TargetTranslocator protein(Rattus norvegicus (rat))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Binding affinity for peripheral benzodiazepine receptor of rat kidneyMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Binding affinity for peripheral benzodiazepine receptor of rat kidneyMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Michigan Medical Center
Curated by ChEMBL
University Of Michigan Medical Center
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Binding affinity for peripheral benzodiazepine receptor of rat kidneyMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Mus musculus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 0.0370nMAssay Description:Inhibition of [3H]nicotine binding to alpha4 nicotinic acetylcholine receptor in Mus musculus (mouse) M10 cells co-expressing beta2 nicotinic acetylc...More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 0.370nMAssay Description:Inhibition of [3H]IMI binding to Drosophila melanogaster neuronal acetylcholine receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Mus musculus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of [3H]nicotine binding to alpha4 nicotinic acetylcholine receptor in Mus musculus (mouse) M10 cells co-expressing beta2 nicotinic acetylc...More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Inhibition of [3H]IMI binding to Drosophila melanogaster neuronal acetylcholine receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Mus musculus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Inhibition of [3H]nicotine binding to alpha4 nicotinic acetylcholine receptor in Mus musculus (mouse) M10 cells co-expressing beta2 nicotinic acetylc...More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Inhibition of [3H]IMI binding to Drosophila melanogaster neuronal acetylcholine receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Mus musculus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of [3H]nicotine binding to alpha4 nicotinic acetylcholine receptor in Mus musculus (mouse) M10 cells co-expressing beta2 nicotinic acetylc...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Mus musculus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 8.20nMAssay Description:Inhibition of [3H]nicotine binding to alpha4 nicotinic acetylcholine receptor in Mus musculus (mouse) M10 cells co-expressing beta2 nicotinic acetylc...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of [3H]nicotine binding to alpha3 nicotinic acetylcholine receptor in Homo sapiens (human) SH-SY5Y cells co-expressing beta2beta4alpha5 Ni...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of [3H]alpha-BGT binding to alpha7 nicotinic acetylcholine receptor in Homo sapiens (human) SH-SY5Y cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of [3H]nicotine binding to alpha3 nicotinic acetylcholine receptor in Homo sapiens (human) SH-SY5Y cells co-expressing beta2beta4alpha5 Ni...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Mus musculus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of [3H]nicotine binding to alpha4 nicotinic acetylcholine receptor in Mus musculus (mouse) M10 cells co-expressing beta2 nicotinic acetylc...More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of [3H]alpha-BGT binding to alpha1 nicotinic acetylcholine receptor in Homo sapiens (human) TE671 cells co-expressing gammaalpha1deltabeta...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of [3H]nicotine binding to alpha3 nicotinic acetylcholine receptor in Homo sapiens (human) SH-SY5Y cells co-expressing beta2beta4alpha5 Ni...More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 185nMAssay Description:Inhibition of [3H]IMI binding to Drosophila melanogaster neuronal acetylcholine receptorMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of [3H]IMI binding to Drosophila melanogaster neuronal acetylcholine receptorMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of [3H]IMI binding to Drosophila melanogaster neuronal acetylcholine receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 660nMAssay Description:Evaluated for inhibition of bovine adrenal cortical mitochondrial 11 beta-hydroxylaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Mus musculus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 860nMAssay Description:Inhibition of [3H]nicotine binding to alpha4 nicotinic acetylcholine receptor in Mus musculus (mouse) M10 cells co-expressing beta2 nicotinic acetylc...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of [3H]alpha-BGT binding to alpha7 nicotinic acetylcholine receptor in Homo sapiens (human) SH-SY5Y cellsMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibition of [3H]IMI binding to Drosophila melanogaster neuronal acetylcholine receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.53E+3nMAssay Description:Evaluated for inhibition of bovine adrenal cortical mitochondrial 11 beta-hydroxylaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.63E+3nMAssay Description:Evaluated for inhibition of bovine adrenal cortical mitochondrial 11 beta-hydroxylaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Mus musculus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of [3H]nicotine binding to alpha4 nicotinic acetylcholine receptor in Mus musculus (mouse) M10 cells co-expressing beta2 nicotinic acetylc...More data for this Ligand-Target Pair
Affinity DataIC50: 2.64E+3nMAssay Description:Evaluated for inhibition of bovine adrenal cortical mitochondrial 11 beta-hydroxylaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Evaluated for inhibition of bovine adrenal cortical mitochondrial 11 beta-hydroxylaseMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit beta-like 2(Drosophila melanogaster)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of [3H]IMI binding to Drosophila melanogaster neuronal acetylcholine receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of [3H]alpha-BGT binding to alpha7 nicotinic acetylcholine receptor in Homo sapiens (human) SH-SY5Y cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.78E+3nMAssay Description:Evaluated for inhibition of bovine adrenal cortical mitochondrial 11 beta-hydroxylaseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.36E+3nMAssay Description:Evaluated for inhibition of bovine adrenal cortical mitochondrial 11 beta-hydroxylaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of [3H]alpha-BGT binding to alpha7 nicotinic acetylcholine receptor in Homo sapiens (human) SH-SY5Y cellsMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of [3H]alpha-BGT binding to alpha1 nicotinic acetylcholine receptor in Homo sapiens (human) TE671 cells co-expressing gammaalpha1deltabeta...More data for this Ligand-Target Pair
Affinity DataIC50: 7.05E+3nMAssay Description:Evaluated for inhibition of bovine adrenal cortical mitochondrial 11 beta-hydroxylaseMore data for this Ligand-Target Pair
Affinity DataIC50: 7.25E+3nMAssay Description:Evaluated for inhibition of bovine adrenal cortical mitochondrial 11 beta-hydroxylaseMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMAssay Description:Evaluated for inhibition of bovine adrenal cortical mitochondrial 11 beta-hydroxylaseMore data for this Ligand-Target Pair
Affinity DataIC50: 7.72E+3nMAssay Description:Evaluated for inhibition of bovine adrenal cortical mitochondrial 11 beta-hydroxylaseMore data for this Ligand-Target Pair
Affinity DataIC50: 7.83E+3nMAssay Description:Evaluated for inhibition of bovine adrenal cortical mitochondrial 11 beta-hydroxylaseMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of [3H]alpha-BGT binding to alpha1 nicotinic acetylcholine receptor in Homo sapiens (human) TE671 cells co-expressing gammaalpha1deltabeta...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of [3H]alpha-BGT binding to alpha7 nicotinic acetylcholine receptor in Homo sapiens (human) SH-SY5Y cellsMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of [3H]alpha-BGT binding to alpha1 nicotinic acetylcholine receptor in Homo sapiens (human) TE671 cells co-expressing gammaalpha1deltabeta...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of [3H]nicotine binding to alpha3 nicotinic acetylcholine receptor in Homo sapiens (human) SH-SY5Y cells co-expressing beta2beta4alpha5 Ni...More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of [3H]alpha-BGT binding to alpha1 nicotinic acetylcholine receptor in Homo sapiens (human) TE671 cells co-expressing gammaalpha1deltabeta...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of [3H]alpha-BGT binding to alpha7 nicotinic acetylcholine receptor in Homo sapiens (human) SH-SY5Y cellsMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 8.10E+4nMAssay Description:Inhibition of [3H]alpha-BGT binding to alpha1 nicotinic acetylcholine receptor in Homo sapiens (human) TE671 cells co-expressing gammaalpha1deltabeta...More data for this Ligand-Target Pair
Affinity DataIC50: 8.75E+4nMAssay Description:Evaluated for inhibition of bovine adrenal cortical mitochondrial 11 beta-hydroxylaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]alpha-BGT binding to alpha7 nicotinic acetylcholine receptor in Homo sapiens (human) SH-SY5Y cellsMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of [3H]alpha-BGT binding to alpha1 nicotinic acetylcholine receptor in Homo sapiens (human) TE671 cells co-expressing gammaalpha1deltabeta...More data for this Ligand-Target Pair