Found 179 with Last Name = 'koca' and Initial = 'm' 
Affinity DataKi: 1.60nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 112nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 112nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 145nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 145nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 741nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 912nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 912nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.09E+3nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.57E+3nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.95E+3nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.39E+3nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium-labelled H2 relaxin from RXFP1 expressed in HEK-293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium-labelled H2 relaxin from RXFP1 expressed in HEK-293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium-labelled H2 relaxin from RXFP1 expressed in HEK-293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of europium-labelled H3 relaxin-B chain/INSL-5 chain from RXFP3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataIC50: 0.140nMAssay Description:Inverse agonist activity at GAL4-tagged mouse PPARgamma LBD expressed in CHO cells measured after 6 hrs by firefly luciferase reporter assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataIC50: 0.160nMAssay Description:Inverse agonist activity at PPARgamma in human RT112/84-FABP4 cells assessed as reduction in PPARgamma transactivation measured by Nanoluciferase rep...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataIC50: 0.170nMAssay Description:Inverse agonist activity at PPARgamma in human RT112/84-FABP4 cells assessed as reduction in PPARgamma transactivation measured by Nanoluciferase rep...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataIC50: 0.220nMAssay Description:Inverse agonist activity at PPARgamma in human RT112/84-FABP4 cells assessed as reduction in PPARgamma transactivation measured by Nanoluciferase rep...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataIC50: 0.230nMAssay Description:Inverse agonist activity at PPARgamma in human RT112/84-FABP4 cells assessed as reduction in PPARgamma transactivation measured by Nanoluciferase rep...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataIC50: 0.25nMAssay Description:Inverse agonist activity at PPARgamma in human RT112/84-FABP4 cells assessed as reduction in PPARgamma transactivation measured by Nanoluciferase rep...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataIC50: 0.290nMAssay Description:Inverse agonist activity at PPARgamma in human RT112/84-FABP4 cells assessed as reduction in PPARgamma transactivation measured by Nanoluciferase rep...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataIC50: 0.320nMAssay Description:Inverse agonist activity at PPARgamma in human RT112/84-FABP4 cells assessed as reduction in PPARgamma transactivation measured by Nanoluciferase rep...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inverse agonist activity at GAL4-tagged human PPARgamma LBD expressed in CHO cells measured after 6 hrs by firefly luciferase reporter assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataIC50: 0.580nMAssay Description:Inverse agonist activity at PPARgamma in human RT112/84-FABP4 cells assessed as reduction in PPARgamma transactivation measured by Nanoluciferase rep...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inverse agonist activity at PPARgamma in human RT112/84-FABP4 cells assessed as reduction in PPARgamma transactivation measured by Nanoluciferase rep...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Inverse agonist activity at PPARgamma in human RT112/84-FABP4 cells assessed as reduction in PPARgamma transactivation measured by Nanoluciferase rep...More data for this Ligand-Target Pair
Affinity DataIC50: 3.47nMAssay Description:Agonist activity at RXFP4 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrs by beta galactosidase r...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inverse agonist activity at PPARgamma in human RT112/84-FABP4 cells assessed as reduction in PPARgamma transactivation measured by Nanoluciferase rep...More data for this Ligand-Target Pair
Affinity DataIC50: 4.27nMAssay Description:Agonist activity at RXFP3 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrs by beta galactosidase r...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Inverse agonist activity at PPARgamma in human RT112/84-FABP4 cells assessed as reduction in PPARgamma transactivation measured by Nanoluciferase rep...More data for this Ligand-Target Pair
Affinity DataIC50: 5.13nMAssay Description:Agonist activity at RXFP3 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrs by beta galactosidase r...More data for this Ligand-Target Pair
