TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 138nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 229nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 282nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 327nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 331nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 383nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 665nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 2.83E+3nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 3.62E+3nMAssay Description:Displacement of [5,6-3H]-nicotinic acid from recombinant human HCA2 receptor expressed in Flp-IN HEK cell membranes after 2 hrs by microbeta counting...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 36nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 80nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 9nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 3.37E+3nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 5.61E+3nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 1.01E+3nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 3.64E+4nMAssay Description:Agonist activity at human HCA2 receptor expressed in Flp-In-293 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 1.25E+4nMAssay Description:Agonist activity at human HCA2 receptor expressed in Flp-In-293 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 2.63E+4nMAssay Description:Agonist activity at human HCA2 receptor expressed in Flp-In-293 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 5.16E+4nMAssay Description:Agonist activity at human HCA2 receptor expressed in Flp-In-293 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 5.80E+3nMAssay Description:Agonist activity at human HCA2 receptor expressed in Flp-In-293 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 6.30E+3nMAssay Description:Agonist activity at human HCA2 receptor expressed in Flp-In-293 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 6.80E+3nMAssay Description:Agonist activity at human HCA2 receptor expressed in Flp-In-293 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 2.74E+4nMAssay Description:Agonist activity at human HCA2 receptor expressed in Flp-In-293 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 4.10E+3nMAssay Description:Agonist activity at human HCA2 receptor expressed in Flp-In-293 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 8.30E+3nMAssay Description:Agonist activity at human HCA2 receptor expressed in Flp-In-293 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 260nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 190nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 450nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 1.96E+4nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 720nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 2.98E+3nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 70nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Latvian Institute Of Organic Synthesis
Curated by ChEMBL
Affinity DataEC50: 630nMAssay Description:Agonist activity at recombinant human HCA2 receptor expressed in Flp-IN HEK cells assessed as reduction in forskolin-stimulated cAMP accumulation mea...More data for this Ligand-Target Pair