Found 106 with Last Name = 'kleinau' and Initial = 'g' 
Affinity DataIC50: 0.900nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
Affinity DataIC50: 163nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
Affinity DataIC50: 890nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
Affinity DataIC50: 1.09E+3nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
Affinity DataIC50: 1.55E+3nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 2.98E+3nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR2 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.06E+3nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
Affinity DataIC50: 4.83E+3nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
Affinity DataIC50: 4.89E+3nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 6.07E+3nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR3 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 6.72E+3nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR1 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR5 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
Affinity DataIC50: 7.88E+3nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 8.64E+3nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR3 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 1.05E+4nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR1 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 1.07E+4nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR4 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 2.84E+4nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR5 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 3.75E+4nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR2 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR4 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 800nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 1.90E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 800nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
TargetThyrotropin receptor(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataEC50: 6.50E+3nMAssay Description:Agonist activity at TSHR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity at human oxytocin receptor expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Ggamma2 and Gbeta1 pro...More data for this Ligand-Target Pair
Affinity DataEC50: 0.265nMAssay Description:Agonist activity at human oxytocin receptor high affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Gga...More data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Agonist activity at human oxytocin receptor C47A mutant expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Ggamma2 an...More data for this Ligand-Target Pair
Affinity DataEC50: 182nMAssay Description:Agonist activity at human oxytocin receptor V43A/C47A double mutant expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagge...More data for this Ligand-Target Pair
Affinity DataEC50: 0.00300nMAssay Description:Agonist activity at human oxytocin receptor high affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Gga...More data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Agonist activity at human oxytocin receptor low affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Ggam...More data for this Ligand-Target Pair
Affinity DataEC50: 33nMAssay Description:Agonist activity at human oxytocin receptor low affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Ggam...More data for this Ligand-Target Pair
Affinity DataEC50: 67nMAssay Description:Agonist activity at human oxytocin receptor low affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Ggam...More data for this Ligand-Target Pair
Affinity DataEC50: 75nMAssay Description:Agonist activity at human oxytocin receptor low affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Ggam...More data for this Ligand-Target Pair
Affinity DataEC50: 29nMAssay Description:Agonist activity at human oxytocin receptor expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Ggamma2 and Gbeta1 pro...More data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Agonist activity at human oxytocin receptor expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Ggamma2 and Gbeta1 pro...More data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Agonist activity at human oxytocin receptor expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Ggamma2 and Gbeta1 pro...More data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at human oxytocin receptor expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Ggamma2 and Gbeta1 pro...More data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Agonist activity at human oxytocin receptor C47A mutant expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP-tagged Ggamma2 an...More data for this Ligand-Target Pair
Affinity DataEC50: 0.00100nMAssay Description:Agonist activity at human oxytocin receptor C47A mutant high affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GF...More data for this Ligand-Target Pair
Affinity DataEC50: 135nMAssay Description:Agonist activity at human oxytocin receptor C47A mutant low affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP...More data for this Ligand-Target Pair
Affinity DataEC50: 301nMAssay Description:Agonist activity at human oxytocin receptor C47A mutant low affinity site expressed in HEK293 cells coexpressing Rluc8-tagged Galphaq, N-terminal GFP...More data for this Ligand-Target Pair
