Compile Data Set for Download or QSAR
maximum 50k data
Found 90 with Last Name = 'matsuoka' and Initial = 'k'
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338672(CHEMBL1209027 | Salaprinol)
Affinity DataIC50:  290nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataIC50:  750nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataIC50:  750nMAssay Description:Inhibition of rat small intestinal sucrase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50269567(CHEMBL515528 | Kynapcin-12)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50046279(CHEMBL3314376)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50394353(CHEMBL2159763)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of rat small intestinal sucrase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50333465((2R,3R,4R,5R,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50333465((2R,3R,4R,5R,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50263044(CHEMBL476960 | Voglibose)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338672(CHEMBL1209027 | Salaprinol)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338672(CHEMBL1209027 | Salaprinol)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50046278(CHEMBL3314375)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHemagglutinin(Influenza A virus (strain A/Aichi/2/1968 H3N2))
Saitama University

Curated by ChEMBL
LigandPNGBDBM50360450(CHEMBL1934618)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of Human influenza virus A/Aichi/2/68 (H3N2) hemagglutinin activity in chicken erythrocytes after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of rat small intestinal maltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50394351(CHEMBL2159632)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of rat small intestinal maltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHemagglutinin(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50360452(CHEMBL1934620)
Affinity DataIC50:  7.81E+3nMAssay Description:Inhibition of Human influenza virus A/PR/8/34 (H1N1) hemagglutinin activity in chicken erythrocytes after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHemagglutinin(Influenza A virus (strain A/Aichi/2/1968 H3N2))
Saitama University

Curated by ChEMBL
LigandPNGBDBM50360452(CHEMBL1934620)
Affinity DataIC50:  7.81E+3nMAssay Description:Inhibition of Human influenza virus A/Aichi/2/68 (H3N2) hemagglutinin activity in chicken erythrocytes after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHemagglutinin(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50360450(CHEMBL1934618)
Affinity DataIC50:  7.81E+3nMAssay Description:Inhibition of Human influenza virus A/PR/8/34 (H1N1) hemagglutinin activity in chicken erythrocytes after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341973(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5R,6S)-2,4,5,6,7-p...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341975(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5R,6R)-2,4,5,6,7-p...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50394352(CHEMBL2159631)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50046273(CHEMBL3314370)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50046275(CHEMBL3314372)
Affinity DataIC50:  1.49E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50046276(CHEMBL3314373)
Affinity DataIC50:  1.51E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50046188(CHEMBL3238007)
Affinity DataIC50:  1.52E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341972(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5S,6R)-2,4,5,6,7-p...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50394349(CHEMBL2159634)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50394350(CHEMBL2159633)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50046277(CHEMBL3314374)
Affinity DataIC50:  1.77E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50394348(CHEMBL2159635)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50394347(CHEMBL2159636)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341974(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5S,6S)-2,4,5,6,7-p...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341974(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5S,6S)-2,4,5,6,7-p...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50394351(CHEMBL2159632)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of rat small intestinal sucrase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50394353(CHEMBL2159763)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of rat small intestinal maltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50046272(CHEMBL3314369)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50046263(CHEMBL3314368)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50046274(CHEMBL3314371)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50394354(CHEMBL2159637)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of rat small intestinal sucrase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 90 total ) | Next | Last >>
Jump to: