TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.160nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of erbB1 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.230nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.270nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.280nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of erbB1 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.360nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.370nMAssay Description:Compound was evaluated for inhibition of plasma renin activity in monkeyMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.480nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of erbB1 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of erbB4 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of HER stimulated human erbB autophosphorylation in MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of erbB2 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.540nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.570nMAssay Description:Compound was evaluated for inhibition of plasma renin activity in humanMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.581nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.590nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of erbB1 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of erbB1 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of erbB2 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of erbB2 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.760nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibition of erbB2 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibition of ligand stimulated erbB2 autophosphorylation in T24 NIH cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibition of erbB4 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.830nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of erbB1 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division Of Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.910nMAssay Description:In vitro inhibition of monkey renin.More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of HER stimulated human erbB autophosphorylation in MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of erbB4 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of erbB4 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of erbB1 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of erbB2 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of erbB4 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of erbB1 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of erbB1 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of erbB1 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibition of erbB1 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of erbB1 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of erbB1 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of erbB4 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of EGF stimulated human erbB1 autophosphorylation in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition of erbB4 fusion protein expressed in baculovirus by ELISAMore data for this Ligand-Target Pair