TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Affinity DataKi: 0.300nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetSubstance-K receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Affinity DataKi: 0.5nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -CD providing a measure of muscarinic m1 receptor agonist affinityMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Affinity DataKi: 0.880nMAssay Description:Binding affinity to recombinant human His6-tagged HDM2 (1 to 118 residues) assessed as reduction in PMDM6-F binding incubated for 15 to 30 mins by fl...More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Affinity DataKi: 1.20nMAssay Description:The compound was evaluated for the inhibition of [125I]-NKA binding to neurokinin NK2 receptor from hamster urinary bladder membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to mineralocorticoid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Inhibition of hexa-His-tagged JNK2 expressed in baculoviral system using GST-tagged cJun as substrate preincubated for 15 mins prior ATP addition mea...More data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -CD providing a measure of muscarinic m1 receptor agonist affinityMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -CD providing a measure of muscarinic m1 receptor agonist affinityMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -CD providing a measure of muscarinic m1 receptor agonist affinityMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database
Sanofi-SynthÉLabo Recherche
Curated by PDSP Ki Database