TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 0.178nMAssay Description:Displacement of [3H]mepyramine from human H1R expressed in HEK293T cell homogenates incubated for 1 hr by radioligand binding assay based liquid scin...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3H]mepyramine from human H1R expressed in HEK293T cells by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 89nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 89nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 126nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 126nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 151nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 151nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 174nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 174nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 186nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 186nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 309nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 309nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 339nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 339nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 372nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 372nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 407nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 407nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 437nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 437nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 437nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 437nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 501nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 501nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 513nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 513nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 550nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 550nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 562nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 562nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 692nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 692nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 794nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 794nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 832nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 832nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 912nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 912nMAssay Description:Displacement of fluorophore-labeled mepyramine from Nluc-tagged human H1R expressed in HEK293T cells incubated for 2 hrs by NanoBRET competition bind...More data for this Ligand-Target Pair