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Found 3818 with Last Name = 'lai' and Initial = 'p'
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  0.00430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  0.00610nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.0420nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.0440nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(mouse)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM85083(NKB [MePhe7])
Affinity DataKi:  0.0530nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.0540nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.0590nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Gerbil)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM85083(NKB [MePhe7])
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281769(Acetic acid 1-[4-(benzoyl-methyl-amino)-3-(3,4-dic...)
Affinity DataKi:  0.300nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281767(Acetic acid 1-{3-(3,4-dichloro-phenyl)-4-[ethyl-(t...)
Affinity DataKi:  0.300nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM85083(NKB [MePhe7])
Affinity DataKi:  0.340nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Gerbil)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  0.420nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM85083(NKB [MePhe7])
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81942(CAS_55582 | NKA | NSC_55582 | Neurokinin alpha | S...)
Affinity DataKi:  0.480nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50071484(CHEMBL308148 | N-[(R)-4-(4-Acetylamino-4-phenyl-pi...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280553(8-Methyl-2,2-diphenyl-1,3-dioxa-8-aza-spiro[4.5]de...)
Affinity DataKi:  0.600nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -CD providing a measure of muscarinic m1 receptor agonist affinityMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50335566(CHEMBL1651026 | Substance P [Sar9,Met(O2)11])
Affinity DataKi:  0.650nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM81942(CAS_55582 | NKA | NSC_55582 | Neurokinin alpha | S...)
Affinity DataKi:  0.760nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50433561(CHEMBL2381408)
Affinity DataKi:  0.880nMAssay Description:Binding affinity to recombinant human His6-tagged HDM2 (1 to 118 residues) assessed as reduction in PMDM6-F binding incubated for 15 to 30 mins by fl...More data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281771(CHEMBL173841 | N-[2-(3,4-Dichloro-phenyl)-4-(4-eth...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H1 receptor(Homo sapiens (Human))
Ucb Pharma

Curated by PDSP Ki Database
LigandPNGBDBM22875(2-(2-{4-[(4-chlorophenyl)(phenyl)methyl]piperazin-...)
In DepthDetails ArticlePubMedDrugBank

TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50129513(CHEMBL71397 | N-[2-(3,4-Dichloro-phenyl)-4-(4-hydr...)
Affinity DataKi:  1nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281768(CHEMBL176588 | Thiophene-3-carboxylic acid [2-(3,4...)
Affinity DataKi:  1nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  1.07nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  1.15nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50071484(CHEMBL308148 | N-[(R)-4-(4-Acetylamino-4-phenyl-pi...)
Affinity DataKi:  1.20nMAssay Description:The compound was evaluated for the inhibition of [125I]-NKA binding to neurokinin NK2 receptor from hamster urinary bladder membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281766(CHEMBL173008 | Thiophene-2-carboxylic acid [2-(3,4...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281773(CHEMBL176853 | Naphthalene-1-carboxylic acid [2-(3...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMineralocorticoid receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50089636(CHEMBL3578271)
Affinity DataKi:  2nMAssay Description:Binding affinity to mineralocorticoid receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Ucb Pharma

Curated by PDSP Ki Database
LigandPNGBDBM22879((1R)-1-(4-tert-butylphenyl)-4-[4-(hydroxydiphenylm...)
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Ucb Pharma

Curated by PDSP Ki Database
LigandPNGBDBM22875(2-(2-{4-[(4-chlorophenyl)(phenyl)methyl]piperazin-...)
In DepthDetails ArticlePubMedDrugBank

TargetSubstance-K receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM81942(CAS_55582 | NKA | NSC_55582 | Neurokinin alpha | S...)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Ucb Pharma

Curated by PDSP Ki Database
LigandPNGBDBM81466(CAS_23095-76-3 | NSC_6445134 | l-Chlorpheniramine)
Affinity DataKi:  2.51nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Ucb Pharma

Curated by PDSP Ki Database
LigandPNGBDBM22890(2-(2-{4-[(4-chlorophenyl)(phenyl)methyl]piperazin-...)
Affinity DataKi:  3.16nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistamine H1 receptor(Homo sapiens (Human))
Ucb Pharma

Curated by PDSP Ki Database
LigandPNGBDBM85849(ucb 29992, (R))
Affinity DataKi:  5.01nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50364378(CHEMBL1950289)
Affinity DataKi:  6.20nMAssay Description:Inhibition of hexa-His-tagged JNK2 expressed in baculoviral system using GST-tagged cJun as substrate preincubated for 15 mins prior ATP addition mea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM73209((+)-CIS-DIOXOLANE | CHEMBL105457 | MLS000069362 | ...)
Affinity DataKi:  6.40nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -CD providing a measure of muscarinic m1 receptor agonist affinityMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50280553(8-Methyl-2,2-diphenyl-1,3-dioxa-8-aza-spiro[4.5]de...)
Affinity DataKi:  8.10nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -CD providing a measure of muscarinic m1 receptor agonist affinityMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H1 receptor(Homo sapiens (Human))
Ucb Pharma

Curated by PDSP Ki Database
LigandPNGBDBM22874(2-(4-{1-hydroxy-4-[4-(hydroxydiphenylmethyl)piperi...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

LigandPNGBDBM50006243(((2S,4R,5S)-4-Hydroxy-5-methyl-tetrahydro-furan-2-...)
Affinity DataKi:  12nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -CD providing a measure of muscarinic m1 receptor agonist affinityMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(mouse)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50051290(CHEMBL299377 | N-(1-{3-[1-Benzoyl-3-(3,4-dichloro-...)
Affinity DataKi:  15nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sanofi Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281770(CHEMBL367542 | N-[4-[4-(Acetylamino-methyl)-4-phen...)
Affinity DataKi:  23nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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