Affinity DataKi: 0.5nMAssay Description:Competitive inhibition of recombinant TAK1-TAB1 assessed as [33P]gamma-ATP incorporation into substrate histone H1 peptide by filter plate assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity at [3H]CD radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity at [3H]QNB and GppNHp radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 0.780nMAssay Description:Binding affinity at [3H]QNB and GppNHp radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding activity to muscarinic acetylcholine receptor in rat heart, assayed using [3H]-QNB as a radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding activity to the muscarinic acetylcholine receptor in rat cortex, assayed using [3H]CD as a radioligand.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity at [3H]CD radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity at [3H]CD radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding activity to the muscarinic acetylcholine receptor in rat cortex, assayed using [3H]CD as a radioligand.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Binding affinity at [3H]QNB radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity at [3H]CD radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Binding affinity at [3H]QNB and GppNHp radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Binding affinity at [3H]PZ radiolabeled muscarinic M1 receptor in rat cortex.More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding activity to the muscarinic acetylcholine receptor in rat cortex, assayed using [3H]PZ as a radioligand.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Binding affinity at [3H]QNB radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 56nMAssay Description:Binding affinity at [3H]CD radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Competitive inhibition of recombinant TAK1-TAB1 assessed as [33P]gamma-ATP incorporation into substrate histone H1 peptide by filter plate assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Binding affinity at [3H]CD radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Binding affinity at [3H]QNB and GppNHp radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Binding affinity at [3H]CD radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Binding affinity at [3H]QNB radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding activity to the muscarinic acetylcholine receptor in rat cortex, assayed using [3H]PZ as a radioligand.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Binding affinity at [3H]QNB radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Binding affinity at [3H]QNB radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding activity to muscarinic acetylcholine receptor in rat heart, assayed using [3H]-QNB as a radioligand.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 71nMAssay Description:Binding affinity at [3H]CD radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Binding affinity at [3H]CD radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Binding affinity at [3H]QNB radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Binding activity against Muscarinic acetylcholine receptor in rat cortex, using [3H]QNB as a radioligand.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Binding affinity at [3H]QNB radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding activity to the muscarinic acetylcholine receptor in rat cortex, assayed using [3H]PZ as a radioligand.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Binding affinity at [3H]QNB radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding activity to the muscarinic acetylcholine receptor in rat cortex, assayed using [3H]CD as a radioligand.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Binding affinity at [3H]QNB radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Binding affinity at [3H]PZ radiolabeled muscarinic M1 receptor in rat cortex.More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Competitive inhibition of recombinant TAK1-TAB1 assessed as [33P]gamma-ATP incorporation into substrate histone H1 peptide by filter plate assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Binding affinity at [3H]PZ radiolabeled muscarinic M1 receptor in rat cortex.More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding activity to muscarinic acetylcholine receptor in rat heart, assayed using [3H]QNB as a radioligand in the presence of Gpp(NH)p.More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding activity to the muscarinic acetylcholine receptor in rat cortex, assayed using [3H]PZ as a radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding activity to the muscarinic acetylcholine receptor in rat cortex, assayed using [3H]PZ as a radioligand.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Binding affinity at [3H]QNB and GppNHp radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Binding activity to the muscarinic acetylcholine receptor in rat cortex, assayed using [3H]PZ as a radioligand.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Binding affinity at [3H]QNB and GppNHp radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Competitive inhibition of recombinant TAK1-TAB1 assessed as [33P]gamma-ATP incorporation into substrate histone H1 peptide by filter plate assayMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Binding activity to the muscarinic acetylcholine receptor in rat cortex, assayed using [3H]PZ as a radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Binding activity to the muscarinic acetylcholine receptor in rat cortex, assayed using [3H]CD as a radioligand.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 240nMAssay Description:Binding affinity at [3H]CD radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Binding affinity at [3H]PZ radiolabeled muscarinic M1 receptor in rat cortex.More data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Competitive inhibition of recombinant TAK1-TAB1 assessed as [33P]gamma-ATP incorporation into substrate histone H1 peptide by filter plate assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Binding affinity at [3H]QNB and GppNHp radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair