TargetProstaglandin E synthase(Homo sapiens (Human))
Eberhard Karls University Tuebingen
Curated by ChEMBL
Eberhard Karls University Tuebingen
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as residual enzyme activity after 1 min by measuring PGE2 level...More data for this Ligand-Target Pair
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Eberhard Karls University Tuebingen
Curated by ChEMBL
Eberhard Karls University Tuebingen
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Binding affinity to FLAPMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of human H-FABP by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibition of human A-FABP by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:Inhibition of human A-FABP by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 96nMAssay Description:Inhibition of human A-FABP by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 98nMAssay Description:Inhibition of human A-FABP by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 570nMAssay Description:In vitro inhibitory concentration against adipocyte fatty acid binding protein(A-FABP)More data for this Ligand-Target Pair
Affinity DataIC50: 580nMAssay Description:Inhibition of human A-FABP by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Inhibition of human A-FABP by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 680nMAssay Description:Inhibition of human H-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 710nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 720nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 730nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 780nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:In vitro inhibitory concentration against adipocyte fatty acid binding protein(A-FABP)More data for this Ligand-Target Pair
Affinity DataIC50: 830nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 930nMAssay Description:In vitro inhibitory concentration against adipocyte fatty acid binding protein(A-FABP)More data for this Ligand-Target Pair
Affinity DataIC50: 970nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:In vitro inhibitory concentration against adipocyte fatty acid binding protein(A-FABP)More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro inhibitory concentration against epithelial fatty acid binding protein(E-FABP)More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:In vitro inhibitory concentration against adipocyte fatty acid binding protein(A-FABP)More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:In vitro inhibitory concentration against adipocyte fatty acid binding protein(A-FABP)More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro inhibitory concentration against adipocyte fatty acid binding protein(A-FABP)More data for this Ligand-Target Pair
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:In vitro inhibitory concentration against intestinal fatty acid binding protein(I-FABP)More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Eberhard Karls University Tuebingen
Curated by ChEMBL
Eberhard Karls University Tuebingen
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as residual enzyme activity after 1 min by measuring PGE2 level...More data for this Ligand-Target Pair
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.03E+3nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Eberhard Karls University Tuebingen
Curated by ChEMBL
Eberhard Karls University Tuebingen
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as residual enzyme activity after 1 min by measuring PGE2 level...More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Eberhard Karls University Tuebingen
Curated by ChEMBL
Eberhard Karls University Tuebingen
Curated by ChEMBL
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as residual enzyme activity after 1 min by measuring PGE2 level...More data for this Ligand-Target Pair
Affinity DataIC50: 2.39E+3nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:In vitro inhibitory concentration against adipocyte fatty acid binding protein(A-FABP)More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:In vitro inhibitory concentration against adipocyte fatty acid binding protein(A-FABP)More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:In vitro inhibitory concentration against heart and muscle fatty acid binding protein(H-FABP)More data for this Ligand-Target Pair
Affinity DataIC50: 2.68E+3nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibitory concentration against epithelial fatty acid binding protein(E-FABP)More data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human A-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:In vitro inhibitory concentration against adipocyte fatty acid binding protein(A-FABP)More data for this Ligand-Target Pair