition of CYP3A4 in human liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379318(CHEMBL2011836)
Affinity DataIC50:  313nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50379327(CHEMBL2011827)
Affinity DataIC50:  314nMAssay Description:Antagonist activity at human GHSR1a receptor assessed as intracellular Ca2+ concentration by aequorin luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Chung-Ang University

Curated by ChEMBL
LigandPNGBDBM50100558(CHEMBL3321850)
Affinity DataIC50:  780nMAssay Description:Inhibition of CYP2C19 in human liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Chung-Ang University

Curated by ChEMBL
LigandPNGBDBM50100557(CHEMBL3321846)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of CYP2C9 in human liver microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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