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Found 65 with Last Name = 'lajis' and Initial = 'nh'
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180622(CHEMBL3814519)
Affinity DataKi:  200nMAssay Description:Mixed type inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180621(CHEMBL3814621)
Affinity DataKi:  1.90E+3nMAssay Description:Mixed type inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  10nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 30 mins by E...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  95nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM22372(4-[(2R,3S)-4-(3,4-dihydroxyphenyl)-2,3-dimethylbut...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human 5-LOX in human peripheral blood mononuclear leukocytes assessed as inhibition of calymycin A23187-stimulated LTB4 production prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  250nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine iodide as substrate after 10 mins by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50357364(CHEMBL1242095)
Affinity DataIC50:  400nMAssay Description:Inhibition of human recombinant COX2 expressed in insect Sf21 cells assessed as inhibition of conversion of arachidonic acid to PGE2 preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM22372(4-[(2R,3S)-4-(3,4-dihydroxyphenyl)-2,3-dimethylbut...)
Affinity DataIC50:  400nMAssay Description:Inhibition of 5-LOX in calcium ionophore A23187-stimulated NMRI mouse macrophage assessed as inhibition of LTC4 production preincubated for 60 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50357364(CHEMBL1242095)
Affinity DataIC50:  420nMAssay Description:Inhibition of human 5-LOX in human peripheral blood mononuclear leukocytes assessed as inhibition of calymycin A23187-stimulated LTB4 production prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50259930(6-(10'Z-heptadecenyl)-salicylicacid | 6-[10'(Z)-he...)
Affinity DataIC50:  573nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine iodide as substrate after 10 mins by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180622(CHEMBL3814519)
Affinity DataIC50:  600nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
University Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50320314(5-(Naphthalen-1-ylmethyl)-3-(piperazin-1-ylmethyl)...)
Affinity DataIC50:  870nMAssay Description:Inhibition of mushroom tyrosinase preincubated for 5 mins before addition of L-DOPA measured after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
University Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50320310(1-ylmethyl)-3-(piperidin-1-ylmethyl)-1,3,4-oxadiaz...)
Affinity DataIC50:  970nMAssay Description:Inhibition of mushroom tyrosinase preincubated for 5 mins before addition of L-DOPA measured after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
University Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50320312((Naphthalen-1-ylmethyl)-3-(pyrrolidin-1-ylmethyl)-...)
Affinity DataIC50:  1.33E+3nMAssay Description:Inhibition of mushroom tyrosinase preincubated for 5 mins before addition of L-DOPA measured after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
University Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50320311((Morpholinomethyl)-5-(naphthalen-1-ylmethyl)-1,3,4...)
Affinity DataIC50:  1.34E+3nMAssay Description:Inhibition of mushroom tyrosinase preincubated for 5 mins before addition of L-DOPA measured after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180620(CHEMBL3814587)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
University Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50320313(3-((4-Methylpiperazin-1-yl)methyl)-5-(naphthalen-1...)
Affinity DataIC50:  1.49E+3nMAssay Description:Inhibition of mushroom tyrosinase preincubated for 5 mins before addition of L-DOPA measured after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180621(CHEMBL3814621)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50357364(CHEMBL1242095)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of 5-LOX in calcium ionophore A23187-stimulated NMRI mouse macrophage assessed as inhibition of LTC4 production preincubated for 60 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180623(CHEMBL3814100)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50292424(Anacardic acid 10'Z-monoene | CHEMBL470264)
Affinity DataIC50:  2.17E+3nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine iodide as substrate after 10 mins by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180623(CHEMBL3814100)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180621(CHEMBL3814621)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180620(CHEMBL3814587)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50347127(CHEMBL1797234)
Affinity DataIC50:  3.18E+3nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine iodide as substrate after 10 mins by Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180622(CHEMBL3814519)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180626(CHEMBL3601745)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180616(CHEMBL3601747)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180599(CHEMBL3813978)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180598(CHEMBL3814375)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180617(CHEMBL3601748)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180624(CHEMBL3601736)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180591(CHEMBL3813909)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180589(CHEMBL3814533)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50357364(CHEMBL1242095)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of COX1 in human platelets assessed as inhibition of conversion of arachidonic acid to PGE2 preincubated for 15 mins before substrate addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180613(CHEMBL3601632)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180614(CHEMBL3601737)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180597(CHEMBL3601636)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180618(CHEMBL3814765)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180596(CHEMBL3601634)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180615(CHEMBL3601738)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180619(CHEMBL3813797)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180593(CHEMBL3815025)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180612(CHEMBL3814991)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180611(CHEMBL3813809)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180594(CHEMBL3814476)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180592(CHEMBL3814230)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180595(CHEMBL3813840)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
University Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50031467(5-HYDROXY-2-(HYDROXYMETHYL)-4H-PYRAN-4-ONE | 5-Hyd...)
Affinity DataIC50:  9.18E+3nMAssay Description:Inhibition of mushroom tyrosinase preincubated for 5 mins before addition of L-DOPA measured after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180590(CHEMBL3601749)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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