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Found 11 with Last Name = 'mariotte' and Initial = 'am'
TargetTyrosinase(Homo sapiens (Human))
Umr-Cnrs 5063

Curated by ChEMBL
LigandPNGBDBM50180259((Z)-2-(4-hydroxybenzylidene)-4-hydroxybenzofuran-3...)
Affinity DataIC50:  3.17E+4nMAssay Description:Inhibitory activity against tyrosinase in human melanocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Umr-Cnrs 5063

Curated by ChEMBL
LigandPNGBDBM50180261((Z)-4,6-dihydroxy-2-(4-hydroxybenzylidene)benzofur...)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibitory activity against tyrosinase in human melanocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Homo sapiens (Human))
Umr-Cnrs 5063

Curated by ChEMBL
LigandPNGBDBM50180260((Z)-2-(4-Hydroxybenzylidene)-6-hydroxybenzofuran-3...)
Affinity DataIC50:  3.84E+4nMAssay Description:Inhibitory activity against tyrosinase in human melanocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
DéPartement De Pharmacochimie MoléCulaire Umr-Cnrs 5063

Curated by ChEMBL
LigandPNGBDBM50084978(3,5,7-trihydroxy-2-(4-methoxyphenyl)-4H-chromen-4-...)
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity of the compound to nucleotide-binding domain (NBD2) of P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
DéPartement De Pharmacochimie MoléCulaire Umr-Cnrs 5063

Curated by ChEMBL
LigandPNGBDBM50049391(3,5,7-Trihydroxyflavone | 3,5,7-triOH-flavone | 3,...)
Affinity DataKd:  5.90E+3nMAssay Description:Binding affinity of the compound to nucleotide-binding domain (NBD2) of P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
DéPartement De Pharmacochimie MoléCulaire Umr-Cnrs 5063

Curated by ChEMBL
LigandPNGBDBM50095342(2-(2,4-Dichloro-phenyl)-3,5,7-trihydroxy-chromen-4...)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity of the compound to nucleotide-binding domain (NBD2) of P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
DéPartement De Pharmacochimie MoléCulaire Umr-Cnrs 5063

Curated by ChEMBL
LigandPNGBDBM7462(3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-...)
Affinity DataKd:  6.70E+3nMAssay Description:Binding affinity of the compound to nucleotide-binding domain (NBD2) of P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
DéPartement De Pharmacochimie MoléCulaire Umr-Cnrs 5063

Curated by ChEMBL
LigandPNGBDBM50095340(2-(4-Fluoro-phenyl)-3,5,7-trihydroxy-chromen-4-one...)
Affinity DataKd:  6.80E+3nMAssay Description:Binding affinity of the compound to nucleotide-binding domain (NBD2) of P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
DéPartement De Pharmacochimie MoléCulaire Umr-Cnrs 5063

Curated by ChEMBL
LigandPNGBDBM50095338(2-(4-Benzhydryl-phenyl)-3,5,7-trihydroxy-chromen-4...)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity of the compound to nucleotide-binding domain (NBD2) of P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
DéPartement De Pharmacochimie MoléCulaire Umr-Cnrs 5063

Curated by ChEMBL
LigandPNGBDBM50095339(3,5,7-Trihydroxy-2-(4-iodo-phenyl)-chromen-4-one |...)
Affinity DataKd:  1.06E+3nMAssay Description:Binding affinity of the compound to nucleotide-binding domain (NBD2) of P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
DéPartement De Pharmacochimie MoléCulaire Umr-Cnrs 5063

Curated by ChEMBL
LigandPNGBDBM50095341(3,5,7-Trihydroxy-2-(4-octyl-phenyl)-chromen-4-one ...)
Affinity DataKd:  57nMAssay Description:Binding affinity of the compound to nucleotide-binding domain (NBD2) of P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed