Compile Data Set for Download or QSAR
maximum 50k data
Found 390 with Last Name = 'mihara' and Initial = 's'
TargetNociceptin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161472(CHEMBL3785095)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in HEK293 cells after 45 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161467(CHEMBL3785560)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in HEK293 cells after 45 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
TargetNociceptin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161471(CHEMBL3785718)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in HEK293 cells after 45 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078977(1-(3-{3-[N'-(4-Hydroxy-phenyl)-guanidino]-2-oxo-2,...)
Affinity DataKi:  2.90nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161400(CHEMBL3785952)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in HEK293 cells after 45 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161399(CHEMBL3786469)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in HEK293 cells after 45 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078965(1-Benzothiazol-6-yl-3-{1-[3-(3-isopropyl-ureido)-b...)
Affinity DataKi:  5.10nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161474(CHEMBL3787174)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in HEK293 cells after 45 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161475(CHEMBL3785605)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in HEK293 cells after 45 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Shionogi

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Shionogi

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]CP55940 from mouse CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50079009(1-(3-{3-[N'-(4-Hydroxy-phenyl)-N''-methyl-guanidin...)
Affinity DataKi:  7.30nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078970(1-(2-Fluoro-phenyl)-3-{1-[3-(3-isopropyl-ureido)-b...)
Affinity DataKi:  7.60nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50079015(1-(2,4-Difluoro-phenyl)-3-{1-[3-(3-isopropyl-ureid...)
Affinity DataKi:  7.80nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50079016(1-Benzofuran-6-yl-3-{1-[3-(3-isopropyl-ureido)-ben...)
Affinity DataKi:  7.80nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50079012(1-Benzo[b]thiophen-6-yl-3-{1-[3-(3-isopropyl-ureid...)
Affinity DataKi:  7.80nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161402(CHEMBL3786899)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in HEK293 cells after 45 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213617((Z)-methyl 2-(2-isopropylphenylimino)-5,5-dimethyl...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213617((Z)-methyl 2-(2-isopropylphenylimino)-5,5-dimethyl...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161473(CHEMBL3785728)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in HEK293 cells after 45 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078958(CHEMBL433216 | {3-[2-Oxo-3-(3-phenyl-ureido)-2,3,4...)
Affinity DataKi: >10nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078966(1-Benzo[b]thiophen-5-yl-3-{1-[3-(3-isopropyl-ureid...)
Affinity DataKi:  13nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078974(1-Isopropyl-3-{3-[3-(N'-methyl-N''-phenyl-guanidin...)
Affinity DataKi:  15nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078971(1-Indan-5-yl-3-{1-[3-(3-isopropyl-ureido)-benzyl]-...)
Affinity DataKi:  17nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078994(1-Benzooxazol-5-yl-3-{1-[3-(3-isopropyl-ureido)-be...)
Affinity DataKi:  17nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078993(1-(1H-Indol-5-yl)-3-{1-[3-(3-isopropyl-ureido)-ben...)
Affinity DataKi:  18nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161476(CHEMBL3785839)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in HEK293 cells after 45 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213619((Z)-methyl 2-(2-methoxyphenylimino)-5,5-dimethyl-1...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078981(1-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-{1-[3-(3-i...)
Affinity DataKi:  18nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161403(CHEMBL3786338)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in HEK293 cells after 45 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213634((Z)-methyl 2-(4-isopropylphenylimino)-5,5-dimethyl...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50079017(1-Benzothiazol-5-yl-3-{1-[3-(3-isopropyl-ureido)-b...)
Affinity DataKi:  24nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078995(1-(1,3-Dioxo-2,3-dihydro-1H-isoindol-5-yl)-3-{1-[3...)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078959(1-(1H-Indazol-5-yl)-3-{1-[3-(3-isopropyl-ureido)-b...)
Affinity DataKi:  26nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078975(1-Benzo[1,3]dioxol-5-yl-3-{1-[3-(3-isopropyl-ureid...)
Affinity DataKi:  28nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078985(1-(4-Fluoro-phenyl)-3-{1-[3-(3-isopropyl-ureido)-b...)
Affinity DataKi:  29nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161405(CHEMBL3787051)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]N/OFQ from human NOP receptor expressed in HEK293 cells after 45 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213637((Z)-methyl 2-(3-isopropylphenylimino)-5,5-dimethyl...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213618((Z)-ethyl 2-(2-isopropylphenylimino)-5,5-dimethyl-...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078957(1-(3-{3-[N'-(4-Hydroxy-phenyl)-N''-isopropyl-guani...)
Affinity DataKi:  36nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078979(1-{1-[3-(3-Isopropyl-ureido)-benzyl]-2-oxo-2,3,4,5...)
Affinity DataKi:  43nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213628((Z)-S-ethyl 2-(2-isopropylphenylimino)-5,5-dimethy...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161475(CHEMBL3785605)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHOK1 cells after 45 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213648((Z)-methyl 2-(2-ethylphenylimino)-5,5-dimethyl-1,3...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50079013(1-{1-[3-(3-Isopropyl-ureido)-benzyl]-2-oxo-2,3,4,5...)
Affinity DataKi:  56nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50078972(1-{1-[3-(3-Isopropyl-ureido)-benzyl]-2-oxo-1,2,3,4...)
Affinity DataKi:  56nMAssay Description:In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213627((Z)-methyl 5,5-dimethyl-2-(2-propylphenylimino)-1,...)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161403(CHEMBL3786338)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHOK1 cells after 45 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 390 total ) | Next | Last >>
Jump to: