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Found 233 with Last Name = 'konishi' and Initial = 'y'
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079482(Arginyl Ketomethylene analogue | CHEMBL410589)
Affinity DataKi:  0.000350nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079489(Arginyl Ketomethylene analogue | CHEMBL428116)
Affinity DataKi:  0.000570nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079476(Arginyl Ketomethylene analogue | CHEMBL437873)
Affinity DataKi:  0.000870nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079479(Arginyl Ketomethylene analogue | CHEMBL407043)
Affinity DataKi:  0.00150nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079485(Arginyl Ketomethylene analogue | CHEMBL414489)
Affinity DataKi:  0.00170nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079478(Arginyl Ketomethylene analogue | CHEMBL414760)
Affinity DataKi:  0.00200nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079491(Arginyl Ketomethylene analogue | CHEMBL412457)
Affinity DataKi:  0.00940nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079480(Arginyl Ketomethylene analogue | CHEMBL415375)
Affinity DataKi:  0.0350nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079488(Arginyl Ketomethylene analogue | CHEMBL414974)
Affinity DataKi:  0.0830nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079490(Arginyl Ketomethylene analogue | CHEMBL437999)
Affinity DataKi:  0.0830nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50004744(CHEMBL2370453 | Hirudin analogue)
Affinity DataKi:  0.140nMAssay Description:Compound was evaluated for their ability to inhibit the alpha-thrombin-mediated hydrolysis of the fluorescent substrate Tos-Gly-Pro-Arg-AmcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50287476(1-((S)-3-{[(S)-1-((R)-2-Amino-3-cyclohexyl-propion...)
Affinity DataKi:  0.190nMAssay Description:Compound was measured for the inhibition of alpha-human thrombin by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50004739(CHEMBL2370455 | Hirudin analogue)
Affinity DataKi:  0.370nMAssay Description:Compound was evaluated for their ability to inhibit the alpha-thrombin-mediated hydrolysis of the fluorescent substrate Tos-Gly-Pro-Arg-AmcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50004745(CHEMBL2370450 | Hirudin analogue)
Affinity DataKi:  0.560nMAssay Description:Compound was evaluated for their ability to inhibit the alpha-thrombin-mediated hydrolysis of the fluorescent substrate Tos-Gly-Pro-Arg-AmcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079487(Arginyl Ketomethylene analogue | CHEMBL415358)
Affinity DataKi:  1.06nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50287477((S)-1-((R)-2-Amino-3-cyclohexyl-propionyl)-pyrroli...)
Affinity DataKi:  1.30nMAssay Description:Compound was measured for the inhibition of alpha-human thrombin by clotting testMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50004743(Ac-(D)Phe-Pro-Arg.Pro.Gln.Ser-H~s.Asn-AspGly-Asp-P...)
Affinity DataKi:  2.80nMAssay Description:Compound was evaluated for their ability to inhibit the alpha-thrombin-mediated hydrolysis of the fluorescent substrate Tos-Gly-Pro-Arg-AmcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50004742(CHEMBL385670 | Hirudin analogue)
Affinity DataKi:  3.20nMAssay Description:Compound was evaluated for their ability to inhibit the alpha-thrombin-mediated hydrolysis of the fluorescent substrate Tos-Gly-Pro-Arg-AmcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50004741(CHEMBL427978 | Hirudin analogue)
Affinity DataKi:  3.5nMAssay Description:Compound was evaluated for their ability to inhibit the alpha-thrombin-mediated hydrolysis of the fluorescent substrate Tos-Gly-Pro-Arg-AmcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50004738(CHEMBL2370451 | Hirudin analogue)
Affinity DataKi:  3.80nMAssay Description:Compound was evaluated for their ability to inhibit the alpha-thrombin-mediated hydrolysis of the fluorescent substrate Tos-Gly-Pro-Arg-AmcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079486(Arginyl Ketomethylene analogue | CHEMBL415237)
Affinity DataKi:  7.30nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121305(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-mercapto-prop...)
Affinity DataKi:  16nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121291(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-methylsulfany...)
Affinity DataKi:  19nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50287475(1-((S)-3-{[(S)-1-((R)-2-Acetylamino-3-cyclohexyl-p...)
Affinity DataKi:  21nMAssay Description:Compound was measured for the inhibition of alpha-human thrombin by clotting testMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121299(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-mercapto-prop...)
Affinity DataKi:  21nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121290(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-mercapto-prop...)
Affinity DataKi:  45nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50287480((S)-1-((R)-2-Amino-3-cyclohexyl-propionyl)-pyrroli...)
Affinity DataKi:  60nMAssay Description:Compound was measured for the inhibition of alpha-human thrombin by clotting testMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121286(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-mercapto-prop...)
Affinity DataKi:  67nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079481(Arginyl Ketomethylene analogue | CHEMBL267326)
Affinity DataKi:  135nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079484(Arginyl Ketomethylene analogue | CHEMBL410552)
Affinity DataKi:  159nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121298(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-mercapto-prop...)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121300(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-mercapto-prop...)
Affinity DataKi:  170nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121300(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-mercapto-prop...)
Affinity DataKi:  170nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50287479((S)-1-((R)-2-Acetylamino-3-cyclohexyl-propionyl)-p...)
Affinity DataKi:  185nMAssay Description:Compound was measured for the inhibition of alpha-human thrombin by clotting testMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121301(5-Amino-2-[2-(2-biphenyl-4-yl-acetylamino)-3-methy...)
Affinity DataKi:  200nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121292(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-methylsulfany...)
Affinity DataKi:  210nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121288(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-mercapto-prop...)
Affinity DataKi:  210nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121295(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-methylsulfany...)
Affinity DataKi:  240nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121289(2-{2-[2-(2-Biphenyl-4-yl-acetylamino)-3-methylsulf...)
Affinity DataKi:  270nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121293(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-mercapto-prop...)
Affinity DataKi:  270nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079477(Arginyl Ketomethylene analogue | CHEMBL408556)
Affinity DataKi:  280nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50004740(CHEMBL2370449 | Hirudin analogue)
Affinity DataKi:  300nMAssay Description:Compound was evaluated for their ability to inhibit the alpha-thrombin-mediated hydrolysis of the fluorescent substrate Tos-Gly-Pro-Arg-AmcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50287478(1-((S)-3-{[(S)-1-((R)-2-Acetylamino-3-phenyl-propi...)
Affinity DataKi:  310nMAssay Description:Compound was measured for the inhibition of alpha-human thrombin by clotting testMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121287(2-[2-(2-Biphenyl-4-yl-acetylamino)-pentanoylamino]...)
Affinity DataKi:  490nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121286(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-mercapto-prop...)
Affinity DataKi:  560nMAssay Description:Specificity of Cathepsin B inhibition by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121302(2-(2-{2-[2-(2-Biphenyl-4-yl-acetylamino)-3-methyls...)
Affinity DataKi:  930nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121286(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-mercapto-prop...)
Affinity DataKi:  1.00E+3nMAssay Description:Specificity of Cathepsin K inhibition by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
National Research Council Canada

Curated by ChEMBL
LigandPNGBDBM50079483(Arginyl Ketomethylene analogue | CHEMBL409563)
Affinity DataKi:  1.46E+3nMAssay Description:Inhibitory constant against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121290(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-mercapto-prop...)
Affinity DataKi:  2.90E+3nMAssay Description:Specificity of Cathepsin K inhibition by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
National Research Council Of Canada

Curated by ChEMBL
LigandPNGBDBM50121297(2-[2-(2-Biphenyl-4-yl-acetylamino)-3-mercapto-prop...)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibitory activity against human Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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