Affinity DataKi: 0.0398nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0501nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0501nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0501nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0501nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0501nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0501nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0525nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0575nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0603nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0631nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0631nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0631nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0759nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0794nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0794nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0794nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0794nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0794nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0794nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0977nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.117nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.126nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.126nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.126nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.126nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.126nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.132nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.141nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.158nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.158nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.158nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.158nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.158nMAssay Description:Displacement of [3H]neurokinin A from human NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.158nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot
Curated by ChEMBL
University Of Naples&Quot;Federico Ii&Quot
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot
Curated by ChEMBL
University Of Naples&Quot;Federico Ii&Quot
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.224nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.234nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.251nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.251nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.251nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot
Curated by ChEMBL
University Of Naples&Quot;Federico Ii&Quot
Curated by ChEMBL
Affinity DataKi: 0.251nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair