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Found 326 with Last Name = 'kraus' and Initial = 'a'
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Iowa State University

Curated by ChEMBL
LigandPNGBDBM50303233(2-(3-aminophenylamino)-6-(2,6-dichlorophenyl)-8-me...)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of recombinant c-Abl after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Iowa State University

Curated by ChEMBL
LigandPNGBDBM50378812(CHEMBL1221411)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of recombinant c-Abl after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Iowa State University

Curated by ChEMBL
LigandPNGBDBM6568(6-(2,6-dichlorophenyl)-8-methyl-2-{[3-(methylsulfa...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of recombinant c-Abl after 30 minsMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Iowa State University

Curated by ChEMBL
LigandPNGBDBM50378803(CHEMBL1223343)
Affinity DataKi:  8nMAssay Description:Inhibition of recombinant c-Abl after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86742(UR-AK64)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Iowa State University

Curated by ChEMBL
LigandPNGBDBM50378810(CHEMBL1223482)
Affinity DataKi:  20nMAssay Description:Inhibition of recombinant c-Abl after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Iowa State University

Curated by ChEMBL
LigandPNGBDBM50378811(CHEMBL1223483)
Affinity DataKi:  20nMAssay Description:Inhibition of recombinant c-Abl after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86747(UR-AK67)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86738(UR-AK46)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86743(UR-AK49)
Affinity DataKi:  22nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKi:  23nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86744(UR-AK62)
Affinity DataKi:  23nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86745(UR-AK51)
Affinity DataKi:  23nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86742(UR-AK64)
Affinity DataKi:  23nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86736(UR-AK68)
Affinity DataKi:  29nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86741(UR-AK59)
Affinity DataKi:  37nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86738(UR-AK46)
Affinity DataKi:  38nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Iowa State University

Curated by ChEMBL
LigandPNGBDBM50378807(CHEMBL1223412)
Affinity DataKi:  40nMAssay Description:Inhibition of recombinant c-Abl after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Iowa State University

Curated by ChEMBL
LigandPNGBDBM50378806(CHEMBL1223411)
Affinity DataKi:  40nMAssay Description:Inhibition of recombinant c-Abl after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86743(UR-AK49)
Affinity DataKi:  46nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86737(UR-AK22)
Affinity DataKi:  56nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Iowa State University

Curated by ChEMBL
LigandPNGBDBM50378804(CHEMBL1223344)
Affinity DataKi:  60nMAssay Description:Inhibition of recombinant c-Abl after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86744(UR-AK62)
Affinity DataKi:  62nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86747(UR-AK67)
Affinity DataKi:  67nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKi:  67nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Iowa State University

Curated by ChEMBL
LigandPNGBDBM50378808(CHEMBL1223413)
Affinity DataKi:  70nMAssay Description:Inhibition of recombinant c-Abl after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86737(UR-AK22)
Affinity DataKi:  72nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86736(UR-AK68)
Affinity DataKi:  75nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86735(UR-AK26)
Affinity DataKi:  76nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86741(UR-AK59)
Affinity DataKi:  99nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86745(UR-AK51)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86735(UR-AK26)
Affinity DataKi:  150nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM7966(2-(1H-imidazol-4-yl)ethan-1-amine | CHEMBL544208 |...)
Affinity DataKi:  190nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistamine H1 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKi:  280nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86742(UR-AK64)
Affinity DataKi:  350nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86737(UR-AK22)
Affinity DataKi:  440nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86739(UR-AK41)
Affinity DataKi:  640nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Iowa State University

Curated by ChEMBL
LigandPNGBDBM50378809(CHEMBL1223481)
Affinity DataKi:  900nMAssay Description:Inhibition of recombinant c-Abl after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKi:  910nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86742(UR-AK64)
Affinity DataKi:  990nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM7966(2-(1H-imidazol-4-yl)ethan-1-amine | CHEMBL544208 |...)
Affinity DataKi:  1.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM7966(2-(1H-imidazol-4-yl)ethan-1-amine | CHEMBL544208 |...)
Affinity DataKi:  1.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86739(UR-AK41)
Affinity DataKi:  1.40E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKi:  1.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Iowa State University

Curated by ChEMBL
LigandPNGBDBM50378805(CHEMBL1223410)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of recombinant c-Abl after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86747(UR-AK67)
Affinity DataKi:  2.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86741(UR-AK59)
Affinity DataKi:  2.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKi:  2.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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