TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.530nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetProlyl endopeptidase(Homo sapiens (Human))
Tufts University Sackler School Of Biomedical Sciences
Curated by ChEMBL
Tufts University Sackler School Of Biomedical Sciences
Curated by ChEMBL
Affinity DataKi: 0.730nMAssay Description:Competitive inhibition of human PREP using Suc-GP-AMC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.760nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 8.30nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Tufts University Sackler School Of Biomedical Sciences
Curated by ChEMBL
Tufts University Sackler School Of Biomedical Sciences
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Competitive inhibition of human FAP using Suc-GP-AMC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 96nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:TP_TRANSPORTER: inhibition of Taurocholate uptake in membrane vesicles from Bsep-expressing Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 880nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 1.46E+3nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin uptake in Oatp2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Hospital
Curated by ChEMBL
University Hospital
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of BSP uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B3(Homo sapiens (Human))
University Hospital
Curated by ChEMBL
University Hospital
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of BSP uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 2B1(Homo sapiens (Human))
University Hospital
Curated by ChEMBL
University Hospital
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of BSP uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetProlyl endopeptidase(Homo sapiens (Human))
Tufts University Sackler School Of Biomedical Sciences
Curated by ChEMBL
Tufts University Sackler School Of Biomedical Sciences
Curated by ChEMBL
Affinity DataKi: 3.10E+3nMAssay Description:Competitive inhibition of human PREP using Suc-GP-AMC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 3.30E+3nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
Affinity DataKi: 3.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of Taurocholate uptake in membrane vesicles from Bsep-expressing Sf9 cellsMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 3.81E+3nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin uptake in Oatp2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+3nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 4.50E+3nMAssay Description:Competitive inhibition of human recombinant DPP4 using AP-pNA as substrate preincubated for 30 mins followed by substrate addition measured after 30 ...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Competitive inhibition of human recombinant DPP4 using AP-pNA as substrate preincubated for 30 mins followed by substrate addition measured after 30 ...More data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B3(Homo sapiens (Human))
University Hospital
Curated by ChEMBL
University Hospital
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of BSP uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B2(Rattus norvegicus)
University Of Zurich
Curated by ChEMBL
University Of Zurich
Curated by ChEMBL
Affinity DataKi: 6.10E+3nMAssay Description:TP_TRANSPORTER: inhibition of E1S uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 6.10E+3nMAssay Description:TP_TRANSPORTER: inhibition of Taurocholate uptake in membrane vesicles from Bsep-expressing Sf9 cellsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School Of Medicine
Curated by ChEMBL
Tufts University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 6.30E+3nMAssay Description:Competitive inhibition of human recombinant DPP4 using AP-pNA as substrate preincubated for 30 mins followed by substrate addition measured after 30 ...More data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
University Of Zurich
Curated by ChEMBL
University Of Zurich
Curated by ChEMBL
Affinity DataKi: 6.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 7.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 8.40E+3nMAssay Description:Inhibition of human recombinant DPP8 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.50E+3nMAssay Description:TP_TRANSPORTER: inhibition of Taurocholate uptake in membrane vesicle from Bsep-expressing Sf9-cellMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
University Of Zurich
Curated by ChEMBL
University Of Zurich
Curated by ChEMBL
Affinity DataKi: 9.27E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair