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Found 3369 with Last Name = 'mills' and Initial = 'sg'
TargetSomatostatin receptor type 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50389603(CHEMBL2069499)
Affinity DataKi:  0.640nMAssay Description:Displacement of [125I]SS-14 from human SST3 receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288674(CHEMBL420674 | [4-(1,3-Dioxo-1,3-dihydro-isoindol-...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50088301((E)-N,N-dimethyl-N-(4-(2-p-tolyl-6,7-dihydro-5H-be...)
Affinity DataKi:  1.40nMAssay Description:Inhibitory activity of the compound against specific binding of [125I]-MIP-1 alpha to human CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50389592(CHEMBL2069500)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to human SST3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288673(CHEMBL264455 | {4-[((S)-1-Benzoyl-pyrrolidine-2-ca...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of gelatinase-A (MMP-2).More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288672(CHEMBL113362 | [4-(1,3-Dioxo-1,3-dihydro-isoindol-...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of gelatinase-A (MMP-2).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288683(CHEMBL109438 | [4-(1,3-Dioxo-1,3-dihydro-isoindol-...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277511(3-[(3aR,4R,5S,7aS)-5-{(1R)-1-[3,5-Bis(trifluoromet...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity to human NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277511(3-[(3aR,4R,5S,7aS)-5-{(1R)-1-[3,5-Bis(trifluoromet...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity to human NK3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288672(CHEMBL113362 | [4-(1,3-Dioxo-1,3-dihydro-isoindol-...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288677(CHEMBL324691 | [(E)-4-(1,3-Dioxo-1,3-dihydro-isoin...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288677(CHEMBL324691 | [(E)-4-(1,3-Dioxo-1,3-dihydro-isoin...)
Affinity DataKi:  4.80nMAssay Description:Inhibition of gelatinase-A (MMP-2).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288678(CHEMBL320968 | [(S)-2-((S)-3-Methyl-1-phenylcarbam...)
Affinity DataKi:  5.5nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288681((4-Benzoylamino-butyl)-[(S)-2-((S)-3-methyl-1-phen...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288687(CHEMBL111975 | {4-[((S)-1-Acetyl-pyrrolidine-2-car...)
Affinity DataKi:  6.10nMAssay Description:Inhibition of gelatinase-A (MMP-2).More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288678(CHEMBL320968 | [(S)-2-((S)-3-Methyl-1-phenylcarbam...)
Affinity DataKi:  7.30nMAssay Description:Inhibition of gelatinase-A (MMP-2).More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288683(CHEMBL109438 | [4-(1,3-Dioxo-1,3-dihydro-isoindol-...)
Affinity DataKi:  12nMAssay Description:Inhibition of gelatinase-A (MMP-2).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288673(CHEMBL264455 | {4-[((S)-1-Benzoyl-pyrrolidine-2-ca...)
Affinity DataKi:  13nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288699((4-Ethoxycarbonylamino-butyl)-[(S)-2-((S)-3-methyl...)
Affinity DataKi:  16nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288668(CHEMBL109829 | [4-(3-Ethyl-ureido)-butyl]-[(S)-2-(...)
Affinity DataKi:  17nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288668(CHEMBL109829 | [4-(3-Ethyl-ureido)-butyl]-[(S)-2-(...)
Affinity DataKi:  19nMAssay Description:Inhibition of gelatinase-A (MMP-2)More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288674(CHEMBL420674 | [4-(1,3-Dioxo-1,3-dihydro-isoindol-...)
Affinity DataKi:  20nMAssay Description:Inhibition of gelatinase-A (MMP-2).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288682(CHEMBL110991 | {4-[((R)-1-Benzoyl-pyrrolidine-2-ca...)
Affinity DataKi:  24nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288675(CHEMBL113234 | {4-[((R)-1-Acetyl-pyrrolidine-2-car...)
Affinity DataKi:  26nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288681((4-Benzoylamino-butyl)-[(S)-2-((S)-3-methyl-1-phen...)
Affinity DataKi:  26nMAssay Description:Inhibition of gelatinase-A (MMP-2).More data for this Ligand-Target Pair
In DepthDetails Article
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50187039(1-(3,4-dichlorobenzyl)-5-hydroxy-1H-indole-2-carbo...)
Affinity DataKi:  29nMAssay Description:Displacement of [125I]MCP1 from human CCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288679(CHEMBL325835 | [(S)-2-((S)-3-Methyl-1-phenylcarbam...)
Affinity DataKi:  30nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288684(CHEMBL324004 | [4-(3-Benzyl-ureido)-butyl]-[(S)-2-...)
Affinity DataKi:  50nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50091438((E)-3-(3,4-Dichloro-phenyl)-N-{5-[4-(5-hydroxy-1H-...)
Affinity DataKi:  50nMAssay Description:Displacement of [125I]MCP1 from human CCR2 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288693((4-Methoxycarbonylamino-butyl)-[(S)-2-((S)-3-methy...)
Affinity DataKi:  54nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288694(CHEMBL322142 | [(S)-2-((S)-3-Methyl-1-phenylcarbam...)
Affinity DataKi:  56nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288687(CHEMBL111975 | {4-[((S)-1-Acetyl-pyrrolidine-2-car...)
Affinity DataKi:  62nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288695((4-Benzyloxycarbonylamino-butyl)-[(S)-2-((S)-3-met...)
Affinity DataKi:  63nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288685(CHEMBL110253 | [(S)-2-((S)-3-Methyl-1-phenylcarbam...)
Affinity DataKi:  70nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288690(CHEMBL109670 | [(S)-2-((S)-3-Methyl-1-phenylcarbam...)
Affinity DataKi:  130nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288679(CHEMBL325835 | [(S)-2-((S)-3-Methyl-1-phenylcarbam...)
Affinity DataKi:  130nMAssay Description:Inhibition of gelatinase-A (MMP-2).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288669(CHEMBL109671 | [(S)-2-((S)-3-Methyl-1-phenylcarbam...)
Affinity DataKi:  170nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50141931((R)-[(2S,3S)-3-[4-(5-Biphenyl-4-ylmethyl-2-ethyl-2...)
Affinity DataKi:  400nMAssay Description:Binding affinity against hERG Voltage-gated potassium channel subunit Kv11.1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288698(CHEMBL112724 | {[2-(1,3-Dioxo-1,3-dihydro-isoindol...)
Affinity DataKi:  410nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288691(CHEMBL111601 | [4-(1,3-Dioxo-1,3-dihydro-isoindol-...)
Affinity DataKi:  440nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288696(CHEMBL110075 | [(S)-2-((S)-3-Methyl-1-phenylcarbam...)
Affinity DataKi:  470nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288676(3-{Hydroxy-[(S)-2-((S)-3-methyl-1-phenylcarbamoyl-...)
Affinity DataKi:  520nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288697((2-Benzylcarbamoyl-ethyl)-[(S)-2-((S)-3-methyl-1-p...)
Affinity DataKi:  540nMAssay Description:Inhibition of stromelysin-1 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288680(CHEMBL326018 | Methyl-[(S)-2-((S)-3-methyl-1-pheny...)
Affinity DataKi:  570nMAssay Description:Inhibition of gelatinase-A (MMP-2).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288671(CHEMBL110997 | [(S)-2-((S)-3-Methyl-1-phenylcarbam...)
Affinity DataKi:  670nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50141911((R)-2-[(2S,3S)-3-{4-[5-(4-Cyano-benzyl)-2-ethyl-2H...)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity against hERG Voltage-gated potassium channel subunit Kv11.1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288676(3-{Hydroxy-[(S)-2-((S)-3-methyl-1-phenylcarbamoyl-...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of gelatinase-A (MMP-2).More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288680(CHEMBL326018 | Methyl-[(S)-2-((S)-3-methyl-1-pheny...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of stromelysin-1 (MMP-3).More data for this Ligand-Target Pair
In DepthDetails Article
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50141908((R)-2-[(2S,3S)-3-{4-[5-(4-tert-Butyl-benzyl)-2-eth...)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity against hERG Voltage-gated potassium channel subunit Kv11.1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50141905((R)-2-[(2S,3S)-3-[4-(5-Biphenyl-4-ylmethyl-2-ethyl...)
Affinity DataKi:  2.30E+3nMAssay Description:Binding affinity against hERG Voltage-gated potassium channel subunit Kv11.1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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