Compile Data Set for Download or QSAR
maximum 50k data
Found 78 with Last Name = 'konkel' and Initial = 'mj'
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50026917(8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...)
Affinity DataKi:  0.460nMAssay Description:Binding affinity for human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50143674(8-{2-[4-(2-Fluoro-phenyl)-piperazin-1-yl]-ethyl}-8...)
Affinity DataKi:  0.830nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50143664(8-{2-[4-(2,5-Difluoro-phenyl)-piperazin-1-yl]-ethy...)
Affinity DataKi:  0.950nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50122803((SNAP-8719)[4-(4-Amino-6,7-dimethoxy-quinazolin-2-...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50026917(8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50165417(8-{2-[4-(2,4,5-Trifluoro-phenyl)-piperazin-1-yl]-e...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50026917(8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity for rat Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187911(1,3-dihydro-1-[3-(2-pyrrolidinylethoxy)phenyl]-3-[...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50143674(8-{2-[4-(2-Fluoro-phenyl)-piperazin-1-yl]-ethyl}-8...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity for rat Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50165418(8-{2-[4-(2,4-Difluoro-phenyl)-piperazin-1-yl]-ethy...)
Affinity DataKi:  5.60nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50143674(8-{2-[4-(2-Fluoro-phenyl)-piperazin-1-yl]-ethyl}-8...)
Affinity DataKi:  7.5nMAssay Description:Binding affinity for human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50165419(8-{2-[4-(3,4-Difluoro-phenyl)-piperazin-1-yl]-ethy...)
Affinity DataKi:  7.90nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187925(1-(3-(2-(piperidin-1-yl)ethoxy)phenyl)-3-(3-(trifl...)
Affinity DataKi:  8nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50143664(8-{2-[4-(2,5-Difluoro-phenyl)-piperazin-1-yl]-ethy...)
Affinity DataKi:  8.10nMAssay Description:Binding affinity for rat Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50026917(8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...)
Affinity DataKi:  14nMAssay Description:Binding affinity for human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50143661(8-{2-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-ethyl}-8...)
Affinity DataKi:  14nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187919(1-(3-(3-(diethylamino)-2-hydroxypropoxy)phenyl)-3-...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187923(1,3-dihydro-1-phenyl-3-[[3-(trilfluoromethyl)pheny...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187923(1,3-dihydro-1-phenyl-3-[[3-(trilfluoromethyl)pheny...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187922(1-(3-(3-(diethylamino)propoxy)phenyl)-3-(3-(triflu...)
Affinity DataKi:  21nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50165417(8-{2-[4-(2,4,5-Trifluoro-phenyl)-piperazin-1-yl]-e...)
Affinity DataKi:  23nMAssay Description:Binding affinity for rat Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50165418(8-{2-[4-(2,4-Difluoro-phenyl)-piperazin-1-yl]-ethy...)
Affinity DataKi:  24nMAssay Description:Binding affinity for human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50143664(8-{2-[4-(2,5-Difluoro-phenyl)-piperazin-1-yl]-ethy...)
Affinity DataKi:  25nMAssay Description:Binding affinity for human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187912(1-(3-(2-(dimethylamino)ethoxy)phenyl)-3-(3-(triflu...)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187908((S)-1-(3-(3-(diethylamino)-2-hydroxypropoxy)phenyl...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187916(1-(3-(3-(dimethylamino)propoxy)phenyl)-3-(3-(trifl...)
Affinity DataKi:  29nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187918(1-(4-(3-(diethylamino)propoxy)phenyl)-3-(3-(triflu...)
Affinity DataKi:  34nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187914(1-(3-((diethylamino)methoxy)phenyl)-3-(3-(trifluor...)
Affinity DataKi:  38nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187913(1-(3-(4-(diethylamino)butoxy)phenyl)-3-(3-(trifluo...)
Affinity DataKi:  45nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187926(1-(3-(3-(pyrrolidin-1-yl)propoxy)phenyl)-3-(3-(tri...)
Affinity DataKi:  49nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189598(1-(ethylpropyl)-3-{[3-(trifluoromethyl)phenyl]azam...)
Affinity DataKi:  52nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50143661(8-{2-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-ethyl}-8...)
Affinity DataKi:  54nMAssay Description:Binding affinity for human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50143664(8-{2-[4-(2,5-Difluoro-phenyl)-piperazin-1-yl]-ethy...)
Affinity DataKi:  54nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50165419(8-{2-[4-(3,4-Difluoro-phenyl)-piperazin-1-yl]-ethy...)
Affinity DataKi:  55nMAssay Description:Binding affinity for human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50143674(8-{2-[4-(2-Fluoro-phenyl)-piperazin-1-yl]-ethyl}-8...)
Affinity DataKi:  67nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187915(1-(4-(4-(diethylamino)butoxy)phenyl)-3-(3-(trifluo...)
Affinity DataKi:  70nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187923(1,3-dihydro-1-phenyl-3-[[3-(trilfluoromethyl)pheny...)
Affinity DataKi:  72nMAssay Description:Binding affinity to human 5HT4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187911(1,3-dihydro-1-[3-(2-pyrrolidinylethoxy)phenyl]-3-[...)
Affinity DataKi:  78nMAssay Description:Binding affinity to human adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187910(1-(4-(2-(diethylamino)ethoxy)phenyl)-3-(3-(trifluo...)
Affinity DataKi:  78nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187909(1-(3-(2-(diethylamino)ethoxy)phenyl)-3-(3-(trifluo...)
Affinity DataKi:  87nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187917(1-(4-(2-(dimethylamino)ethoxy)phenyl)-3-(3-(triflu...)
Affinity DataKi:  89nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189596(1-(2-propynyl)-3-{[3-(trifluoromethyl)phenyl]azame...)
Affinity DataKi:  89nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50143661(8-{2-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-ethyl}-8...)
Affinity DataKi:  91nMAssay Description:Binding affinity for rat Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50122803((SNAP-8719)[4-(4-Amino-6,7-dimethoxy-quinazolin-2-...)
Affinity DataKi:  120nMAssay Description:Binding affinity for rat Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50143664(8-{2-[4-(2,5-Difluoro-phenyl)-piperazin-1-yl]-ethy...)
Affinity DataKi:  120nMAssay Description:Binding affinity for human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50099326(8-{(S)-1-Methyl-2-[4-(2,4,5-trifluoro-phenyl)-pipe...)
Affinity DataKi: >124nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50143674(8-{2-[4-(2-Fluoro-phenyl)-piperazin-1-yl]-ethyl}-8...)
Affinity DataKi:  140nMAssay Description:Binding affinity for human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189600((E)-1-allyl-3-(3,4-dichlorophenylimino)indolin-2-o...)
Affinity DataKi:  150nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50165419(8-{2-[4-(3,4-Difluoro-phenyl)-piperazin-1-yl]-ethy...)
Affinity DataKi:  160nMAssay Description:Binding affinity for rat Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50122803((SNAP-8719)[4-(4-Amino-6,7-dimethoxy-quinazolin-2-...)
Affinity DataKi:  165nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 78 total ) | Next | Last >>
Jump to: