Affinity DataIC50: 29nMAssay Description:Inhibition of CDK6 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of CDK6 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of CDK6 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibition of CDK6 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of CDK6 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 89nMAssay Description:Inhibition of recombinant full length human N-terminal GST-tagged C-terminal His6-tagged MEK1 expressed in Escherichia coli using myelin basic protei...More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant full length human N-terminal GST-tagged C-terminal His6-tagged MEK1 expressed in Escherichia coli using myelin basic protei...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 522nMAssay Description:Inhibition of CDK1 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 569nMAssay Description:Inhibition of CDK1 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 571nMAssay Description:Inhibition of CDK1 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 584nMAssay Description:Inhibition of CDK1 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Inhibition of MEK1 in BRAF mutant human A549 cells assessed as reduction in ERK1/2 phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 610nMAssay Description:Inhibition of CDK1 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of PI3Kgamma after 4 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.42E+3nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.42E+3nMAssay Description:Inhibition of CDK7 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of CDK7 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.65E+3nMAssay Description:Inhibition of CDK7 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.79E+3nMAssay Description:Inhibition of CDK7 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.88E+3nMAssay Description:Inhibition of CDK7 (unknown origin) using histone H1 as substrate after 10 mins in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 2.87E+3nMAssay Description:Inhibition of PI3Kgamma after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 3.12E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.12E+3nMAssay Description:Inhibition of PI3Kgamma after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 5.74E+3nMAssay Description:Inhibition of PI3Kgamma after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 6.48E+3nMAssay Description:Inhibition of PI3Kgamma after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 6.57E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 7.22E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 7.41E+3nMAssay Description:Inhibition of PI3Kgamma after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 8.03E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of Aurora A (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 9.08E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 9.36E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.56E+4nMAssay Description:Inhibition of FAK in human MCF7 cellsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University
Curated by ChEMBL
Anhui Agricultural University
Curated by ChEMBL
Affinity DataIC50: 1.76E+4nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair