TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.530nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.760nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 8.30nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 96nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 880nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 3.30E+3nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
Affinity DataKi: 4.30E+3nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.40E+3nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.540nMAssay Description:Inhibition of human placental DPP4 at pH 2More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human placental DPP4 at pH 2More data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of EGFR1 (unknown origin) after 1 hr in presence of adenosine 5'[gamma-33P]triphosphate by microbeta microplate counting methodMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human placental DPP4 at pH 8More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human placental DPP4 at pH 2More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:Inhibition of human placental DPP4 at pH 8More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Inhibition of human placental DPP4 at pH 2More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human placental DPP4 at pH 8More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human placental DPP4 at pH 8More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human placental DPP4 at pH 2More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: >2.30E+3nMAssay Description:Inhibition of human placental DPP4 at pH 8More data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of human recombinant DPP9 expressed in intact HEK293T cells after 2 hrsMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of recombinant human CDK2/cyclin A using histone H1 as substrate after 30 mins in presence of ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of recombinant full length human GST-fused DYRK1A expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of recombinant full length human GST-fused DYRK1A expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of recombinant full length human GST-fused DYRK1A expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of recombinant full length human GST-fused DYRK1A expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of recombinant mouse GST-fused CLK1 expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of ATP by scinti...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of recombinant mouse GST-fused CLK1 expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of ATP by scinti...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of recombinant mouse GST-fused CLK1 expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of ATP by scinti...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of recombinant mouse GST-fused CLK1 expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of ATP by scinti...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Rajiv Gandhi Proudyogiki Vishwavidyalaya
Curated by ChEMBL
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of recombinant mouse GST-fused CLK1 expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of ATP by scinti...More data for this Ligand-Target Pair