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Found 72 with Last Name = 'kull' and Initial = 'fc'
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040317(CHEMBL262756 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040307(1-naphthyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)
Affinity DataIC50:  0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040299(CHEMBL410783 | cyclopropylbenzene(CO)His-Trp-Ala-V...)
Affinity DataIC50:  0.0300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040325(CHEMBL268386 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  0.0380nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040299(CHEMBL410783 | cyclopropylbenzene(CO)His-Trp-Ala-V...)
Affinity DataIC50:  0.0490nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040307(1-naphthyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)
Affinity DataIC50:  0.0500nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040301(4-OHPhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50:  0.0500nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040312(2-tetrahydronaphthyl(CO)His-Trp-Ala-Val-DAla-His-D...)
Affinity DataIC50:  0.0790nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040308(2-aminoPhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50:  0.100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040310(3-CF3PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50:  0.160nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040315((CH3)2PhC(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe...)
Affinity DataIC50:  0.180nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040315((CH3)2PhC(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe...)
Affinity DataIC50:  0.180nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040317(CHEMBL262756 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  0.220nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040301(4-OHPhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50:  0.230nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040312(2-tetrahydronaphthyl(CO)His-Trp-Ala-Val-DAla-His-D...)
Affinity DataIC50:  0.300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040320(CHEMBL264122 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  0.330nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407275(CHEMBL2112786)
Affinity DataIC50:  0.490nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040316(3-isoquinolyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50:  0.570nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040324(CHEMBL266516 | PhCH2CH2(CO)His-(BzthAla)-Ala-Val-D...)
Affinity DataIC50:  0.75nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040310(3-CF3PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50:  1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407276(CHEMBL2111952)
Affinity DataIC50:  1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407276(CHEMBL2111952)
Affinity DataIC50:  1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407273(CHEMBL2111953)
Affinity DataIC50:  1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040314((CH3)2PhCCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50:  1.20nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407273(CHEMBL2111953)
Affinity DataIC50:  1.30nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040323(CHEMBL265736 | phenothiazoneCH2CH2(CO)His-Trp-Ala-...)
Affinity DataIC50:  1.90nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040308(2-aminoPhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50:  2nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040298(CHEMBL386478 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  2nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407277(CHEMBL2112785)
Affinity DataIC50:  3nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407277(CHEMBL2112785)
Affinity DataIC50:  3nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040319(4-CF3PhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)
Affinity DataIC50:  3.70nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040298(CHEMBL386478 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  5nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040304(CHEMBL267943 | PhCH2CH2(CO)ThiAla-Trp-Ala-Val-DAla...)
Affinity DataIC50:  5.60nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040304(CHEMBL267943 | PhCH2CH2(CO)ThiAla-Trp-Ala-Val-DAla...)
Affinity DataIC50:  5.60nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040321(CHEMBL385805 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  7.30nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040321(CHEMBL385805 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  7.30nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50453525(CHEMBL2370862)
Affinity DataIC50:  7.70nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040305(3-CF3PhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)
Affinity DataIC50:  8.40nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040314((CH3)2PhCCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50:  10nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040306(2-CF3PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50:  12nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040302(CHEMBL415455 | PhCH2CH2(CO)His-Trp-Ala-Val-Sar-His...)
Affinity DataIC50:  21nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040302(CHEMBL415455 | PhCH2CH2(CO)His-Trp-Ala-Val-Sar-His...)
Affinity DataIC50:  21nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM32362(5-[[3-methoxy-4-[(4-methoxyphenyl)methoxy]phenyl]m...)
Affinity DataIC50:  30nMAssay Description:Inhibition of recombinant human GST-tagged CFMS kinase catalytic domain using biotin-EAIYAPFAKKK-NH2 as substrate after 40 mins by NXT scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407274(CHEMBL2111954)
Affinity DataIC50:  31nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407274(CHEMBL2111954)
Affinity DataIC50:  50nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040303(CHEMBL383984 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  140nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040303(CHEMBL383984 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  140nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040318(CHEMBL386476 | PhCH2CH2(CO)His-Trp-Ala-(psi)Val-DA...)
Affinity DataIC50: >1.00E+3nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM32362(5-[[3-methoxy-4-[(4-methoxyphenyl)methoxy]phenyl]m...)
Affinity DataIC50: >4.80E+3nMAssay Description:Inhibition of recombinant human His-tagged B-RAF after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase LCK(Mus musculus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM32362(5-[[3-methoxy-4-[(4-methoxyphenyl)methoxy]phenyl]m...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mouse LCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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