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Found 19 with Last Name = 'lee' and Initial = 'rb'
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiled plasmid DNA formation after 30 mins by electrophoretic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50184425(CHEMBL206161 | Purealin)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50117089(CHEMBL204484 | CHEMBL83995 | N-[2-(2-Amino-3H-imid...)
Affinity DataIC50:  4.20E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50184421(3-[4-(3-aminopropoxy)-3-bromophenyl]-2-hydroxyimin...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50184423(3-[2-(3-aminopropoxy)-3,5-dibromophenyl]-N-[2-(4-c...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50184424(3-[2-(3-aminopropoxy)-3,5-dichlorophenyl]-2-hydrox...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50184426(3-[4-(3-aminopropoxy)-3-bromophenyl]-N-[2-(4-chlor...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50184427(CHEMBL206373 | Lipopurealin A)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50184420(3-[2-(3-aminopropoxy)-3,5-dibromophenyl]-2-hydroxy...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM21691(1-ethyl-7-methyl-4-oxo-1,4-dihydro-1,8-naphthyridi...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiled plasmid DNA formation after 30 mins by electrophoretic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50027668(CHEMBL3357531)
Affinity DataIC50:  2.50E+5nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiled plasmid DNA formation after 30 mins by electrophoretic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50027673(Olympicin A)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiled plasmid DNA formation after 30 mins by electrophoretic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50027665((E)-1-(2,4-dihydroxyphenyl)-3-(2-allyloxyphenyl)-2...)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiled plasmid DNA formation after 30 mins by electrophoretic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50027672(CHEMBL3357489)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiled plasmid DNA formation after 30 mins by electrophoretic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50027671(CHEMBL3357510)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiled plasmid DNA formation after 30 mins by electrophoretic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50027670(CHEMBL3357527)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiled plasmid DNA formation after 30 mins by electrophoretic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50027669(CHEMBL3357528)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiled plasmid DNA formation after 30 mins by electrophoretic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50027667(CHEMBL3357537)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiled plasmid DNA formation after 30 mins by electrophoretic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50027666(CHEMBL3357535)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiled plasmid DNA formation after 30 mins by electrophoretic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed