Compile Data Set for Download or QSAR
maximum 50k data
Found 154 with Last Name = 'michels' and Initial = 'pa'
TargetDihydrofolate reductase(Homo sapiens (Human))
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM18050(2-[(4-{[(2,4-diaminopteridin-6-yl)methyl](methyl)a...)
Affinity DataKi:  0.000340nMAssay Description:Inhibition of human DHFR by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetPteridine reductase 1(Leishmania major)
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398391(CHEMBL2178602)
Affinity DataKi:  30nMAssay Description:Inhibition of Leishmania major PTR1 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398394(CHEMBL1232702)
Affinity DataKi:  37nMAssay Description:Inhibition of Leishmania major PTR1 by spectrophotometric assayMore data for this Ligand-Target Pair
TargetATP-dependent 6-phosphofructokinase(Trypanosoma brucei)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446088(CHEMBL3108870)
Affinity DataKi:  52nMAssay Description:Competitive inhibition Trypanosoma brucei PFK using fructose-6-phosphate as substrate by Line-weaver Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398392(CHEMBL2178603)
Affinity DataKi:  60nMAssay Description:Inhibition of Leishmania major PTR1 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398390(CHEMBL2177120)
Affinity DataKi:  78nMAssay Description:Inhibition of Leishmania major PTR1 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398389(CHEMBL2178601)
Affinity DataKi:  100nMAssay Description:Inhibition of Leishmania major PTR1 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398395(CHEMBL1232399)
Affinity DataKi:  100nMAssay Description:Inhibition of Leishmania major PTR1 by spectrophotometric assayMore data for this Ligand-Target Pair
TargetPteridine reductase 1(Leishmania major)
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM18050(2-[(4-{[(2,4-diaminopteridin-6-yl)methyl](methyl)a...)
Affinity DataKi:  180nMAssay Description:Inhibition of Leishmania major PTR1 by spectrophotometric assayMore data for this Ligand-Target Pair
TargetPteridine reductase 1(Leishmania major)
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398396(CHEMBL2178600)
Affinity DataKi:  210nMAssay Description:Inhibition of Leishmania major PTR1 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma brucei)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446088(CHEMBL3108870)
Affinity DataKi:  240nMAssay Description:Mixed type inhibition Trypanosoma brucei PFK using ATP as substrate by Line-weaver Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398393(CHEMBL2178599)
Affinity DataKi:  390nMAssay Description:Inhibition of Leishmania major PTR1 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-6-phosphate 1-dehydrogenase(Trypanosoma brucei)
Universidade De SãO Paulo

Curated by ChEMBL
LigandPNGBDBM50236240(5alpha-androstan-3beta-OL-17-one | CHEMBL272195 | ...)
Affinity DataKi:  460nMAssay Description:Inhibition of Trypanosoma brucei G6PDH using NADP as substrate by Lineweaver-Burk plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-6-phosphate 1-dehydrogenase(Trypanosoma brucei)
Universidade De SãO Paulo

Curated by ChEMBL
LigandPNGBDBM50236240(5alpha-androstan-3beta-OL-17-one | CHEMBL272195 | ...)
Affinity DataKi:  490nMAssay Description:Inhibition of Trypanosoma brucei G6PDH using glucose-6-phosphate as substrate by Lineweaver-Burk plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398388(CHEMBL2178604)
Affinity DataKi:  590nMAssay Description:Inhibition of human DHFR by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM18050(2-[(4-{[(2,4-diaminopteridin-6-yl)methyl](methyl)a...)
Affinity DataKi:  600nMAssay Description:Inhibition of human TS by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398394(CHEMBL1232702)
Affinity DataKi:  800nMAssay Description:Inhibition of human DHFR by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-6-phosphate 1-dehydrogenase(Trypanosoma brucei)
Universidade De SãO Paulo

Curated by ChEMBL
LigandPNGBDBM50223368(3beta-hydroxyandrost-5-en-17-one | CHEMBL90593 | D...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of Trypanosoma brucei G6PDH using NADP as substrate by Lineweaver-Burk plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-6-phosphate 1-dehydrogenase(Trypanosoma brucei)
Universidade De SãO Paulo

Curated by ChEMBL
LigandPNGBDBM50223368(3beta-hydroxyandrost-5-en-17-one | CHEMBL90593 | D...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of Trypanosoma brucei G6PDH using glucose-6-phosphate as substrate by Lineweaver-Burk plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-6-phosphate 1-dehydrogenase(Homo sapiens (Human))
Universidade De SãO Paulo

Curated by ChEMBL
LigandPNGBDBM50236240(5alpha-androstan-3beta-OL-17-one | CHEMBL272195 | ...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human G6PDH using NADP as substrate by Lineweaver-Burk plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-6-phosphate 1-dehydrogenase(Homo sapiens (Human))
Universidade De SãO Paulo

Curated by ChEMBL
LigandPNGBDBM50236240(5alpha-androstan-3beta-OL-17-one | CHEMBL272195 | ...)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of human G6PDH using glucose-6-phosphate as substrate by Lineweaver-Burk plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPteridine reductase 1(Leishmania major)
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398388(CHEMBL2178604)
Affinity DataKi:  4.17E+3nMAssay Description:Inhibition of Leishmania major PTR1 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398391(CHEMBL2178602)
Affinity DataKi:  4.33E+3nMAssay Description:Inhibition of human DHFR by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398392(CHEMBL2178603)
Affinity DataKi:  4.68E+3nMAssay Description:Inhibition of human DHFR by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-6-phosphate 1-dehydrogenase(Homo sapiens (Human))
Universidade De SãO Paulo

Curated by ChEMBL
LigandPNGBDBM50223368(3beta-hydroxyandrost-5-en-17-one | CHEMBL90593 | D...)
Affinity DataKi:  6.20E+3nMAssay Description:Inhibition of human G6PDH using NADP as substrate by Lineweaver-Burk plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-6-phosphate 1-dehydrogenase(Homo sapiens (Human))
Universidade De SãO Paulo

Curated by ChEMBL
LigandPNGBDBM50223368(3beta-hydroxyandrost-5-en-17-one | CHEMBL90593 | D...)
Affinity DataKi:  8.90E+3nMAssay Description:Inhibition of human G6PDH using glucose-6-phosphate as substrate by Lineweaver-Burk plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398395(CHEMBL1232399)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of human DHFR by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398393(CHEMBL2178599)
Affinity DataKi:  1.54E+4nMAssay Description:Inhibition of human DHFR by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-bisphosphate aldolase, glycosomal(Trypanosoma brucei brucei)
Université

Curated by ChEMBL
LigandPNGBDBM50183272(5-formyl-6-hydroxy-2-naphthyl di-sodium phosphate ...)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibition of Trypanosoma brucei class1 AldolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Universita` Degli Studi Di Sassari

Curated by ChEMBL
LigandPNGBDBM50398391(CHEMBL2178602)
Affinity DataKi:  6.40E+4nMAssay Description:Inhibition of human TS by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma brucei)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446088(CHEMBL3108870)
Affinity DataIC50:  15nMAssay Description:Inhibition of Trypanosoma brucei PFK-mediated ADP production using ATP/fructose-6-phosphate as substrate by luciferase based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma brucei)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446090(CHEMBL3108868)
Affinity DataIC50:  24nMAssay Description:Inhibition of Trypanosoma brucei PFK-mediated ADP production using ATP/fructose-6-phosphate as substrate by luciferase based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma cruzi)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446091(CHEMBL3108867)
Affinity DataIC50:  41nMAssay Description:Inhibition of Trypanosoma cruzi PFKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma cruzi)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446089(CHEMBL3108869)
Affinity DataIC50:  52nMAssay Description:Inhibition of Trypanosoma cruzi PFKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma brucei)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446091(CHEMBL3108867)
Affinity DataIC50:  79nMAssay Description:Inhibition of Trypanosoma brucei PFK-mediated ADP production using ATP/fructose-6-phosphate as substrate by luciferase based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma brucei)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446089(CHEMBL3108869)
Affinity DataIC50:  112nMAssay Description:Inhibition of Trypanosoma brucei PFK-mediated ADP production using ATP/fructose-6-phosphate as substrate by luciferase based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma cruzi)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446090(CHEMBL3108868)
Affinity DataIC50:  120nMAssay Description:Inhibition of Trypanosoma cruzi PFKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma cruzi)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446100(CHEMBL3108858)
Affinity DataIC50:  130nMAssay Description:Inhibition of Trypanosoma cruzi PFKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma brucei)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446095(CHEMBL3108863)
Affinity DataIC50:  160nMAssay Description:Inhibition of Trypanosoma brucei PFK-mediated ADP production using ATP/fructose-6-phosphate as substrate by luciferase based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma cruzi)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446088(CHEMBL3108870)
Affinity DataIC50:  172nMAssay Description:Inhibition of Trypanosoma cruzi PFKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma cruzi)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446129(CHEMBL1394402)
Affinity DataIC50:  230nMAssay Description:Inhibition of Trypanosoma cruzi PFKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma brucei)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446097(CHEMBL3108861)
Affinity DataIC50:  260nMAssay Description:Inhibition of Trypanosoma brucei PFK-mediated ADP production using ATP/fructose-6-phosphate as substrate by luciferase based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma cruzi)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446095(CHEMBL3108863)
Affinity DataIC50:  290nMAssay Description:Inhibition of Trypanosoma cruzi PFKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlyceraldehyde-3-phosphate dehydrogenase(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50030947(CHEMBL331845 | N-[2-(6-Amino-purin-9-yl)-4-hydroxy...)
Affinity DataIC50:  300nMAssay Description:Tested for the inhibitory activity against Glycosomal glyceraldehyde 3-phosphate dehydrogenase (gGAPDH) of Leishmania mexicanaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma brucei)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446100(CHEMBL3108858)
Affinity DataIC50:  370nMAssay Description:Inhibition of Trypanosoma brucei PFK-mediated ADP production using ATP/fructose-6-phosphate as substrate by luciferase based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma brucei)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446129(CHEMBL1394402)
Affinity DataIC50:  410nMAssay Description:Inhibition of Trypanosoma brucei PFK-mediated ADP production using ATP/fructose-6-phosphate as substrate by luciferase based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma cruzi)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446111(CHEMBL3108848)
Affinity DataIC50:  460nMAssay Description:Inhibition of Trypanosoma cruzi PFKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma cruzi)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446102(CHEMBL3108856)
Affinity DataIC50:  460nMAssay Description:Inhibition of Trypanosoma cruzi PFKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlyceraldehyde-3-phosphate dehydrogenase(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50030949((2R,3R,4S,5R)-2-(6-Amino-8-thiophen-2-yl-purin-9-y...)
Affinity DataIC50:  500nMAssay Description:Tested for the inhibitory activity against Glycosomal glyceraldehyde 3-phosphate dehydrogenase (gGAPDH) of Leishmania mexicanaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent 6-phosphofructokinase(Trypanosoma brucei)
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50446099(CHEMBL3108859)
Affinity DataIC50:  520nMAssay Description:Inhibition of Trypanosoma brucei PFK-mediated ADP production using ATP/fructose-6-phosphate as substrate by luciferase based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 154 total ) | Next | Last >>
Jump to: