Affinity DataKi: 2.10E+4nMAssay Description:Competitive inhibition of human purified TDO by Henri-Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.0800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.0900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human Integrin alpha5beta3 receptors expressed in HOP cells assessed as cell attachment after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human Integrin alpha5beta3 receptors expressed in HOP cells assessed as cell attachment after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetG-protein coupled receptor 183(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at EBI2 receptor in human U937 cells assessed as inhibition of 7-alpha,25-OHC-induced cell migration after 3 hrs by flow cytometr...More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.480nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human Integrin alpha5beta3 receptors expressed in HOP cells assessed as cell attachment after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.810nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair