Affinity DataKi: 600nMAssay Description:Inhibition of Trypanosoma brucei TryR assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Inhibition of Crithidia fasciculata TryR overexpressed in escherichia coli assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of Trypanosoma brucei TryR assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+3nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 7.50E+3nMAssay Description:Mixed-type inhibition of Trypanosoma brucei trypanothione reductase assessed as enzyme-inhibitor complex using varying levels of TS2 as substrate in ...More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+4nMAssay Description:Inhibition of Trypanosoma brucei TryR assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.59E+4nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 1.90E+4nMAssay Description:Inhibition of Trypanosoma brucei TryR assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+4nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+4nMAssay Description:Mixed-type inhibition of Trypanosoma brucei trypanothione reductase assessed as enzyme-inhibitor-substrate complex using varying levels of TS2 as sub...More data for this Ligand-Target Pair
Affinity DataKi: 2.70E+4nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 3.70E+4nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 8.50E+4nMAssay Description:Inhibition of Crithidia fasciculata TryR overexpressed in escherichia coli assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 8.60E+4nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constant by TR assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 9.00E+4nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constant by TR assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of Trypanosoma brucei TryR assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+6nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constant in presence of NADPHMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: >2.00E+6nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constant in presence of NADPHMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: >2.00E+6nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constant in presence of NADPHMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: >2.00E+6nMAssay Description:Inhibition of Trypanosoma cruzi TryR assessed as inhibition constant in presence of NADPHMore data for this Ligand-Target Pair
Ligand Info
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Cnrs Upr2301
Curated by ChEMBL
Cnrs Upr2301
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesyl pyrophosphate and Dansyl-GCVLS peptide after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Cnrs Upr2301
Curated by ChEMBL
Cnrs Upr2301
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesyl pyrophosphate and Dansyl-GCVLS peptide after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of Crithidia fasciculata His tagged TryS in presence of ATP by LDH/PK assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacteria using GRSRSRSRSRSR as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Cnrs Upr2301
Curated by ChEMBL
Cnrs Upr2301
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesyl pyrophosphate and Dansyl-GCVLS peptide after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Cnrs Upr2301
Curated by ChEMBL
Cnrs Upr2301
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesyl pyrophosphate and Dansyl-GCVLS peptide after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant human CK1 epsilon expressed in baculovirus infected Sf9 cells using RRKHAAIGSpAYSITA as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacteria using GRSRSRSRSRSR as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant human CK1 epsilon expressed in baculovirus infected Sf9 cells using RRKHAAIGSpAYSITA as substrateMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Cnrs Upr2301
Curated by ChEMBL
Cnrs Upr2301
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesyl pyrophosphate and Dansyl-GCVLS peptide after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of Trypanosoma cruzi TryRMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human CK1 epsilon expressed in baculovirus infected Sf9 cells using RRKHAAIGSpAYSITA as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacteria using GRSRSRSRSRSR as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Cnrs Upr2301
Curated by ChEMBL
Cnrs Upr2301
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesyl pyrophosphate and Dansyl-GCVLS peptide after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Cnrs Upr2301
Curated by ChEMBL
Cnrs Upr2301
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesyl pyrophosphate and Dansyl-GCVLS peptide after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Cnrs Upr2301
Curated by ChEMBL
Cnrs Upr2301
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesyl pyrophosphate and Dansyl-GCVLS peptide after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Cnrs Upr2301
Curated by ChEMBL
Cnrs Upr2301
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesyl pyrophosphate and Dansyl-GCVLS peptide after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of human recombinant CDK9/CyclinT expressed in baculovirus infected Sf9 cells using YSPTSPSYSPTSPSYSPTSPSKKK as substrate in presence of [...More data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:Inhibition of Trypanosoma cruzi TryRMore data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacteria using GRSRSRSRSRSR as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of Trypanosoma cruzi TryRMore data for this Ligand-Target Pair
Ligand Info
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Cnrs Upr2301
Curated by ChEMBL
Cnrs Upr2301
Curated by ChEMBL
Affinity DataIC50: 640nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesyl pyrophosphate and Dansyl-GCVLS peptide after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Cnrs Upr2301
Curated by ChEMBL
Cnrs Upr2301
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesyl pyrophosphate and Dansyl-GCVLS peptide after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Inhibition of Trypanosoma brucei TryRMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 800nMAssay Description:Inhibition of Trypanosoma cruzi TryRMore data for this Ligand-Target Pair
Ligand Info