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Found 224 with Last Name = 'laurent' and Initial = 's'
TargetTryptophan 2,3-dioxygenase(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50289137(6-Fluoro-3-((E)-2-pyridin-3-yl-vinyl)-1H-indole | ...)
Affinity DataKi:  30nMAssay Description:Inhibition of liver TDOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptophan 2,3-dioxygenase(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50350281(CHEMBL1812527)
Affinity DataKi:  2.10E+4nMAssay Description:Competitive inhibition of human purified TDO by Henri-Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470233(CHEMBL80177)
Affinity DataIC50:  0.0800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470229(CHEMBL76870)
Affinity DataIC50:  0.0900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313793((S)-3-(3-amino-4-(3-(5,6,7,8-tetrahydro-1,8-naphth...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of human Integrin alpha5beta3 receptors expressed in HOP cells assessed as cell attachment after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470239(CHEMBL311312)
Affinity DataIC50:  0.100nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470236(CHEMBL309313)
Affinity DataIC50:  0.100nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50213569(CHEMBL78866)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470206(CHEMBL445365)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470250(CHEMBL77308)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50213557(CHEMBL309602)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50031491(2-propyl-4-(methythio)-1-[[[2'-[(propylamino)carbo...)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470235(CHEMBL308135)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470226(CHEMBL311827)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470225(CHEMBL80700)
Affinity DataIC50:  0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470249(CHEMBL309845)
Affinity DataIC50:  0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470227(CHEMBL76538)
Affinity DataIC50:  0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313795((S)-3-(4-(3-(5,6,7,8-tetrahydro-1,8-naphthyridin-2...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of human Integrin alpha5beta3 receptors expressed in HOP cells assessed as cell attachment after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470223(CHEMBL312386)
Affinity DataIC50:  0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470241(CHEMBL305638)
Affinity DataIC50:  0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 183(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50011716(CHEMBL3262896)
Affinity DataIC50:  0.300nMAssay Description:Antagonist activity at EBI2 receptor in human U937 cells assessed as inhibition of 7-alpha,25-OHC-induced cell migration after 3 hrs by flow cytometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50031537(2-Butyl-3-(N'-propylureidylsulfonyl-biphenyl-4-ylm...)
Affinity DataIC50:  0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470234(CHEMBL76948)
Affinity DataIC50:  0.400nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470228(CHEMBL80971)
Affinity DataIC50:  0.400nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50031530(2-Butyl-4-(methylthio)-1-[[2'-[[[(propylamino)carb...)
Affinity DataIC50:  0.480nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470243(CHEMBL306157)
Affinity DataIC50:  0.5nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470219(CHEMBL305604)
Affinity DataIC50:  0.600nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470212(CHEMBL80622)
Affinity DataIC50:  0.600nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50313794((S)-3-(3-(20-amino-3,6,9,12,15,18-hexaoxaicosanami...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of human Integrin alpha5beta3 receptors expressed in HOP cells assessed as cell attachment after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470214(CHEMBL77360)
Affinity DataIC50:  0.800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470230(CHEMBL76799)
Affinity DataIC50:  0.800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470240(CHEMBL432158)
Affinity DataIC50:  0.800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470217(CHEMBL77138)
Affinity DataIC50:  0.800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093978(2-(4-Carboxy-cyclohexylmethyl)-4-(6-chloro-benzo[1...)
Affinity DataIC50:  0.810nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470224(CHEMBL311189)
Affinity DataIC50:  0.900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470208(CHEMBL80900)
Affinity DataIC50:  0.900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470248(CHEMBL311847)
Affinity DataIC50:  0.900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470231(CHEMBL76613)
Affinity DataIC50:  1nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470246(CHEMBL306085)
Affinity DataIC50:  1nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470237(CHEMBL306778)
Affinity DataIC50:  1nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093997(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093996(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470238(CHEMBL80908)
Affinity DataIC50:  1.10nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470222(CHEMBL443069)
Affinity DataIC50:  1.10nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50094000(2-(3-Carboxy-cyclohexylmethyl)-4-(6-chloro-benzo[1...)
Affinity DataIC50:  1.30nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093987(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  1.30nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470216(CHEMBL310267)
Affinity DataIC50:  1.30nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470245(CHEMBL78169)
Affinity DataIC50:  1.5nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470207(CHEMBL413491)
Affinity DataIC50:  1.70nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093997(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  1.70nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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