Compile Data Set for Download or QSAR
maximum 50k data
Found 164 with Last Name = 'liu' and Initial = 'zy'
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of TrkAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of Flt3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fgr(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of FgrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of BTKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase SIK1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of SIKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of PhKg2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  8.70nMAssay Description:Inhibition of FGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50014323(2-PHENYL-4H-BENZO[H]CHROMEN-4-ONE | 2-Phenyl-benzo...)
Affinity DataIC50:  12nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate incubated for 5 mins followed by NADPH addition and measured after 20 mi...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  13.4nMAssay Description:Inhibition of SAPK2aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  17.2nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  18.2nMAssay Description:Inhibition of cSrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM8610(1-[4-(4-{[(2R,4S)-2-(2,4-dichlorophenyl)-2-(1H-imi...)
Affinity DataIC50:  22nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate incubated for 5 mins followed by NADPH addition and measured after 20 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTestis-specific serine/threonine-protein kinase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  30.6nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  34.1nMAssay Description:Inhibition of ALKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50121975((6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2...)
Affinity DataIC50:  36nMAssay Description:Inhibition of CYP2D6 in human liver microsomes using dextromethorphan as substrate incubated for 5 mins followed by NADPH addition and measured after...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  44.3nMAssay Description:Inhibition of MLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  64nMAssay Description:Inhibition of FLT4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  68.3nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  72.2nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase WNK3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50:  99.8nMAssay Description:Inhibition of WNK3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129663(3-But-3-enoylamino-pyridine-2-carboxylic acid thia...)
Affinity DataIC50:  130nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129648(3-(4-Methyl-pent-3-enoylamino)-pyridine-2-carboxyl...)
Affinity DataIC50:  140nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129660(3-(3-Methyl-but-3-enoylamino)-pyridine-2-carboxyli...)
Affinity DataIC50:  150nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM17847(CHEMBL327579 | pyridine-2-carboxylic acid inhibito...)
Affinity DataIC50:  180nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129642(CHEMBL86427 | Phenyl-acetic acid 2-(thiazol-2-ylca...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129640(3-(3-Methyl-but-2-enoylamino)-pyridine-2-carboxyli...)
Affinity DataIC50:  220nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129648(3-(4-Methyl-pent-3-enoylamino)-pyridine-2-carboxyl...)
Affinity DataIC50:  240nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129672(3-Propionylamino-pyridine-2-carboxylic acid thiazo...)
Affinity DataIC50:  260nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129672(3-Propionylamino-pyridine-2-carboxylic acid thiazo...)
Affinity DataIC50:  260nMAssay Description:Inhibitory concentration against Escherichia coli methionine aminopeptidase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129657(3-(2-Fluoro-benzoylamino)-pyridine-2-carboxylic ac...)
Affinity DataIC50:  280nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129674(3-(2-Methyl-but-2-enoylamino)-pyridine-2-carboxyli...)
Affinity DataIC50:  280nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129669(3-(5-Methyl-hex-4-enoylamino)-pyridine-2-carboxyli...)
Affinity DataIC50:  310nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129649(CHEMBL315098 | Cyclohexanecarboxylic acid 2-(thiaz...)
Affinity DataIC50:  320nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129635(3-Formylamino-pyridine-2-carboxylic acid thiazol-2...)
Affinity DataIC50:  320nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129635(3-Formylamino-pyridine-2-carboxylic acid thiazol-2...)
Affinity DataIC50:  330nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM17849(3-(2,2-dimethylpropanamido)-N-(1,3-thiazol-2-yl)py...)
Affinity DataIC50:  340nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129670(3-(2,2,2-Trifluoro-acetylamino)-pyridine-2-carboxy...)
Affinity DataIC50:  340nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129672(3-Propionylamino-pyridine-2-carboxylic acid thiazo...)
Affinity DataIC50:  350nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129672(3-Propionylamino-pyridine-2-carboxylic acid thiazo...)
Affinity DataIC50:  350nMAssay Description:Inhibitory concentration against Saccharomyces cerevisiae methionine aminopeptidase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129656(3-Hexanoylamino-pyridine-2-carboxylic acid thiazol...)
Affinity DataIC50:  380nMAssay Description:Inhibitory concentration against Escherichia coli methionine aminopeptidase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129656(3-Hexanoylamino-pyridine-2-carboxylic acid thiazol...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129650(CHEMBL314448 | Propionic acid 2-(thiazol-2-ylcarba...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129663(3-But-3-enoylamino-pyridine-2-carboxylic acid thia...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129641(2-Methyl-but-2-enoic acid 2-(thiazol-2-ylcarbamoyl...)
Affinity DataIC50:  390nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129666(3-Phenylacetylamino-pyridine-2-carboxylic acid thi...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129646(3-Methyl-but-2-enoic acid 2-(thiazol-2-ylcarbamoyl...)
Affinity DataIC50:  490nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM17849(3-(2,2-dimethylpropanamido)-N-(1,3-thiazol-2-yl)py...)
Affinity DataIC50:  540nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129642(CHEMBL86427 | Phenyl-acetic acid 2-(thiazol-2-ylca...)
Affinity DataIC50:  540nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Saccharomyces cerevisiae)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129675(2-Methoxy-benzoic acid 2-(thiazol-2-ylcarbamoyl)-p...)
Affinity DataIC50:  550nMAssay Description:Inhibitory activity against type I methionine aminopeptidase from Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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