Compile Data Set for Download or QSAR
maximum 50k data
Found 185 with Last Name = 'kornberg' and Initial = 'be'
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187923(1,3-dihydro-1-phenyl-3-[[3-(trilfluoromethyl)pheny...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189598(1-(ethylpropyl)-3-{[3-(trifluoromethyl)phenyl]azam...)
Affinity DataKi:  52nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187923(1,3-dihydro-1-phenyl-3-[[3-(trilfluoromethyl)pheny...)
Affinity DataKi:  72nMAssay Description:Binding affinity to human 5HT4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189596(1-(2-propynyl)-3-{[3-(trifluoromethyl)phenyl]azame...)
Affinity DataKi:  89nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189600((E)-1-allyl-3-(3,4-dichlorophenylimino)indolin-2-o...)
Affinity DataKi:  150nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189597((E)-3-(2,3-dichlorophenylimino)indolin-2-one | CHE...)
Affinity DataKi:  437nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189595(3-{[3-(trifluoromethyl)phenyl]azamethylene}benzo[d...)
Affinity DataKi:  596nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189599((E)-3-(4-chlorophenylimino)indolin-2-one | CHEMBL2...)
Affinity DataKi:  850nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189601((E)-3-(4-methoxyphenylimino)indolin-2-one | (E/Z)-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008145(CHEMBL286147 | Morpholine-4-carboxylic acid (1-{1-...)
Affinity DataIC50:  0.100nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50005417(CHEMBL266334 | N-[(1-Cyclohexylmethyl-2,3-dihydrox...)
Affinity DataIC50:  0.130nMAssay Description:Inhibitory activity against monkey renin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50005437(CHEMBL8477 | N-[Allylsulfanyl-(1-cyclohexylmethyl-...)
Affinity DataIC50:  0.170nMAssay Description:Inhibitory activity against monkey renin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50005443(CHEMBL441325 | N-[(1-Cyclohexylmethyl-2,3-dihydrox...)
Affinity DataIC50:  0.180nMAssay Description:Inhibitory activity against monkey renin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008141(2-[2-(Morpholine-4-sulfonylamino)-3-phenyl-propion...)
Affinity DataIC50:  0.210nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50005431(CHEMBL8665 | N-[(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  0.210nMAssay Description:Inhibitory activity against monkey renin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008130(2-[3-Phenyl-2-(3-pyridin-3-yl-propionylamino)-prop...)
Affinity DataIC50:  0.220nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50005442(CHEMBL262712 | N-[Allyloxy-(1-cyclohexylmethyl-2,3...)
Affinity DataIC50:  0.220nMAssay Description:Inhibitory activity against monkey renin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008151(2-[3-Phenyl-2-(3-pyridin-3-yl-propionylamino)-prop...)
Affinity DataIC50:  0.230nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008129(2-[2-(Morpholine-4-sulfonylamino)-3-phenyl-propion...)
Affinity DataIC50:  0.230nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50005445(CHEMBL267277 | N-[1-(1-Cyclohexylmethyl-2,3-dihydr...)
Affinity DataIC50:  0.230nMAssay Description:Inhibitory activity against monkey reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008138(2-[2-(Morpholine-4-sulfonylamino)-3-phenyl-propion...)
Affinity DataIC50:  0.240nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008132(5-Cyclohexyl-2,2-difluoro-4-{2-[2-(morpholine-4-su...)
Affinity DataIC50:  0.25nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50005428(CHEMBL8836 | N-[(1-Cyclohexylmethyl-2,3-dihydroxy-...)
Affinity DataIC50:  0.25nMAssay Description:Inhibitory activity against monkey renin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008153(CHEMBL32575 | Morpholine-4-carboxylic acid (1-{1-[...)
Affinity DataIC50:  0.280nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008147(2-[3-(4-Methoxy-phenyl)-2-(morpholine-4-sulfonylam...)
Affinity DataIC50:  0.300nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008121(2-[2-(Morpholine-4-sulfonylamino)-3-phenyl-propion...)
Affinity DataIC50:  0.310nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008158(2-[2-(Morpholine-4-sulfonylamino)-3-phenyl-propion...)
Affinity DataIC50:  0.320nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008127(2-[3-Phenyl-2-(piperazine-1-sulfonylamino)-propion...)
Affinity DataIC50:  0.350nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008133(2-[2-(Morpholine-4-sulfonylamino)-3-phenyl-propion...)
Affinity DataIC50:  0.350nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008136(2-[2-(Morpholine-4-sulfonylamino)-3-phenyl-propion...)
Affinity DataIC50:  0.360nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008122(5-Cyclohexyl-2,2-difluoro-4-{2-[2-(morpholine-4-su...)
Affinity DataIC50:  0.400nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008137(2-[2-(4-Methyl-piperazine-1-sulfonylamino)-3-pheny...)
Affinity DataIC50:  0.420nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50005422(5-Cyclohexyl-2,2-difluoro-3-hydroxy-4-{2-[2-(morph...)
Affinity DataIC50:  0.440nMAssay Description:Inhibitory activity against monkey renin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008148(5-Cyclohexyl-2,2-difluoro-3-hydroxy-4-{2-[2-(morph...)
Affinity DataIC50:  0.440nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008142(2-[2-(Morpholine-4-sulfonylamino)-3-phenyl-propion...)
Affinity DataIC50:  0.460nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006856(4-{3-(2-Amino-thiazol-4-yl)-2-[2-(morpholine-4-sul...)
Affinity DataIC50:  0.5nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50005423(CHEMBL266139 | N-[(1-Cyclohexylmethyl-2,3-dihydrox...)
Affinity DataIC50:  0.520nMAssay Description:Inhibitory activity against monkey renin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008154(2-[3-Phenyl-2-(piperazine-1-sulfonylamino)-propion...)
Affinity DataIC50:  0.570nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008125(CHEMBL285207 | N-[1-Cyclohexylmethyl-3,3-difluoro-...)
Affinity DataIC50:  0.620nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008144(4-{3-(2-Amino-thiazol-4-yl)-2-[2-(morpholine-4-sul...)
Affinity DataIC50:  0.690nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008156(2-[2-(Morpholine-4-sulfonylamino)-3-phenyl-propion...)
Affinity DataIC50:  0.700nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008162(CHEMBL31621 | N-[1-Cyclohexylmethyl-3,3-difluoro-3...)
Affinity DataIC50:  0.790nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008149(2-[2-(Morpholine-4-sulfonylamino)-3-phenyl-propion...)
Affinity DataIC50:  0.810nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368310(CHEMBL1790136)
Affinity DataIC50:  0.820nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008124(2-[2-(Morpholine-4-sulfonylamino)-3-phenyl-propion...)
Affinity DataIC50:  0.870nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008123(5-Cyclohexyl-2,2-difluoro-4-{3-(1H-imidazol-4-yl)-...)
Affinity DataIC50:  0.900nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008131(2-[2-(4-Methyl-piperazine-1-sulfonylamino)-3-pheny...)
Affinity DataIC50:  0.920nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50367254(ENALAPRILAT)
Affinity DataIC50:  1.20nMAssay Description:In vitro inhibition of Angiotensin I converting enzyme in Hog plasmaMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008139(2-[2-(Morpholine-4-sulfonylamino)-3-phenyl-propion...)
Affinity DataIC50:  1.20nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008140(5-Cyclohexyl-2,2-difluoro-4-{2-[2-(morpholine-4-su...)
Affinity DataIC50:  1.20nMAssay Description:The concentration producing 50% inhibition of renin activity in monkey plasma was determined by radioimmunoassay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 185 total ) | Next | Last >>
Jump to: