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Found 43 with Last Name = 'lazarus' and Initial = 'mb'
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50111577(CHEMBL3605055)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of SUMO-tagged ULK1 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase ULK2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50111577(CHEMBL3605055)
Affinity DataIC50:  13nMAssay Description:Inhibition of SUMO-tagged ULK2 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50111575(CHEMBL3603853)
Affinity DataIC50:  56nMAssay Description:Inhibition of recombinant PDK1 (unknown origin) using PDK1tide substrate incubated for 7 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM17051(BX-795 | BX-795, 3 | N-(3-{[5-iodo-4-({3-[(thiophe...)
Affinity DataIC50:  65nMAssay Description:Inhibition of recombinant PDK1 (unknown origin) using PDK1tide substrate incubated for 7 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50111575(CHEMBL3603853)
Affinity DataIC50:  67nMAssay Description:Inhibition of SUMO-tagged ULK1 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM17051(BX-795 | BX-795, 3 | N-(3-{[5-iodo-4-({3-[(thiophe...)
Affinity DataIC50:  87nMAssay Description:Inhibition of SUMO-tagged ULK1 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50111573(CHEMBL3605056)
Affinity DataIC50:  120nMAssay Description:Inhibition of SUMO-tagged ULK1 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubat...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ULK1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50111572(CHEMBL3605057)
Affinity DataIC50:  170nMAssay Description:Inhibition of SUMO-tagged ULK1 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase ULK2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50111575(CHEMBL3603853)
Affinity DataIC50:  200nMAssay Description:Inhibition of SUMO-tagged ULK2 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase ULK2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50111572(CHEMBL3605057)
Affinity DataIC50:  230nMAssay Description:Inhibition of SUMO-tagged ULK2 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubat...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ULK2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM17051(BX-795 | BX-795, 3 | N-(3-{[5-iodo-4-({3-[(thiophe...)
Affinity DataIC50:  310nMAssay Description:Inhibition of SUMO-tagged ULK2 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase ULK2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50111573(CHEMBL3605056)
Affinity DataIC50:  360nMAssay Description:Inhibition of SUMO-tagged ULK2 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50111577(CHEMBL3605055)
Affinity DataIC50:  420nMAssay Description:Inhibition of recombinant PDK1 (unknown origin) using PDK1tide substrate incubated for 7 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50111572(CHEMBL3605057)
Affinity DataIC50:  421nMAssay Description:Inhibition of recombinant PDK1 (unknown origin) using PDK1tide substrate incubated for 7 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50111573(CHEMBL3605056)
Affinity DataIC50:  710nMAssay Description:Inhibition of recombinant PDK1 (unknown origin) using PDK1tide substrate incubated for 7 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147122(US8957075, Table 1 Compound 17)
Affinity DataKd:  1.30E+4nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147123(US8957075, Table 1 Compound 18)
Affinity DataKd:  4.70E+3nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147124(US8957075, Table 1 Compound 19 | US8957075, Table ...)
Affinity DataKd:  5.00E+4nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147125(US8957075, Table 1 Compound 20)
Affinity DataKd:  7.20E+3nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147124(US8957075, Table 1 Compound 19 | US8957075, Table ...)
Affinity DataKd:  4.10E+3nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147127(US8957075, Table 1 Compound 22)
Affinity DataKd:  9.00E+3nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147128(US8957075, Table 1 Compound 23)
Affinity DataKd:  6.00E+4nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147129(US8957075, Table 1 Compound 24)
Affinity DataKd:  1.25E+5nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147130(US8957075, Table 1 Compound 25)
Affinity DataKd:  5.00E+4nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147119(US8957075, Table 1 Compound 14 | US8957075, Table ...)
Affinity DataKd:  7.00E+3nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147132(US8957075, Table 1 Compound 27)
Affinity DataKd:  4.00E+3nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147133(US8957075, Table 1 Compound 28)
Affinity DataKd:  400nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147121(US8957075, Table 1 Compound 16)
Affinity DataKd:  1.50E+4nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147120(US8957075, Table 1 Compound 15)
Affinity DataKd:  2.10E+4nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147119(US8957075, Table 1 Compound 14 | US8957075, Table ...)
Affinity DataKd:  5.70E+3nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147118(US8957075, Table 1 Compound 13)
Affinity DataKd:  5.60E+3nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147117(US8957075, Table 1 Compound 12)
Affinity DataKd:  1.60E+3nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147116(US8957075, Table 1 Compound 11)
Affinity DataKd:  3.20E+3nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147115(US8957075, Table 1 Compound 10)
Affinity DataKd:  1.10E+4nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147114(US8957075, Table 1 Compound 9)
Affinity DataKd:  5.20E+4nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147113(US8957075, Table 1 Compound 8)
Affinity DataKd:  2.00E+4nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147112(US8957075, Table 1 Compound 7)
Affinity DataKd:  9.70E+4nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM51358(2-keto-N-[2-keto-1-phenyl-2-[4-(2-pyridyl)piperazi...)
Affinity DataKd:  4.20E+3nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147111(US8957075, Table 1 Compound 5)
Affinity DataKd:  3.70E+4nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147110(US8957075, Table 1 Compound 4)
Affinity DataKd:  2.00E+3nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147109(US8957075, Table 1 Compound 3)
Affinity DataKd:  6.60E+3nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147107(US8957075, Table 1 Compound 1)
Affinity DataKd:  7.40E+3nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
President and Fellows of Harvard College

US Patent
LigandPNGBDBM147108(US8957075, Table 1 Compound 2)
Affinity DataKd:  6.30E+3nMAssay Description:384-well plates (Costar #3654) were filled using a liquid handling robot with 20 uL of a mixture of 50 nM of a fluorescein-linked UDP-GlcNAc analog (...More data for this Ligand-Target Pair
In DepthDetails US Patent