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Found 65 with Last Name = 'luetje' and Initial = 'cw'
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86041(NFEP)
Affinity DataKi:  0.00240nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86042(NEP)
Affinity DataKi:  0.00310nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86041(NFEP)
Affinity DataKi:  0.00380nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.00400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86042(NEP)
Affinity DataKi:  0.00850nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86041(NFEP)
Affinity DataKi:  0.00920nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.0130nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86042(NEP)
Affinity DataKi:  0.0280nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor, nicotinic alpha 1(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.0440nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.0550nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86045(NNEP)
Affinity DataKi:  0.0620nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86045(NNEP)
Affinity DataKi:  0.0770nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor nicotinic alpha 5 subunit(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86040(NBEP)
Affinity DataKi:  0.220nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86045(NNEP)
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor, nicotinic alpha 1(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86041(NFEP)
Affinity DataKi:  0.480nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86041(NFEP)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor nicotinic alpha 5 subunit(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86041(NFEP)
Affinity DataKi:  2.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor, nicotinic alpha 1(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86042(NEP)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86042(NEP)
Affinity DataKi:  3.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86045(NNEP)
Affinity DataKi:  3.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor, nicotinic alpha 1(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86045(NNEP)
Affinity DataKi:  4.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor nicotinic alpha 5 subunit(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86045(NNEP)
Affinity DataKi:  7.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86044(NTEP)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinergic receptor nicotinic alpha 5 subunit(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86042(NEP)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50063218((R)-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]...)
Affinity DataKi:  14nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM50063218((R)-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]...)
Affinity DataKi:  30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50166908(5,8,14-triazatetracyclo[10.3.1.02,11.04,9]hexadeca...)
Affinity DataKi:  32.5nMAssay Description:Displacement of [125I]iodoMLA from rat cerebral cortex alpha7 nAChR at 50 nM incubated for 2 hrs by microplate scintillation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinergic receptor, nicotinic alpha 1(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM50063218((R)-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]...)
Affinity DataKi:  85nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM50063218((R)-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]...)
Affinity DataKi:  87nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86043(NDMNEP)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM50119631(5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-pyridin-2-ol | C...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86043(NDMNEP)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50119631(5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-pyridin-2-ol | C...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86044(NTEP)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86043(NDMNEP)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM50119631(5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-pyridin-2-ol | C...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM86044(NTEP)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinergic receptor nicotinic alpha 5 subunit(Xenopus)
University of Miami

Curated by PDSP Ki Database
LigandPNGBDBM50063218((R)-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]...)
Affinity DataKi:  300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50395217(CHEMBL2164667 | US9150581, RTI-7527-168)
Affinity DataKi:  1.87E+3nMAssay Description:Displacement of [125I]iodoMLA from rat cerebral cortex alpha7 nAChR at 50 nM incubated for 2 hrs by microplate scintillation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50395221(CHEMBL2164663 | US9150581, RTI-7527-153)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [125I]iodoMLA from rat cerebral cortex alpha7 nAChR at 50 nM incubated for 2 hrs by microplate scintillation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50395219(CHEMBL2164665 | US9150581, RTI-7527-193)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [125I]iodoMLA from rat cerebral cortex alpha7 nAChR at 50 nM incubated for 2 hrs by microplate scintillation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50395220(CHEMBL2164664 | US9150581, RTI-7527-(+/-)-154)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [125I]iodoMLA from rat cerebral cortex alpha7 nAChR at 50 nM incubated for 2 hrs by microplate scintillation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50151495(2-[6-Fluoro-5-(4-nitro-phenyl)-pyridin-3-yl]-7-aza...)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [125I]iodoMLA from rat cerebral cortex alpha7 nAChR at 50 nM incubated for 2 hrs by microplate scintillation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50395218(CHEMBL2164666 | US9150581, RTI-7527-192)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [125I]iodoMLA from rat cerebral cortex alpha7 nAChR at 50 nM incubated for 2 hrs by microplate scintillation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50171007(4-[5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-2-fluoro-pyri...)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [125I]iodoMLA from rat cerebral cortex alpha7 nAChR at 50 nM incubated for 2 hrs by microplate scintillation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50448763(CHEMBL3128030)
Affinity DataIC50:  3.90E+3nMAssay Description:Antagonist activity at rat alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current by two-elect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50395221(CHEMBL2164663 | US9150581, RTI-7527-153)
Affinity DataIC50:  4.00E+3nMAssay Description:Antagonist activity at rat alpha7 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced response after 2 to 6 day...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50448767(CHEMBL3128029)
Affinity DataIC50:  7.90E+3nMAssay Description:Antagonist activity at rat alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current by two-elect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50448766(CHEMBL3128031)
Affinity DataIC50:  8.00E+3nMAssay Description:Antagonist activity at rat alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current by two-elect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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